KR20240111787A - 신경학적 질환의 치료를 위한 설폰아미드 화합물 - Google Patents

신경학적 질환의 치료를 위한 설폰아미드 화합물 Download PDF

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KR20240111787A
KR20240111787A KR1020247020803A KR20247020803A KR20240111787A KR 20240111787 A KR20240111787 A KR 20240111787A KR 1020247020803 A KR1020247020803 A KR 1020247020803A KR 20247020803 A KR20247020803 A KR 20247020803A KR 20240111787 A KR20240111787 A KR 20240111787A
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compound
ring
alkyl
formula
pharmaceutically acceptable
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헤닝 슈타인하겐
파올로 페바레로
마리아 피아 카탈라니
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라리오 테라퓨틱스 리미티드
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Publication of KR20240111787A publication Critical patent/KR20240111787A/ko
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    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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