KR20100075679A - 트랜스-ｎ-이소부틸-3-플루오로-3-[3-플루오로-4-(피롤리딘-1-일메틸)-페닐]-사이클로부탄카복스아미드의 토실레이트 염 - Google Patents
트랜스-ｎ-이소부틸-3-플루오로-3-[3-플루오로-4-(피롤리딘-1-일메틸)-페닐]-사이클로부탄카복스아미드의 토실레이트 염 Download PDFInfo
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- KR20100075679A KR20100075679A KR1020107012321A KR20107012321A KR20100075679A KR 20100075679 A KR20100075679 A KR 20100075679A KR 1020107012321 A KR1020107012321 A KR 1020107012321A KR 20107012321 A KR20107012321 A KR 20107012321A KR 20100075679 A KR20100075679 A KR 20100075679A
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Classifications
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- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/06—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by halogen atoms or nitro radicals
- C07D295/073—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by halogen atoms or nitro radicals with the ring nitrogen atoms and the substituents separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
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Landscapes
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- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
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| US569607P | 2007-12-07 | 2007-12-07 | |
| US61/005,696 | 2007-12-07 |
Publications (1)
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| KR20100075679A true KR20100075679A (ko) | 2010-07-02 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| KR1020107012321A Abandoned KR20100075679A (ko) | 2007-12-07 | 2008-12-04 | 트랜스-ｎ-이소부틸-3-플루오로-3-[3-플루오로-4-(피롤리딘-1-일메틸)-페닐]-사이클로부탄카복스아미드의 토실레이트 염 |
Country Status (15)
| Country | Link |
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| US (1) | US8178574B2 (https=) |
| EP (1) | EP2231630B1 (https=) |
| JP (1) | JP4566259B2 (https=) |
| KR (1) | KR20100075679A (https=) |
| CN (1) | CN101939306A (https=) |
| AR (1) | AR069611A1 (https=) |
| AU (1) | AU2008332880C1 (https=) |
| CA (1) | CA2708043C (https=) |
| IL (1) | IL205963A0 (https=) |
| MX (1) | MX2010006162A (https=) |
| NZ (1) | NZ585671A (https=) |
| RU (1) | RU2451016C2 (https=) |
| TW (1) | TW200932213A (https=) |
| WO (1) | WO2009071988A1 (https=) |
| ZA (1) | ZA201004768B (https=) |
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| EP2124933B1 (en) | 2007-01-22 | 2012-10-17 | Pfizer Products Inc. | Tosylate salt of a therapeutic compound and pharmaceutical compositions thereof |
| WO2013151982A1 (en) | 2012-04-03 | 2013-10-10 | Arena Pharmaceuticals, Inc. | Methods and compounds useful in treating pruritus, and methods for identifying such compounds |
| US20140206667A1 (en) | 2012-11-14 | 2014-07-24 | Michela Gallagher | Methods and compositions for treating schizophrenia |
| AR103406A1 (es) * | 2015-01-30 | 2017-05-10 | Lilly Co Eli | Sal de tosilato |
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| US5498626A (en) * | 1992-04-10 | 1996-03-12 | Pfizer Inc. | Acylaminoindole derivatives as 5-ht1 agonists |
| US8158673B2 (en) * | 2005-10-27 | 2012-04-17 | Pfizer Inc. | Histamine-3 receptor antagonists |
| EP2124933B1 (en) * | 2007-01-22 | 2012-10-17 | Pfizer Products Inc. | Tosylate salt of a therapeutic compound and pharmaceutical compositions thereof |
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2010
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- 2010-07-06 ZA ZA2010/04768A patent/ZA201004768B/en unknown
Also Published As
| Publication number | Publication date |
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| IL205963A0 (en) | 2010-11-30 |
| AR069611A1 (es) | 2010-02-03 |
| NZ585671A (en) | 2012-06-29 |
| CA2708043A1 (en) | 2009-06-11 |
| RU2010122972A (ru) | 2011-12-10 |
| WO2009071988A1 (en) | 2009-06-11 |
| AU2008332880C1 (en) | 2012-07-19 |
| EP2231630B1 (en) | 2012-11-07 |
| CN101939306A (zh) | 2011-01-05 |
| JP2009161517A (ja) | 2009-07-23 |
| CA2708043C (en) | 2012-11-13 |
| ZA201004768B (en) | 2011-03-30 |
| AU2008332880A1 (en) | 2009-06-11 |
| AU2008332880B2 (en) | 2012-01-19 |
| TW200932213A (en) | 2009-08-01 |
| JP4566259B2 (ja) | 2010-10-20 |
| US20100256213A1 (en) | 2010-10-07 |
| US8178574B2 (en) | 2012-05-15 |
| MX2010006162A (es) | 2010-06-25 |
| RU2451016C2 (ru) | 2012-05-20 |
| EP2231630A1 (en) | 2010-09-29 |
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