KR101516606B1 - 4-아미노부트-2-에놀라이드의 제조방법 - Google Patents
4-아미노부트-2-에놀라이드의 제조방법 Download PDFInfo
- Publication number
- KR101516606B1 KR101516606B1 KR1020107007178A KR20107007178A KR101516606B1 KR 101516606 B1 KR101516606 B1 KR 101516606B1 KR 1020107007178 A KR1020107007178 A KR 1020107007178A KR 20107007178 A KR20107007178 A KR 20107007178A KR 101516606 B1 KR101516606 B1 KR 101516606B1
- Authority
- KR
- South Korea
- Prior art keywords
- alkyl
- formula
- aryl
- compound
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Links
- 0 *C(C(C(OC1)=O)=C1N=O)=O Chemical compound *C(C(C(OC1)=O)=C1N=O)=O 0.000 description 2
- NXSHHTJWIOPOBF-UHFFFAOYSA-N CCOC(C(C(OC1)=O)=C1O)=O Chemical compound CCOC(C(C(OC1)=O)=C1O)=O NXSHHTJWIOPOBF-UHFFFAOYSA-N 0.000 description 1
- FXXCNSJWPDVASC-UHFFFAOYSA-N CCOC(C(C([O]=C1)=O)=C1O)=O Chemical compound CCOC(C(C([O]=C1)=O)=C1O)=O FXXCNSJWPDVASC-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07116639.1 | 2007-09-18 | ||
| EP07116639A EP2042496A1 (de) | 2007-09-18 | 2007-09-18 | Verfahren zur Herstellung von 4-Aminobut-2-enoliden |
| PCT/EP2008/007270 WO2009036899A1 (de) | 2007-09-18 | 2008-09-05 | Verfahren zur herstellung von 4-aminobut-2-enoliden |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| KR20100061826A KR20100061826A (ko) | 2010-06-09 |
| KR101516606B1 true KR101516606B1 (ko) | 2015-04-30 |
Family
ID=39167552
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020107007178A Active KR101516606B1 (ko) | 2007-09-18 | 2008-09-05 | 4-아미노부트-2-에놀라이드의 제조방법 |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US8273904B2 (https=) |
| EP (2) | EP2042496A1 (https=) |
| JP (1) | JP5611043B2 (https=) |
| KR (1) | KR101516606B1 (https=) |
| CN (2) | CN102775305A (https=) |
| BR (1) | BRPI0816911B1 (https=) |
| DK (1) | DK2193128T3 (https=) |
| ES (1) | ES2612058T3 (https=) |
| IL (1) | IL203761A (https=) |
| MX (1) | MX2010001963A (https=) |
| TW (1) | TWI432419B (https=) |
| WO (1) | WO2009036899A1 (https=) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2230237A1 (de) | 2009-03-16 | 2010-09-22 | Bayer CropScience AG | Neues Verfahren zur Herstellung von Enaminocarbonyl-Verbindungen |
| EP2230236A1 (de) | 2009-03-16 | 2010-09-22 | Bayer CropScience AG | Neues Verfahren zur Herstellung von Enaminocarbonyl-Verbindungen |
| MX2012001675A (es) | 2009-08-11 | 2012-03-06 | Bayer Cropscience Ag | Procedimiento para preparar 2,4-dioxotetrahidrofuran-3-carboxilato s. |
| TW201111370A (en) | 2009-08-18 | 2011-04-01 | Bayer Cropscience Ag | Novel process for the preparation of 4-aminobut-2-enolides |
| EP2493881A1 (de) * | 2009-10-26 | 2012-09-05 | Bayer CropScience AG | Neue feste form von 4-[[(6-chlorpyridin-3-yl)methyl](2,2-difluorethyl)amino]furan-2(5h)-on |
| WO2011051241A1 (de) | 2009-10-27 | 2011-05-05 | Bayer Technology Services Gmbh | Co-kristall von 4-{[(6-chlorpyrid-3yl)methyl](2,2-difluorethyl)amino}furan-2(5h)-on mit oxalsäure und dessen verwendung als pestizid |
| US20120283294A1 (en) | 2009-10-27 | 2012-11-08 | Bayer Technology Services Gmbh | Co-crystal of 4-furan-2(5h)-one with benzoic acid and use thereof as pesticide |
| WO2011051242A1 (de) | 2009-10-27 | 2011-05-05 | Bayer Technology Services Gmbh | Co-kristall von 4- { [ (6-chlorpyrid-3-yl) methyl] (2,2-difluorethyl) amino} furan-2 (5h) -on mit salizylsäure und dessen verwendung als pestizid |
| WO2011076715A1 (de) * | 2009-12-23 | 2011-06-30 | Bayer Cropscience Ag | Neues verfahren zur herstellung von 4-aminobut-2-enoliden ausgehend von 4-alkoxyfuran-2(5h)-on oder 4-arylalkoxyfuran-2-(5h)-on |
| BR112013014270A2 (pt) * | 2010-12-09 | 2017-10-24 | Bayer Ip Gmbh | misturas inseticidas com propriedades aperfeiçoadas |
| US20130317067A1 (en) * | 2010-12-09 | 2013-11-28 | Bayer Intellectual Property Gmbh | Pesticidal mixtures with improved properties |
| JP5970002B2 (ja) * | 2011-03-03 | 2016-08-17 | バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH | 4−ヒドロキシ−2−オキソ−2,5−ジヒドロフラン−3−カルボン酸化合物のナトリウム塩またはカリウム塩の製造方法 |
| DK2880022T3 (en) * | 2012-08-01 | 2016-08-15 | Bayer Cropscience Ag | MULTI-STEP PROCEDURE FOR PREPARING ALKALIMETAL SALTS OF SPECIAL 4-HYDROXY-2-OXO-2,5-DIHYDROFURAN-3-CARBOXYL ACID ESTERS |
| CN105503708B (zh) * | 2016-01-26 | 2018-05-29 | 南开大学 | 一类含二氟乙基的杂环化合物及其制备方法和用途 |
| EP4295683A1 (en) | 2022-06-21 | 2023-12-27 | Bayer Aktiengesellschaft | Agrochemical formulations comprising crystalline form a of 4-[(6-chloro-3-pyridylmethyl)(2,2-difluoroethyl)amino]furan-2(5h)-one |
| KR20250020435A (ko) | 2022-06-06 | 2025-02-11 | 바이엘 악티엔게젤샤프트 | 4-[(6-클로로-3-피리딜메틸)(2,2-디플루오로에틸)아미노]푸란-2(5h)-온의결정질 형태 a를 포함하는 농약 제제 |
| WO2025114238A1 (en) | 2023-12-01 | 2025-06-05 | Bayer Aktiengesellschaft | Solid agrochemical formulations comprising crystalline form a of 4-[(6-chloro-3-pyridylmethyl)(2,2- difluoroethyl)amino]furan-2(5h)-one |
| WO2025119860A1 (en) | 2023-12-05 | 2025-06-12 | Bayer Aktiengesellschaft | Liquid agrochemical formulations comprising flupyradifurone |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0539588A1 (en) * | 1990-07-05 | 1993-05-05 | Nippon Soda Co., Ltd. | Amine derivative |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH503722A (de) | 1969-05-28 | 1971-02-28 | Lonza Ag | Verfahren zur Herstellung von Tetronsäure |
| DE3311003A1 (de) | 1983-03-25 | 1984-09-27 | Bayer Ag, 5090 Leverkusen | Chromon- und thiochromonsubstituierte 1,4-dihydropyridinlactone, mehrere verfahren zu ihrer herstellung und ihre verwendung in arzneimitteln |
| CH658056A5 (de) | 1984-02-09 | 1986-10-15 | Lonza Ag | Verfahren zur herstellung von tetronsaeure. |
| US5010176A (en) | 1988-11-10 | 1991-04-23 | Eli Lilly And Company | Antibody-drug conjugates |
| JPH054966A (ja) * | 1990-07-05 | 1993-01-14 | Nippon Soda Co Ltd | アミン誘導体、その製法及び殺虫剤 |
| DE102006015467A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
| DE102006015470A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
| DE102006015468A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
| CN1974532B (zh) * | 2006-12-13 | 2010-12-29 | 井冈山学院 | 羧酸二异丙基二乙基酯的制备方法及其应用 |
-
2007
- 2007-09-18 EP EP07116639A patent/EP2042496A1/de not_active Ceased
-
2008
- 2008-09-05 WO PCT/EP2008/007270 patent/WO2009036899A1/de not_active Ceased
- 2008-09-05 DK DK08801865.0T patent/DK2193128T3/en active
- 2008-09-05 MX MX2010001963A patent/MX2010001963A/es active IP Right Grant
- 2008-09-05 BR BRPI0816911-0A patent/BRPI0816911B1/pt active IP Right Grant
- 2008-09-05 EP EP08801865.0A patent/EP2193128B1/de active Active
- 2008-09-05 ES ES08801865.0T patent/ES2612058T3/es active Active
- 2008-09-05 KR KR1020107007178A patent/KR101516606B1/ko active Active
- 2008-09-05 US US12/677,769 patent/US8273904B2/en active Active
- 2008-09-05 CN CN2012102326181A patent/CN102775305A/zh active Pending
- 2008-09-05 CN CN200880107465XA patent/CN101801948B/zh active Active
- 2008-09-05 JP JP2010525229A patent/JP5611043B2/ja active Active
- 2008-09-17 TW TW097135546A patent/TWI432419B/zh active
-
2010
- 2010-02-07 IL IL203761A patent/IL203761A/en active IP Right Grant
-
2012
- 2012-08-22 US US13/591,431 patent/US9550745B2/en active Active
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0539588A1 (en) * | 1990-07-05 | 1993-05-05 | Nippon Soda Co., Ltd. | Amine derivative |
Non-Patent Citations (4)
| Title |
|---|
| A. C. CAMPBELL et al, J. CHEM. SOC. PERKIN TRANS 1, 1985, pp. 1567-1576 * |
| A. C. CAMPBELL et al, J. CHEM. SOC. PERKIN TRANS 1, 1985, pp. 1567-1576* |
| T. P. C. MULHOLLAND et al, J. CHEM. SOC. PERKIN TRANS 1, 1972, pp. 1225-1231 * |
| T. P. C. MULHOLLAND et al, J. CHEM. SOC. PERKIN TRANS 1, 1972, pp. 1225-1231* |
Also Published As
| Publication number | Publication date |
|---|---|
| DK2193128T3 (en) | 2017-01-30 |
| MX2010001963A (es) | 2010-03-10 |
| EP2193128B1 (de) | 2016-10-26 |
| JP2011500513A (ja) | 2011-01-06 |
| BRPI0816911A2 (pt) | 2015-03-17 |
| EP2193128A1 (de) | 2010-06-09 |
| WO2009036899A1 (de) | 2009-03-26 |
| US9550745B2 (en) | 2017-01-24 |
| EP2042496A1 (de) | 2009-04-01 |
| US8273904B2 (en) | 2012-09-25 |
| US20120323023A1 (en) | 2012-12-20 |
| BRPI0816911B1 (pt) | 2022-04-12 |
| TWI432419B (zh) | 2014-04-01 |
| CN102775305A (zh) | 2012-11-14 |
| ES2612058T3 (es) | 2017-05-11 |
| TW200920741A (en) | 2009-05-16 |
| CN101801948A (zh) | 2010-08-11 |
| BRPI0816911A8 (pt) | 2015-10-27 |
| US20100190990A1 (en) | 2010-07-29 |
| IL203761A (en) | 2015-09-24 |
| KR20100061826A (ko) | 2010-06-09 |
| JP5611043B2 (ja) | 2014-10-22 |
| CN101801948B (zh) | 2013-10-30 |
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