KR100432303B1 - 레조르시놀 유도체의 제조방법 - Google Patents

레조르시놀 유도체의 제조방법 Download PDF

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Publication number
KR100432303B1
KR100432303B1 KR10-2001-0013250A KR20010013250A KR100432303B1 KR 100432303 B1 KR100432303 B1 KR 100432303B1 KR 20010013250 A KR20010013250 A KR 20010013250A KR 100432303 B1 KR100432303 B1 KR 100432303B1
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KR
South Korea
Prior art keywords
formula
compound
delete delete
alkyl
protecting group
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KR10-2001-0013250A
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English (en)
Korean (ko)
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KR20010096608A (ko
Inventor
브레들리스튜어트에드워드
키친존
윈그라함마이클
Original Assignee
화이자 프로덕츠 인코포레이티드
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Publication of KR20010096608A publication Critical patent/KR20010096608A/ko
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Publication of KR100432303B1 publication Critical patent/KR100432303B1/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C37/00—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom of a six-membered aromatic ring
    • C07C37/06—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom of a six-membered aromatic ring by conversion of non-aromatic six-membered rings or of such rings formed in situ into aromatic six-membered rings, e.g. by dehydrogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/72—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 spiro-condensed with carbocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C37/00—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom of a six-membered aromatic ring
    • C07C37/06—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom of a six-membered aromatic ring by conversion of non-aromatic six-membered rings or of such rings formed in situ into aromatic six-membered rings, e.g. by dehydrogenation
    • C07C37/07—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom of a six-membered aromatic ring by conversion of non-aromatic six-membered rings or of such rings formed in situ into aromatic six-membered rings, e.g. by dehydrogenation with simultaneous reduction of C=O group in that ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/56—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds
    • C07C45/57—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds with oxygen as the only heteroatom
    • C07C45/59—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds with oxygen as the only heteroatom in five-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C07C45/70—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form
    • C07C45/71—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form being hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/703—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups
    • C07C49/747—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/18—Systems containing only non-condensed rings with a ring being at least seven-membered
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S977/00—Nanotechnology
    • Y10S977/902—Specified use of nanostructure
    • Y10S977/904—Specified use of nanostructure for medical, immunological, body treatment, or diagnosis
    • Y10S977/926—Topical chemical, e.g. cosmetic or sunscreen

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
KR10-2001-0013250A 2000-03-15 2001-03-14 레조르시놀 유도체의 제조방법 KR100432303B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US18970400P 2000-03-15 2000-03-15
US60/189,704 2000-03-15

Publications (2)

Publication Number Publication Date
KR20010096608A KR20010096608A (ko) 2001-11-07
KR100432303B1 true KR100432303B1 (ko) 2004-05-20

Family

ID=22698426

Family Applications (1)

Application Number Title Priority Date Filing Date
KR10-2001-0013250A KR100432303B1 (ko) 2000-03-15 2001-03-14 레조르시놀 유도체의 제조방법

Country Status (18)

Country Link
US (3) US6504037B2 (US20070244113A1-20071018-C00087.png)
EP (1) EP1134207A1 (US20070244113A1-20071018-C00087.png)
JP (1) JP2001294549A (US20070244113A1-20071018-C00087.png)
KR (1) KR100432303B1 (US20070244113A1-20071018-C00087.png)
CN (1) CN1325838A (US20070244113A1-20071018-C00087.png)
AR (1) AR030055A1 (US20070244113A1-20071018-C00087.png)
AU (1) AU782397B2 (US20070244113A1-20071018-C00087.png)
BR (1) BR0100982A (US20070244113A1-20071018-C00087.png)
CA (1) CA2340486A1 (US20070244113A1-20071018-C00087.png)
CZ (1) CZ2001930A3 (US20070244113A1-20071018-C00087.png)
HK (1) HK1040987A1 (US20070244113A1-20071018-C00087.png)
ID (1) ID29673A (US20070244113A1-20071018-C00087.png)
IL (1) IL141915A0 (US20070244113A1-20071018-C00087.png)
IN (1) IN192530B (US20070244113A1-20071018-C00087.png)
PL (1) PL346463A1 (US20070244113A1-20071018-C00087.png)
RU (1) RU2213087C2 (US20070244113A1-20071018-C00087.png)
YU (1) YU18601A (US20070244113A1-20071018-C00087.png)
ZA (1) ZA200102070B (US20070244113A1-20071018-C00087.png)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6828460B2 (en) * 1999-03-22 2004-12-07 Pfizer Inc. Resorcinol derivatives
US6863897B2 (en) * 2002-03-22 2005-03-08 Unilever Home & Personal Care Usa, Division Of Conopco, Inc. Stabilization of resorcinol derivatives in cosmetic compositions
JP4228605B2 (ja) 2002-07-02 2009-02-25 住友化学株式会社 改変型還元酵素、その遺伝子及びそれらの利用
JP4228606B2 (ja) 2002-07-03 2009-02-25 住友化学株式会社 改変型還元酵素、その遺伝子及びそれらの利用
US6852310B2 (en) 2002-08-23 2005-02-08 Unilever Home & Personal Care Usa Division Of Conopco, Inc. Skin lightening agents, compositions and methods
US7163327B2 (en) * 2002-12-02 2007-01-16 3M Innovative Properties Company Illumination system using a plurality of light sources
US6875425B2 (en) 2002-12-12 2005-04-05 Unilever Home & Personal Care Usa Skin lightening agents, compositions and methods
US7524485B2 (en) 2002-12-12 2009-04-28 Unilever Home & Personal Care, Usa, Division Of Conopco, Inc. Skin lightening agents, compositions and methods
US7338979B2 (en) 2003-02-11 2008-03-04 Warner-Lambert Company Depigmentation agents
US7300646B2 (en) * 2004-02-27 2007-11-27 Unilever Home & Personal Care Usa, Division Of Conopco, Inc. Skin lightening agents, compositions and methods
US20060062865A1 (en) * 2004-09-17 2006-03-23 Nebojsa Ilic Tyrosinase inhibitor and method for preparation
US20060210498A1 (en) 2005-03-18 2006-09-21 Unilever Home & Personal Care Usa, Division Of Conopco, Inc. Novel resorcinol derivatives for skin
US20060210497A1 (en) * 2005-03-18 2006-09-21 Unilever Home & Personal Care Usa, Division Of Conopco, Inc. Novel resorcinol derivatives
US7270805B1 (en) 2006-03-30 2007-09-18 Conopco, Inc. Skin lightening agents, compositions and methods
US7247294B1 (en) 2006-03-30 2007-07-24 Conopco, Inc. Skin lightening agents, compositions and methods
US7250158B1 (en) 2006-03-30 2007-07-31 Conopco, Inc. Skin lightening agents, compositions and methods
US20140256830A1 (en) 2013-03-08 2014-09-11 Ampere Life Sciences, Inc. Resorcinol compounds for dermatological use
MX369987B (es) 2016-06-15 2019-11-27 Unilever Nv Metodo y composicion cosmetica para un suministro transdermico mejorado de resorcinol alquilo sustituido.
CN111909012B (zh) * 2020-08-24 2022-10-21 浙江工业大学台州研究院 一种高选择性、高转化制备1,3-环己二酮的方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PA8469601A1 (es) * 1998-04-10 2000-09-29 Pfizer Prod Inc Procedimiento para alquilar sulfonamidas impedidas estericamente
CA2362698C (en) * 1999-03-22 2005-02-01 Pfizer Inc. Resorcinol derivatives

Also Published As

Publication number Publication date
ID29673A (id) 2001-09-20
US6861564B2 (en) 2005-03-01
US20020032352A1 (en) 2002-03-14
KR20010096608A (ko) 2001-11-07
CZ2001930A3 (cs) 2001-10-17
JP2001294549A (ja) 2001-10-23
BR0100982A (pt) 2001-12-04
EP1134207A1 (en) 2001-09-19
US20030088113A1 (en) 2003-05-08
CN1325838A (zh) 2001-12-12
RU2213087C2 (ru) 2003-09-27
YU18601A (sh) 2003-07-07
CA2340486A1 (en) 2001-09-15
ZA200102070B (en) 2002-09-13
IL141915A0 (en) 2002-03-10
AR030055A1 (es) 2003-08-13
US6504037B2 (en) 2003-01-07
AU782397B2 (en) 2005-07-21
IN192530B (US20070244113A1-20071018-C00087.png) 2004-04-24
PL346463A1 (en) 2001-09-24
HK1040987A1 (zh) 2002-06-28
US20050143594A1 (en) 2005-06-30
AU2647701A (en) 2001-09-20

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