JPS6442488A - Production of 7-acylaminodeacetoxycephalosporanic acid or ester thereof - Google Patents
Production of 7-acylaminodeacetoxycephalosporanic acid or ester thereofInfo
- Publication number
- JPS6442488A JPS6442488A JP20039887A JP20039887A JPS6442488A JP S6442488 A JPS6442488 A JP S6442488A JP 20039887 A JP20039887 A JP 20039887A JP 20039887 A JP20039887 A JP 20039887A JP S6442488 A JPS6442488 A JP S6442488A
- Authority
- JP
- Japan
- Prior art keywords
- acid
- coor
- formula
- nitrogen atom
- butyl acetate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Cephalosporin Compounds (AREA)
Abstract
PURPOSE:To industrially and advantageously obtain the titled compound useful as a starting raw material for an intermediate of an antibacterial agent, by heating esters of an acylamidopenicillanic acid sulfoxide in butyl acetate in the presence of a base containing both acid and nitrogen atom. CONSTITUTION:Esters (example; 2,2,2-trichloroethyl 6-phenylacetamidopenici llanate) of a 6-acylamidopenicillanic acid sulfoxide expressed by formula I (R<1> represents phenylacetyl or phenoxyacetyl; -COOR<2> represents esterified carboxyl) are heated in butyl acetate in the presence of a base containing both acid and nitrogen atom (example. pyridine trichloroethylphosphate) up to 130 deg.C at the highest, and, as necessary, followed by esterification to afford the aimed compound expressed by formula II (COOR represents carboxyl or esterified carboxyl).
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP20039887A JPS6442488A (en) | 1987-08-11 | 1987-08-11 | Production of 7-acylaminodeacetoxycephalosporanic acid or ester thereof |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP20039887A JPS6442488A (en) | 1987-08-11 | 1987-08-11 | Production of 7-acylaminodeacetoxycephalosporanic acid or ester thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS6442488A true JPS6442488A (en) | 1989-02-14 |
Family
ID=16423658
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP20039887A Pending JPS6442488A (en) | 1987-08-11 | 1987-08-11 | Production of 7-acylaminodeacetoxycephalosporanic acid or ester thereof |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS6442488A (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102584853A (en) * | 2011-12-14 | 2012-07-18 | 伊犁川宁生物技术有限公司 | Preparation method of 7-aminodeacetoxy cephalosporanic acid |
-
1987
- 1987-08-11 JP JP20039887A patent/JPS6442488A/en active Pending
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102584853A (en) * | 2011-12-14 | 2012-07-18 | 伊犁川宁生物技术有限公司 | Preparation method of 7-aminodeacetoxy cephalosporanic acid |
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