JPS5718664A - N-substituted-bicyclo- 2.2.1 -hept-5-ene-2,3-dicarboximide derivative - Google Patents
N-substituted-bicyclo- 2.2.1 -hept-5-ene-2,3-dicarboximide derivativeInfo
- Publication number
- JPS5718664A JPS5718664A JP9369080A JP9369080A JPS5718664A JP S5718664 A JPS5718664 A JP S5718664A JP 9369080 A JP9369080 A JP 9369080A JP 9369080 A JP9369080 A JP 9369080A JP S5718664 A JPS5718664 A JP S5718664A
- Authority
- JP
- Japan
- Prior art keywords
- hept
- bicyclo
- ene
- bond
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
Abstract
NEW MATERIAL:An N-substituted-bicyclo-[2.2.1]-hept-5-ene-2,3-dicarboximide derivative expressed by formula I (n is 4W6; the bond between the 5- and the 6- positions represents a double bond).
EXAMPLE: N-(1-Hydroxycyclopentylmethyl)-bicyclo-[2.2.1]-hept-5-ene-2,3-dicarboximide.
USE: A remedy for cholecystitis, cholangitis, cholecystolithiasis and bile duct dyskinesia having improved cholagogic action.
PROCESS: A bicyclo-[2.2.1]-hept-5-ene-2,3-dicarboxylic anhydride expressed by formula II is refluxed with 1-aminomethylcyclopentanol hydrochloride, etc. in the presence of an organic base, e.g. triethylamine, in an organic solvent for several hours under heating to give the compound expressed by formula I in which the bond between the 5- and the 6- positions is a double bond. The resultant compound is then reduced in the presence of a catalyst, e.g. Raney nickel, to afford the compound expressed by formula I in which the bond between the 5- and the 6- positions is a single bond.
COPYRIGHT: (C)1982,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP9369080A JPS5718664A (en) | 1980-07-07 | 1980-07-07 | N-substituted-bicyclo- 2.2.1 -hept-5-ene-2,3-dicarboximide derivative |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP9369080A JPS5718664A (en) | 1980-07-07 | 1980-07-07 | N-substituted-bicyclo- 2.2.1 -hept-5-ene-2,3-dicarboximide derivative |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS5718664A true JPS5718664A (en) | 1982-01-30 |
Family
ID=14089394
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP9369080A Pending JPS5718664A (en) | 1980-07-07 | 1980-07-07 | N-substituted-bicyclo- 2.2.1 -hept-5-ene-2,3-dicarboximide derivative |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5718664A (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4743805A (en) * | 1985-09-09 | 1988-05-10 | Kabushiki Kaisha Toshiba | Anode assembly of magnetron and method of manufacturing the same |
-
1980
- 1980-07-07 JP JP9369080A patent/JPS5718664A/en active Pending
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4743805A (en) * | 1985-09-09 | 1988-05-10 | Kabushiki Kaisha Toshiba | Anode assembly of magnetron and method of manufacturing the same |
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