JPS57158763A - Novel substituted quinazolines - Google Patents

Novel substituted quinazolines

Info

Publication number
JPS57158763A
JPS57158763A JP57035004A JP3500482A JPS57158763A JP S57158763 A JPS57158763 A JP S57158763A JP 57035004 A JP57035004 A JP 57035004A JP 3500482 A JP3500482 A JP 3500482A JP S57158763 A JPS57158763 A JP S57158763A
Authority
JP
Japan
Prior art keywords
novel substituted
substituted quinazolines
quinazolines
novel
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP57035004A
Other languages
English (en)
Other versions
JPS621947B2 (ja
Inventor
Hans-Jurgen Ernst Hess
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of JPS57158763A publication Critical patent/JPS57158763A/ja
Publication of JPS621947B2 publication Critical patent/JPS621947B2/ja
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • GPHYSICS
    • G01MEASURING; TESTING
    • G01NINVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N33/00Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
    • G01N33/48Biological material, e.g. blood, urine; Haemocytometers
    • G01N33/50Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
    • G01N33/94Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving narcotics or drugs or pharmaceuticals, neurotransmitters or associated receptors
    • G01N33/9453Cardioregulators, e.g. antihypotensives, antiarrhythmics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Biotechnology (AREA)
  • Food Science & Technology (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cell Biology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Microbiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Physics & Mathematics (AREA)
  • Analytical Chemistry (AREA)
  • Biochemistry (AREA)
  • General Physics & Mathematics (AREA)
  • Pathology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
JP57035004A 1981-03-05 1982-03-05 Novel substituted quinazolines Granted JPS57158763A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24074581A 1981-03-05 1981-03-05

Publications (2)

Publication Number Publication Date
JPS57158763A true JPS57158763A (en) 1982-09-30
JPS621947B2 JPS621947B2 (ja) 1987-01-16

Family

ID=22907776

Family Applications (1)

Application Number Title Priority Date Filing Date
JP57035004A Granted JPS57158763A (en) 1981-03-05 1982-03-05 Novel substituted quinazolines

Country Status (8)

Country Link
EP (1) EP0060081B1 (ja)
JP (1) JPS57158763A (ja)
AU (1) AU528068B2 (ja)
CA (1) CA1170259A (ja)
DE (1) DE3264718D1 (ja)
DK (1) DK94382A (ja)
GR (1) GR75878B (ja)
IE (1) IE52578B1 (ja)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CS236097B1 (en) * 1983-06-01 1985-05-15 Jan Koenig Acylderivatives of 2-piperazinochinazoline and method of their preparation
DE3346675A1 (de) * 1983-12-23 1985-07-04 Beiersdorf Ag, 2000 Hamburg Substituierte 1-(4-amino-6,7-dialkoxy-chinazolinyl)-4- cyclohexenyl-derivate des piperazins und homopiperazins, verfahren zu ihrer herstellung und ihre verwendung sowie diese verbindungen enthaltende zubereitungen und zwischenprodukte
JPH0647540B2 (ja) * 1985-07-16 1994-06-22 エーザイ株式会社 虚血性心疾患・不整脈治療・予防剤
AT384218B (de) * 1985-12-04 1987-10-12 Gerot Pharmazeutika Verfahren zur herstellung von neuen chinazolin-derivaten
FR2601141A1 (fr) * 1986-07-02 1988-01-08 Centre Nat Rech Scient Produit de couplage a base d'haptene, utile notamment comme substance immunogene, anticorps correspondants et applications

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4189484A (en) * 1977-11-08 1980-02-19 Mitsubishi Yuka Pharmaceutical Co., Ltd. Antihypertensive quinazoline derivatives
DE2901218A1 (de) * 1979-01-13 1980-07-17 Byk Gulden Lomberg Chem Fab Ung von theophyllin

Also Published As

Publication number Publication date
EP0060081A3 (en) 1982-12-22
JPS621947B2 (ja) 1987-01-16
CA1170259A (en) 1984-07-03
DE3264718D1 (en) 1985-08-22
GR75878B (ja) 1984-08-02
IE52578B1 (en) 1987-12-23
DK94382A (da) 1982-09-06
EP0060081A2 (en) 1982-09-15
EP0060081B1 (en) 1985-07-17
AU8111582A (en) 1982-11-04
AU528068B2 (en) 1983-04-14
IE820486L (en) 1982-09-05

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