JPS5321140A - Production of 11substituted enkephalin derivatives - Google Patents

Production of 11substituted enkephalin derivatives

Info

Publication number
JPS5321140A
JPS5321140A JP9491877A JP9491877A JPS5321140A JP S5321140 A JPS5321140 A JP S5321140A JP 9491877 A JP9491877 A JP 9491877A JP 9491877 A JP9491877 A JP 9491877A JP S5321140 A JPS5321140 A JP S5321140A
Authority
JP
Japan
Prior art keywords
production
enkephalin derivatives
enkephalin
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP9491877A
Other languages
Japanese (ja)
Inventor
Akurei Jiyoonzu Debitsudo
Mairon Shiyuratsutaa Jieemuzu
Andoriyuu Mikuretsu Richiyaado
An Roitaa Jiyudeisu
Henrii Mazuuru Robaato
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
GD Searle LLC
Original Assignee
GD Searle LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by GD Searle LLC filed Critical GD Searle LLC
Publication of JPS5321140A publication Critical patent/JPS5321140A/en
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • C07K14/70—Enkephalins
    • C07K14/702—Enkephalins with at least 1 amino acid in D-form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12—Antidiarrhoeals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1005—Tetrapeptides with the first amino acid being neutral and aliphatic
    • C07K5/1008—Tetrapeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
JP9491877A 1976-08-09 1977-08-08 Production of 11substituted enkephalin derivatives Pending JPS5321140A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US71262676A 1976-08-09 1976-08-09

Publications (1)

Publication Number Publication Date
JPS5321140A true JPS5321140A (en) 1978-02-27

Family

ID=24862912

Family Applications (1)

Application Number Title Priority Date Filing Date
JP9491877A Pending JPS5321140A (en) 1976-08-09 1977-08-08 Production of 11substituted enkephalin derivatives

Country Status (5)

Country Link
JP (1) JPS5321140A (en)
AU (1) AU2768977A (en)
DE (1) DE2735674A1 (en)
FR (1) FR2361349A1 (en)
GB (1) GB1532148A (en)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2655149A1 (en) * 1975-12-17 1977-06-23 Sandoz Ag Analgesic glycine-contg. peptide derivs. - e.g. tyrosyl-glycyl-glycyl-phenylalanyl-norleucine
NL7700785A (en) * 1976-01-26 1977-07-28 Wellcome Found BIOLOGICALLY ACTIVE PEPTIDES FOR MORPHINE REPLACEMENT.
DK28377A (en) * 1976-02-02 1977-08-03 Sandoz Ag PROCEDURE FOR PREPARING POLYPEPTIDE DERIVATIVES

Also Published As

Publication number Publication date
FR2361349A1 (en) 1978-03-10
AU2768977A (en) 1979-02-15
DE2735674A1 (en) 1978-02-16
GB1532148A (en) 1978-11-15

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