JPS5271456A - Synthesis of 1alpha-hydroxysteroid derivatives - Google Patents

Synthesis of 1alpha-hydroxysteroid derivatives

Info

Publication number
JPS5271456A
JPS5271456A JP14737375A JP14737375A JPS5271456A JP S5271456 A JPS5271456 A JP S5271456A JP 14737375 A JP14737375 A JP 14737375A JP 14737375 A JP14737375 A JP 14737375A JP S5271456 A JPS5271456 A JP S5271456A
Authority
JP
Japan
Prior art keywords
1alpha
synthesis
derivatives
hydroxysteroid
hydroxysteroid derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP14737375A
Other languages
Japanese (ja)
Other versions
JPS5512919B2 (en
Inventor
Hiroyuki Nagano
Sadao Tanaka
Kiyoshige Ochi
Isao Matsunaga
Minoru Shindo
Masayuki Ishikawa
Chikara Kaneko
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Chugai Pharmaceutical Co Ltd
Original Assignee
Chugai Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chugai Pharmaceutical Co Ltd filed Critical Chugai Pharmaceutical Co Ltd
Priority to JP14737375A priority Critical patent/JPS5271456A/en
Publication of JPS5271456A publication Critical patent/JPS5271456A/en
Publication of JPS5512919B2 publication Critical patent/JPS5512919B2/ja
Granted legal-status Critical Current

Links

Abstract

PURPOSE: To prepare intermediates for active vitamine D,s by direct introduction of 1α-OH to 3β-hydroxy-1,5-diene-steroid derivatives by a specific mercuration process.
COPYRIGHT: (C)1977,JPO&Japio
JP14737375A 1975-12-12 1975-12-12 Synthesis of 1alpha-hydroxysteroid derivatives Granted JPS5271456A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP14737375A JPS5271456A (en) 1975-12-12 1975-12-12 Synthesis of 1alpha-hydroxysteroid derivatives

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP14737375A JPS5271456A (en) 1975-12-12 1975-12-12 Synthesis of 1alpha-hydroxysteroid derivatives

Publications (2)

Publication Number Publication Date
JPS5271456A true JPS5271456A (en) 1977-06-14
JPS5512919B2 JPS5512919B2 (en) 1980-04-04

Family

ID=15428755

Family Applications (1)

Application Number Title Priority Date Filing Date
JP14737375A Granted JPS5271456A (en) 1975-12-12 1975-12-12 Synthesis of 1alpha-hydroxysteroid derivatives

Country Status (1)

Country Link
JP (1) JPS5271456A (en)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4284577A (en) * 1979-02-16 1981-08-18 Sachiko Yamada Novel vitamin D3 derivative and process for preparing the same
US4341774A (en) * 1979-08-10 1982-07-27 Chugai Seiyaku Kabushiki Kaisha Method for suppressing abnormal rise in immunological function and agent useful therefor
WO2001040177A2 (en) 1999-12-02 2001-06-07 Women And Infants Hospital Esters of vitamin d3 and uses thereof
WO2005082375A2 (en) 2004-03-01 2005-09-09 Bioxell Spa Treatment of interstitial cystitis with vitamin d compounds
WO2006051106A1 (en) 2004-11-12 2006-05-18 Bioxell Spa Combined use of vitamin d derivatives and anti-proliferative agents for treating bladder cancer
US7462610B2 (en) 2003-04-01 2008-12-09 Hollis-Eden Pharmaceuticals, Inc. Prostate cancer treatment

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS59164065A (en) * 1983-03-07 1984-09-17 日機装株式会社 Simple cooler

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4284577A (en) * 1979-02-16 1981-08-18 Sachiko Yamada Novel vitamin D3 derivative and process for preparing the same
US4341774A (en) * 1979-08-10 1982-07-27 Chugai Seiyaku Kabushiki Kaisha Method for suppressing abnormal rise in immunological function and agent useful therefor
WO2001040177A2 (en) 1999-12-02 2001-06-07 Women And Infants Hospital Esters of vitamin d3 and uses thereof
US7462610B2 (en) 2003-04-01 2008-12-09 Hollis-Eden Pharmaceuticals, Inc. Prostate cancer treatment
WO2005082375A2 (en) 2004-03-01 2005-09-09 Bioxell Spa Treatment of interstitial cystitis with vitamin d compounds
WO2006051106A1 (en) 2004-11-12 2006-05-18 Bioxell Spa Combined use of vitamin d derivatives and anti-proliferative agents for treating bladder cancer

Also Published As

Publication number Publication date
JPS5512919B2 (en) 1980-04-04

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