JPS51143673A - New derivatives of 4-aminopiperidines - Google Patents

New derivatives of 4-aminopiperidines

Info

Publication number
JPS51143673A
JPS51143673A JP51061548A JP6154876A JPS51143673A JP S51143673 A JPS51143673 A JP S51143673A JP 51061548 A JP51061548 A JP 51061548A JP 6154876 A JP6154876 A JP 6154876A JP S51143673 A JPS51143673 A JP S51143673A
Authority
JP
Japan
Prior art keywords
alkyl
aminopiperidines
new derivatives
new
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP51061548A
Other languages
Japanese (ja)
Other versions
JPS6241223B2 (en
Inventor
Nobuo Soma
Tomoyuki Kurumada
Burunetsuchi Heimo
Rodei Jiyan
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Sankyo Co Ltd
Original Assignee
Ciba Geigy AG
Sankyo Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG, Sankyo Co Ltd filed Critical Ciba Geigy AG
Publication of JPS51143673A publication Critical patent/JPS51143673A/en
Publication of JPS6241223B2 publication Critical patent/JPS6241223B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/20—Spiro-condensed ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D211/74—Oxygen atoms
    • C07D211/76—Oxygen atoms attached in position 2 or 6
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/92—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with a hetero atom directly attached to the ring nitrogen atom
    • C07D211/94—Oxygen atom, e.g. piperidine N-oxide
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576—Six-membered rings
    • C07F9/58—Pyridine rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576—Six-membered rings
    • C07F9/59—Hydrogenated pyridine rings
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08K—Use of inorganic or non-macromolecular organic substances as compounding ingredients
    • C08K5/00—Use of organic ingredients
    • C08K5/16—Nitrogen-containing compounds
    • C08K5/34—Heterocyclic compounds having nitrogen in the ring
    • C08K5/3412—Heterocyclic compounds having nitrogen in the ring having one nitrogen atom in the ring
    • C08K5/3432—Six-membered rings
    • C08K5/3435—Piperidines

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Polymers & Plastics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hydrogenated Pyridines (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

PURPOSE: 4-Aminopiperidine derivatives and their salts of the following formula (where R1 is C2-6 alkyl; R2 is C1-6 alkyl; R3 is C1-9 alkyl, phenyl, benzyl or phenylethyl; R4 is C1-6 alkyl, cyclopentyl or cyclohexyl formed from R3 and R4 together; R5 is C1-5 alkyl, C3-4 alkenyl, etc.; R6 is C1-5 alkyl, C7-8 aralkyl, etc.; R7 is H, C1-12 alkyl, cycloalkyl, etc.; X is H, oxyl radical, alkyl, etc.; Y is H or -CO-R13 group, etc.; n is 1, 2 or 3) are new.
COPYRIGHT: (C)1976,JPO&Japio
JP51061548A 1975-05-28 1976-05-27 New derivatives of 4-aminopiperidines Granted JPS51143673A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB23226/75A GB1492494A (en) 1975-05-28 1975-05-28 Derivatives of 4-aminopiperidine

Publications (2)

Publication Number Publication Date
JPS51143673A true JPS51143673A (en) 1976-12-10
JPS6241223B2 JPS6241223B2 (en) 1987-09-02

Family

ID=10192206

Family Applications (2)

Application Number Title Priority Date Filing Date
JP51061548A Granted JPS51143673A (en) 1975-05-28 1976-05-27 New derivatives of 4-aminopiperidines
JP59065524A Expired JPS6046142B2 (en) 1975-05-28 1984-04-02 Stabilized organic polymer composition

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP59065524A Expired JPS6046142B2 (en) 1975-05-28 1984-04-02 Stabilized organic polymer composition

Country Status (9)

Country Link
JP (2) JPS51143673A (en)
AT (1) ATA389276A (en)
BE (1) BE842236A (en)
CH (1) CH601401A5 (en)
DE (1) DE2621870A1 (en)
FR (3) FR2333795A1 (en)
GB (1) GB1492494A (en)
NL (1) NL7605796A (en)
SE (1) SE7605286L (en)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS567764A (en) * 1979-06-21 1981-01-27 Ciba Geigy Ag Novel polyalkylpiperidylurea and stabilizer made therefrom
JPS56122352A (en) * 1980-02-02 1981-09-25 Huels Chemische Werke Ag Manufacture of 44aminoo2*2*6*66 tetramethylpiperidine
JPS56152462A (en) * 1980-03-28 1981-11-26 Ciba Geigy Ag Amide derivative of polyalkylpiperidine and its use
JPH01121265A (en) * 1987-11-06 1989-05-12 Sankyo Co Ltd Production of aminopiperidine derivative
JPH01160959A (en) * 1987-11-14 1989-06-23 Basf Ag 4-formylaminopiperidine derivative, its use as stabilizer and orgnaic material stabilized thereby
JPH11322714A (en) * 1998-03-09 1999-11-24 Ciba Specialty Chem Holding Inc 1-alkoxy-polyalkyl-piperidine derivative and use thereof as polymerization adjusting agent

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2642446A1 (en) * 1976-09-21 1978-03-30 Bayer Ag METHYLOL DERIVATIVES OF 2,2,6,6-TETRAALKYLPIPERIDINE, THEIR PRODUCTION AND USE
US4144224A (en) * 1976-11-26 1979-03-13 Ciba-Geigy Corporation Phosphonate stabilizers
IT1088576B (en) * 1977-11-29 1985-06-10 Montedison Spa POLYMER STABILIZERS AND POLYMER COMPOSITIONS WITH THEM STABILIZED
IT1088581B (en) * 1977-12-02 1985-06-10 Montedison Spa POLYMER STABILIZERS AND POLYMER COMPOSITIONS WITH THEM STABILIZED
DE2920918A1 (en) * 1979-05-23 1980-11-27 Hoechst Ag COPOLYMERS SUBSTITUTED PIPERIDINE, THEIR PRODUCTION AND USE
IT1141369B (en) * 1980-02-22 1986-10-01 Montedison Spa ACIDS AND CORRESPONDING SALTS CONTAINING THE GROUP OF 4-AMINOPIPERIDINE TETRA-ALCHIL REPLACED AND POLYMERIC COMPOSITIONS STABILIZED BY THEM
US4326063A (en) * 1980-07-24 1982-04-20 The B. F. Goodrich Company High molecular weight piperidine derivatives as UV stabilizers
US4316837A (en) * 1980-09-10 1982-02-23 Carstab Corporation Polyalkylated 4-aminopiperidine derivatives as stabilizers for synthetic polymers
DE3111209A1 (en) * 1981-03-21 1982-09-30 Hoechst Ag, 6000 Frankfurt HIGH MOLECULAR PIPERIDING GROUP-CONTAINING ESTERS AND URETHANES, METHOD FOR THE PRODUCTION THEREOF, THEIR USE AS STABILIZERS FOR POLYMERS AND POLYMERS CONTAINING THESE COMPOUNDS
US4520171A (en) * 1982-05-05 1985-05-28 Hercules Incorporated Polymeric hindered amines
US4661594A (en) * 1984-02-29 1987-04-28 Ciba-Geigy Corporation Certain [(2,2,6,6-tetramethyl-4-piperidyl)amino]-1,3,2-dioxaphosphorinanes useful as stabilizers for protecting resins
US4605743A (en) * 1985-04-16 1986-08-12 Uniroyal Chemical Company, Inc. Process for the production of 2,2,6,6-tetraalkyl-4-piperidylamines
JPH0618927B2 (en) * 1985-04-17 1994-03-16 住友化学工業株式会社 Stabilizer for synthetic resins
CH669195A5 (en) * 1985-09-03 1989-02-28 Basf Ag FURANE-3-carboxylic acid derivatives and their use as SUNSCREEN AGENTS OUTSIDE THE TEXTILE INDUSTRY.
FR2587340B1 (en) * 1985-09-13 1990-04-20 Sandoz Sa NOVEL TETRAALKYLPIPERIDINES, THEIR PREPARATION AND THEIR USE AS STABILIZERS OF POLYMERIC MATERIALS
EP0253010B1 (en) * 1986-07-16 1992-12-02 The B.F. GOODRICH Company N-(substituted cyclic alkyleneimine)-alpha-(3,5-di-alkyl-4-hydroxy-phenyl)-alpha, alpha-dialkyl acetamides
GB8626609D0 (en) * 1986-11-07 1986-12-10 Sandoz Ltd Organic compounds
ATE102666T1 (en) * 1988-06-14 1994-03-15 Ciba Geigy Ag PROCESS FOR THE PHOTOCHEMICAL STABILIZATION OF DYED AND DYED POLYPROPYLENE FIBERS.
GB9103415D0 (en) * 1991-02-19 1991-04-03 Sandoz Ltd Improvements in or relating to organic compounds
DE19704460A1 (en) * 1997-02-06 1998-08-13 Huels Chemische Werke Ag Continuous process for the production of 4-aminopiperidines
TW541303B (en) * 2000-03-22 2003-07-11 Ciba Sc Holding Ag 2,2,6,6 diethyl-dimethyl-1-alkoxy-piperidine compounds and their corresponding 1-oxides
MXPA05000307A (en) * 2002-08-07 2005-03-31 Ciba Sc Holding Ag Beta-nucleating, light stabilizing agents for polypropylene.
ES2381710T3 (en) * 2008-08-28 2012-05-30 Basf Se Stabilizers for inanimate organic materials

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS567764A (en) * 1979-06-21 1981-01-27 Ciba Geigy Ag Novel polyalkylpiperidylurea and stabilizer made therefrom
JPH0135826B2 (en) * 1979-06-21 1989-07-27 Ciba Geigy
JPS56122352A (en) * 1980-02-02 1981-09-25 Huels Chemische Werke Ag Manufacture of 44aminoo2*2*6*66 tetramethylpiperidine
JPH031305B2 (en) * 1980-02-02 1991-01-10 Huels Ag
JPS56152462A (en) * 1980-03-28 1981-11-26 Ciba Geigy Ag Amide derivative of polyalkylpiperidine and its use
JPH01121265A (en) * 1987-11-06 1989-05-12 Sankyo Co Ltd Production of aminopiperidine derivative
JPH01160959A (en) * 1987-11-14 1989-06-23 Basf Ag 4-formylaminopiperidine derivative, its use as stabilizer and orgnaic material stabilized thereby
JPH11322714A (en) * 1998-03-09 1999-11-24 Ciba Specialty Chem Holding Inc 1-alkoxy-polyalkyl-piperidine derivative and use thereof as polymerization adjusting agent

Also Published As

Publication number Publication date
FR2333797A1 (en) 1977-07-01
ATA389276A (en) 1977-05-15
FR2333795B1 (en) 1978-08-25
DE2621870A1 (en) 1976-12-16
JPS6241223B2 (en) 1987-09-02
SE7605286L (en) 1976-11-29
FR2333795A1 (en) 1977-07-01
FR2357546A1 (en) 1978-02-03
NL7605796A (en) 1976-11-30
JPS6046142B2 (en) 1985-10-14
CH601401A5 (en) 1978-07-14
BE842236A (en) 1976-11-26
FR2357546B1 (en) 1981-10-09
GB1492494A (en) 1977-11-23
FR2333797B1 (en) 1980-10-03
JPS59182826A (en) 1984-10-17

Similar Documents

Publication Publication Date Title
JPS51143673A (en) New derivatives of 4-aminopiperidines
JPS51143674A (en) New derivatives of 4-oxopiperidines
ES435246A1 (en) Piperidine derivatives
JPS51125291A (en) A process for preparing novel carbostyryl derivatives
JPS5271492A (en) Synthesis of 9-substituted-2-substituted thioadenines
JPS5297934A (en) N#-arylsulfonyl-l-argininamides and their salts acceptable as medicine s
JPS51143691A (en) New derivatives of 1,4-diaza-5-oxo- cycloheptanes
JPS51115411A (en) Process for preparation of novel peroxyesters
JPS51138670A (en) Process for preparing phthalimide derivatives
JPS51128980A (en) Process for preparing 3,4- dihydrocarbostyril derivatives
JPS5356677A (en) 5-fluorouracil derivatives
JPS51146474A (en) Process for preparing piperidylbenzimidazole derivatives
JPS51123823A (en) A barbituric acid insecticide and tickicide
JPS51118799A (en) Method for preparing pyridindole derivatives
JPS5283672A (en) Novel 2-amino-1,4-dihydropyridine derivatives
JPS5287174A (en) Preparation of novel 2-amino 1,4-dihydropyridine derivatives
JPS51128977A (en) Process for preparing carbostyril derivatives
JPS5363382A (en) Nicotinic acid esters and their preparation
JPS51145548A (en) Stabilizers for polymeric materials
JPS53108997A (en) Optical active halolactone and its synthesis
JPS51151326A (en) Nonmedical germicide
JPS51136677A (en) Process for preparation of carbostyril derivatives
JPS5283571A (en) Glutarimide derivatives
JPS5350179A (en) Novel 2-pyridone compounds and their preparation
JPS51141864A (en) Process for preparing oxyindole derivatives.