JPS51125232A - Process for preparing 4-substituted amido-3,5-dihalogeno-alpha-substituted aminomethylbenzyl alcohols - Google Patents

Process for preparing 4-substituted amido-3,5-dihalogeno-alpha-substituted aminomethylbenzyl alcohols

Info

Publication number
JPS51125232A
JPS51125232A JP1499375A JP1499375A JPS51125232A JP S51125232 A JPS51125232 A JP S51125232A JP 1499375 A JP1499375 A JP 1499375A JP 1499375 A JP1499375 A JP 1499375A JP S51125232 A JPS51125232 A JP S51125232A
Authority
JP
Japan
Prior art keywords
substituted
aminomethylbenzyl
dihalogeno
alcohols
alpha
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP1499375A
Other languages
Japanese (ja)
Other versions
JPS5740819B2 (en
Inventor
Kiyoshi Murase
Masuo Murakami
Kozo Takahashi
Toshiyasu Mase
Akira Ida
Takaichi Takenaka
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Yamanouchi Pharmaceutical Co Ltd
Original Assignee
Yamanouchi Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yamanouchi Pharmaceutical Co Ltd filed Critical Yamanouchi Pharmaceutical Co Ltd
Priority to JP1499375A priority Critical patent/JPS51125232A/en
Priority to GB254476A priority patent/GB1523974A/en
Priority to US05/651,738 priority patent/US4063025A/en
Priority to DE19762603417 priority patent/DE2603417A1/en
Priority to DK46176A priority patent/DK46176A/en
Priority to FR7603192A priority patent/FR2299855A1/en
Publication of JPS51125232A publication Critical patent/JPS51125232A/en
Priority to US05/809,998 priority patent/US4145363A/en
Publication of JPS5740819B2 publication Critical patent/JPS5740819B2/ja
Granted legal-status Critical Current

Links

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  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

PURPOSE: 4-Substituted amodo-3,5-dihalogeno-α-substituted aminomethylbenzyl alcohols and their acid adduct salts of formula I where X is halogen; R is alkyl,alkoxycarbonyl,acyl,methanesulfonyl or carbamoyl; R2 is alkyl,chloroalkyl or formula III (where R3 and R4 are H or alkyl; R5 and R6 are H,alkyl,alkoxy or OH; n is 1-3) are new: in an example,3,5-dichloro4-methylamino-α-(N-t-butylaminomethyl)-benzyl alcohol.
COPYRIGHT: (C)1976,JPO&Japio
JP1499375A 1975-02-05 1975-02-05 Process for preparing 4-substituted amido-3,5-dihalogeno-alpha-substituted aminomethylbenzyl alcohols Granted JPS51125232A (en)

Priority Applications (7)

Application Number Priority Date Filing Date Title
JP1499375A JPS51125232A (en) 1975-02-05 1975-02-05 Process for preparing 4-substituted amido-3,5-dihalogeno-alpha-substituted aminomethylbenzyl alcohols
GB254476A GB1523974A (en) 1975-02-05 1976-01-22 4-substituted amino- -aminomethylbenzyl alcohol derivatives
US05/651,738 US4063025A (en) 1975-02-05 1976-01-23 4-Substituted amino-α-aminomethylbenzyl alcohol derivatives
DE19762603417 DE2603417A1 (en) 1975-02-05 1976-01-30 4-SUBSTITUTED AMINO-ALPHA-AMINOMETHYLBENZYL ALCOHOL DERIVATIVES
DK46176A DK46176A (en) 1975-02-05 1976-02-04 PROCEDURE FOR PREPARING 4-AMINO-ALFA-AMINOMETHYL-BENZYL ALCOHOL COMPOUNDS
FR7603192A FR2299855A1 (en) 1975-02-05 1976-02-05 AMINO-4-SUBSTITUTE-AMINOMETHYLBENZYL ALCOHOL DERIVATIVE
US05/809,998 US4145363A (en) 1975-02-05 1977-06-27 4-Carbamoylamino-α-aminomethylbenzyl alcohol derivatives

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP1499375A JPS51125232A (en) 1975-02-05 1975-02-05 Process for preparing 4-substituted amido-3,5-dihalogeno-alpha-substituted aminomethylbenzyl alcohols

Publications (2)

Publication Number Publication Date
JPS51125232A true JPS51125232A (en) 1976-11-01
JPS5740819B2 JPS5740819B2 (en) 1982-08-30

Family

ID=11876451

Family Applications (1)

Application Number Title Priority Date Filing Date
JP1499375A Granted JPS51125232A (en) 1975-02-05 1975-02-05 Process for preparing 4-substituted amido-3,5-dihalogeno-alpha-substituted aminomethylbenzyl alcohols

Country Status (1)

Country Link
JP (1) JPS51125232A (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57122048A (en) * 1980-12-10 1982-07-29 Thomae Gmbh Dr K Novel phenylalkylamine compound

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57122048A (en) * 1980-12-10 1982-07-29 Thomae Gmbh Dr K Novel phenylalkylamine compound

Also Published As

Publication number Publication date
JPS5740819B2 (en) 1982-08-30

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