JP6992284B2 - ジヒドロインドリジノン誘導体を含有する医薬組成物 - Google Patents

ジヒドロインドリジノン誘導体を含有する医薬組成物 Download PDF

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JP6992284B2
JP6992284B2 JP2017111066A JP2017111066A JP6992284B2 JP 6992284 B2 JP6992284 B2 JP 6992284B2 JP 2017111066 A JP2017111066 A JP 2017111066A JP 2017111066 A JP2017111066 A JP 2017111066A JP 6992284 B2 JP6992284 B2 JP 6992284B2
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fluoro
edema
chloro
phenyl
tetrazole
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Japanese (ja)
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JP2017218449A5 (https=
JP2017218449A (ja
Inventor
元之 田中
隆史 近藤
康男 廣岡
泰平 西山
篤 平松
智之 耕田
祥 神山
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Ono Pharmaceutical Co Ltd
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Ono Pharmaceutical Co Ltd
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2017111066A 2016-06-06 2017-06-05 ジヒドロインドリジノン誘導体を含有する医薬組成物 Expired - Fee Related JP6992284B2 (ja)

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JP2016112327 2016-06-06
JP2016112327 2016-06-06

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JP2017218449A JP2017218449A (ja) 2017-12-14
JP2017218449A5 JP2017218449A5 (https=) 2020-07-09
JP6992284B2 true JP6992284B2 (ja) 2022-01-13

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JP2017111066A Expired - Fee Related JP6992284B2 (ja) 2016-06-06 2017-06-05 ジヒドロインドリジノン誘導体を含有する医薬組成物

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Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ776666A (en) * 2018-11-30 2024-11-29 Ono Pharmaceutical Co Novel crystal of (3s)-3-[2-(6-amino-2-fluoropyridin-3-yl)-4-fluoro-1h-imidazol-5-yl]-7-[5-chloro-2-(1h-tetrazol-1-yl)phenyl]-2,3-dihydroindolizin-5(1h)-one
WO2020259668A1 (zh) * 2019-06-28 2020-12-30 上海济煜医药科技有限公司 三并环类化合物及其制备方法和用途
CN116133660B (zh) 2020-07-22 2025-05-02 詹森药业有限公司 可用作因子XIa抑制剂的化合物
JP2024125436A (ja) * 2021-07-20 2024-09-19 小野薬品工業株式会社 イミダゾール化合物の製造方法
TWI833610B (zh) * 2022-03-21 2024-02-21 大陸商上海濟煜醫藥科技有限公司 三并環類化合物製備方法及其中間體
UY40234A (es) 2022-04-22 2023-11-15 Vertex Pharma Compuestos heteroarilo para el tratamiento del dolor

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2015500868A (ja) 2011-12-21 2015-01-08 小野薬品工業株式会社 第ＸＩａ因子阻害剤としての新規ピリジノンおよびピリミジノン誘導体
JP6610562B2 (ja) 2014-12-10 2019-11-27 小野薬品工業株式会社 ジヒドロインドリジノン誘導体

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2015500868A (ja) 2011-12-21 2015-01-08 小野薬品工業株式会社 第ＸＩａ因子阻害剤としての新規ピリジノンおよびピリミジノン誘導体
JP6610562B2 (ja) 2014-12-10 2019-11-27 小野薬品工業株式会社 ジヒドロインドリジノン誘導体
JP6791338B2 (ja) 2014-12-10 2020-11-25 小野薬品工業株式会社 ジヒドロインドリジノン誘導体

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
MEDCHEM NEWS，2009年，19(2)，p.7-12
ファルマシア，2014年，50(1)，p.34-38

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