JP6367545B2 - ルキソリチニブの重水素化誘導体 - Google Patents
ルキソリチニブの重水素化誘導体 Download PDFInfo
- Publication number
- JP6367545B2 JP6367545B2 JP2013259713A JP2013259713A JP6367545B2 JP 6367545 B2 JP6367545 B2 JP 6367545B2 JP 2013259713 A JP2013259713 A JP 2013259713A JP 2013259713 A JP2013259713 A JP 2013259713A JP 6367545 B2 JP6367545 B2 JP 6367545B2
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- deuterium
- hydrogen
- compound
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- pharmaceutically acceptable
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- 0 CC1(*)C(*)([C@@](*)(C(*)(*)C#N)[n]2nc(*)c(-c3nc(*)nc4c3c(*)c(*)[n]4)c2*)C(*)(*)C(*)(*)C1(*)* Chemical compound CC1(*)C(*)([C@@](*)(C(*)(*)C#N)[n]2nc(*)c(-c3nc(*)nc4c3c(*)c(*)[n]4)c2*)C(*)(*)C(*)(*)C1(*)* 0.000 description 1
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- Nitrogen Condensed Heterocyclic Rings (AREA)
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Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2013259713A JP6367545B2 (ja) | 2013-12-17 | 2013-12-17 | ルキソリチニブの重水素化誘導体 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2013259713A JP6367545B2 (ja) | 2013-12-17 | 2013-12-17 | ルキソリチニブの重水素化誘導体 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018128417A Division JP6830460B2 (ja) | 2018-07-05 | 2018-07-05 | ルキソリチニブの重水素化誘導体 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2015117185A JP2015117185A (ja) | 2015-06-25 |
| JP2015117185A5 JP2015117185A5 (enrdf_load_stackoverflow) | 2017-02-09 |
| JP6367545B2 true JP6367545B2 (ja) | 2018-08-01 |
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ID=53530252
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013259713A Active JP6367545B2 (ja) | 2013-12-17 | 2013-12-17 | ルキソリチニブの重水素化誘導体 |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JP6367545B2 (enrdf_load_stackoverflow) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2018172421A (ja) * | 2018-07-05 | 2018-11-08 | コンサート ファーマシューティカルズ インコーポレイテッド | ルキソリチニブの重水素化誘導体 |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ776616A (en) * | 2015-06-30 | 2024-11-29 | Eiger Group Int Inc | Use of chloroquine and clemizole compounds for treatment of inflammatory and cancerous conditions |
| AU2016332236B2 (en) * | 2015-09-29 | 2019-04-11 | Kangpu Biopharmaceuticals, Ltd. | Pharmaceutical composition and application thereof |
| RS66006B1 (sr) * | 2016-05-04 | 2024-10-31 | Sun Pharmaceutical Industries Inc | Lečenјe poremećaja opadanјa kose deuterisanim jak inhibitorima |
| US10995103B2 (en) | 2016-07-25 | 2021-05-04 | Shenzhen Targetrx, Inc. | Substituted boric acid compound, pharmaceutical composition comprising same, and application thereof |
| GB201907871D0 (en) * | 2019-06-03 | 2019-07-17 | Small Pharma Ltd | Therapeutic compositions |
| EP4151210A3 (en) * | 2020-01-10 | 2023-06-14 | Harmony Biosciences, LLC | Pyridine-carboline derivatives as mchr1 antagonists for use in therapy |
| WO2021116503A2 (en) * | 2020-06-02 | 2021-06-17 | Small Pharma Ltd | Deuterated compounds |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HUE030418T2 (en) * | 2005-12-13 | 2017-05-29 | Incyte Holdings Corp | Heteroaryl-substituted pyrrolo [2,3-b] pyridines and pyrrolo [2,3-b] pyrimidines as Janus kinase inhibitors |
| EP3050882B1 (en) * | 2010-03-10 | 2018-01-31 | Incyte Holdings Corporation | Piperidin-4-yl azetidine derivatives as jak1 inhibitors |
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2013
- 2013-12-17 JP JP2013259713A patent/JP6367545B2/ja active Active
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2018172421A (ja) * | 2018-07-05 | 2018-11-08 | コンサート ファーマシューティカルズ インコーポレイテッド | ルキソリチニブの重水素化誘導体 |
Also Published As
| Publication number | Publication date |
|---|---|
| JP2015117185A (ja) | 2015-06-25 |
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