JP4234430B2 - チオールを含むｎａａｌａｄアーゼ抑制物質 - Google Patents

チオールを含むｎａａｌａｄアーゼ抑制物質 Download PDF

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JP4234430B2
JP4234430B2 JP2002557903A JP2002557903A JP4234430B2 JP 4234430 B2 JP4234430 B2 JP 4234430B2 JP 2002557903 A JP2002557903 A JP 2002557903A JP 2002557903 A JP2002557903 A JP 2002557903A JP 4234430 B2 JP4234430 B2 JP 4234430B2
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hydrogen
compound
alpha
mercaptopropyl
halo
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JP2004524294A (ja
JP2004524294A5 (enExample
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タカシ ツカモト
パヴェル メイジャー
ドリス ストアマー
バーバラ エス スルシャー
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Eisai Corp of North America
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Guilford Pharmaceuticals Inc
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  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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JP2002557903A 2001-01-17 2002-01-17 チオールを含むｎａａｌａｄアーゼ抑制物質 Expired - Fee Related JP4234430B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US26175401P 2001-01-17 2001-01-17
US34277201P 2001-12-28 2001-12-28
PCT/US2002/001205 WO2002057222A2 (en) 2001-01-17 2002-01-17 Thiol-based naaladase inhibitors

Related Child Applications (1)

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JP2008270033A Division JP2009051854A (ja) 2001-01-17 2008-10-20 チオールを含むｎａａｌａｄアーゼ抑制物質

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JP2004524294A JP2004524294A (ja) 2004-08-12
JP2004524294A5 JP2004524294A5 (enExample) 2005-12-22
JP4234430B2 true JP4234430B2 (ja) 2009-03-04

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JP2002557903A Expired - Fee Related JP4234430B2 (ja) 2001-01-17 2002-01-17 チオールを含むｎａａｌａｄアーゼ抑制物質
JP2008270033A Abandoned JP2009051854A (ja) 2001-01-17 2008-10-20 チオールを含むｎａａｌａｄアーゼ抑制物質

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JP2008270033A Abandoned JP2009051854A (ja) 2001-01-17 2008-10-20 チオールを含むｎａａｌａｄアーゼ抑制物質

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US (4) US6586623B2 (enExample)
EP (1) EP1353903A2 (enExample)
JP (2) JP4234430B2 (enExample)
AU (1) AU2002245271B2 (enExample)
CA (1) CA2435273A1 (enExample)
MX (1) MXPA03006467A (enExample)
WO (1) WO2002057222A2 (enExample)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7105159B1 (en) 1992-11-05 2006-09-12 Sloan-Kettering Institute For Cancer Research Antibodies to prostate-specific membrane antigen
US7070782B1 (en) * 1992-11-05 2006-07-04 Sloan-Kettering Institute For Cancer Research Prostate-specific membrane antigen
US6953668B1 (en) 1992-11-05 2005-10-11 Sloan-Kettering Institute For Cancer Research Prostate-specific membrane antigen
US6569432B1 (en) * 1995-02-24 2003-05-27 Sloan-Kettering Institute For Cancer Research Prostate-specific membrane antigen and uses thereof
US7037647B1 (en) 1995-02-24 2006-05-02 Sloan-Kettering Institute For Cancer Research Prostate-specific membrane antigen and uses thereof
US20040253246A1 (en) * 1996-02-23 2004-12-16 Israeli Ron S. Prostate-specific membrane antigen and uses thereof
JP4234430B2 (ja) * 2001-01-17 2009-03-04 エムジーアイ ジーピー インコーポレイティッド チオールを含むｎａａｌａｄアーゼ抑制物質
CA2436408A1 (en) 2001-02-07 2002-12-12 Beth Israel Deaconess Medical Center Modified psma ligands and uses related thereto
WO2003057670A2 (en) * 2001-12-28 2003-07-17 Guilford Pharmaceuticals Inc. Indoles as naaladase inhibitors
WO2004078180A2 (en) * 2003-03-03 2004-09-16 Guilford Pharmaceuticals Inc. Naaladase inhibitors for treating opioid tolerance
US7125907B2 (en) 2003-03-03 2006-10-24 Guilford Pharmaceuticals Inc. Thiolactones
DE602005024690D1 (de) 2004-07-08 2010-12-23 Aposense Ltd Verfahren und verbindungen zum nachweis von medizinischen erkrankungen
US8023934B2 (en) * 2008-03-28 2011-09-20 Ianywhere Solutions, Inc. Synchronizing communications and data between mobile devices and servers
US8019863B2 (en) 2008-03-28 2011-09-13 Ianywhere Solutions, Inc. Synchronizing events between mobile devices and servers
US20110093619A1 (en) * 2009-10-16 2011-04-21 Ianywhere Solutions, Inc. Synchronizing Tasks between Mobile Devices and Servers
US8434097B2 (en) * 2009-12-30 2013-04-30 Sybase, Inc. Dynamic data binding for MBOs for container based application
JP6798075B2 (ja) * 2015-06-15 2020-12-09 エヌエムディー ファーマ エー／エス 神経筋障害を処置するのにおける使用のための化合物
US10385028B2 (en) 2017-12-14 2019-08-20 Nmd Pharma A/S Compounds for the treatment of neuromuscular disorders
US11147788B2 (en) 2017-12-14 2021-10-19 Nmd Pharma A/S Compounds for the treatment of neuromuscular disorders
US11591284B2 (en) 2017-12-14 2023-02-28 Nmd Pharma A/S Compounds for the treatment of neuromuscular disorders
US11730714B2 (en) 2017-12-14 2023-08-22 Nmd Pharma A/S Compounds for the treatment of neuromuscular disorders
US12440477B2 (en) 2017-12-14 2025-10-14 Nmd Pharma A/S Compounds for the treatment of neuromuscular disorders

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1998053812A1 (en) * 1997-05-27 1998-12-03 Guilford Pharmaceuticals Inc. Inhibitors of naaladase enzyme activity
EP1093453B1 (en) * 1998-07-06 2005-09-28 Guilford Pharmaceuticals Inc. Naaladase inhibitors useful as pharmaceutical compounds and compositions
AU6661901A (en) * 2000-05-30 2001-12-11 Guilford Pharm Inc Naaladase inhibitors for treating retinal disorders and glaucoma
WO2001092273A2 (en) * 2000-05-30 2001-12-06 Guilford Pharmaceuticals Inc. Benzenedicarboxylic acid derivatives
WO2001091738A2 (en) * 2000-05-30 2001-12-06 Guilford Pharmaceuticals Inc. Naaladase inhibitors for treating amyotrophic lateral sclerosis
JP4234430B2 (ja) * 2001-01-17 2009-03-04 エムジーアイ ジーピー インコーポレイティッド チオールを含むｎａａｌａｄアーゼ抑制物質

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US6992215B2 (en) 2006-01-31
US6586623B2 (en) 2003-07-01
WO2002057222A2 (en) 2002-07-25
US20030216468A1 (en) 2003-11-20
JP2004524294A (ja) 2004-08-12
JP2009051854A (ja) 2009-03-12
MXPA03006467A (es) 2004-01-29
US20050085503A1 (en) 2005-04-21
CA2435273A1 (en) 2002-07-25
WO2002057222A9 (en) 2004-05-06
EP1353903A2 (en) 2003-10-22
US6812364B2 (en) 2004-11-02
AU2002245271B2 (en) 2008-01-31
WO2002057222A3 (en) 2002-12-19
US20060135812A1 (en) 2006-06-22
US20030105088A1 (en) 2003-06-05

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