JP4234430B2 - チオールを含むｎａａｌａｄアーゼ抑制物質 - Google Patents

チオールを含むｎａａｌａｄアーゼ抑制物質 Download PDF

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JP4234430B2
JP4234430B2 JP2002557903A JP2002557903A JP4234430B2 JP 4234430 B2 JP4234430 B2 JP 4234430B2 JP 2002557903 A JP2002557903 A JP 2002557903A JP 2002557903 A JP2002557903 A JP 2002557903A JP 4234430 B2 JP4234430 B2 JP 4234430B2
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hydrogen
compound
alpha
mercaptopropyl
halo
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JP2004524294A (ja
JP2004524294A5 (enExample
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タカシ ツカモト
パヴェル メイジャー
ドリス ストアマー
バーバラ エス スルシャー
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Eisai Corp of North America
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Guilford Pharmaceuticals Inc
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  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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JP2002557903A 2001-01-17 2002-01-17 チオールを含むｎａａｌａｄアーゼ抑制物質 Expired - Fee Related JP4234430B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US26175401P 2001-01-17 2001-01-17
US34277201P 2001-12-28 2001-12-28
PCT/US2002/001205 WO2002057222A2 (en) 2001-01-17 2002-01-17 Thiol-based naaladase inhibitors

Related Child Applications (1)

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JP2008270033A Division JP2009051854A (ja) 2001-01-17 2008-10-20 チオールを含むｎａａｌａｄアーゼ抑制物質

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JP2004524294A JP2004524294A (ja) 2004-08-12
JP2004524294A5 JP2004524294A5 (enExample) 2005-12-22
JP4234430B2 true JP4234430B2 (ja) 2009-03-04

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JP2002557903A Expired - Fee Related JP4234430B2 (ja) 2001-01-17 2002-01-17 チオールを含むｎａａｌａｄアーゼ抑制物質
JP2008270033A Abandoned JP2009051854A (ja) 2001-01-17 2008-10-20 チオールを含むｎａａｌａｄアーゼ抑制物質

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JP2008270033A Abandoned JP2009051854A (ja) 2001-01-17 2008-10-20 チオールを含むｎａａｌａｄアーゼ抑制物質

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US (4) US6586623B2 (enExample)
EP (1) EP1353903A2 (enExample)
JP (2) JP4234430B2 (enExample)
AU (1) AU2002245271B2 (enExample)
CA (1) CA2435273A1 (enExample)
MX (1) MXPA03006467A (enExample)
WO (1) WO2002057222A2 (enExample)

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7105159B1 (en) 1992-11-05 2006-09-12 Sloan-Kettering Institute For Cancer Research Antibodies to prostate-specific membrane antigen
US6953668B1 (en) 1992-11-05 2005-10-11 Sloan-Kettering Institute For Cancer Research Prostate-specific membrane antigen
US7070782B1 (en) * 1992-11-05 2006-07-04 Sloan-Kettering Institute For Cancer Research Prostate-specific membrane antigen
WO1996026272A1 (en) 1995-02-24 1996-08-29 Sloan-Kettering Institute For Cancer Research Prostate-specific membrane antigen and uses thereof
US6569432B1 (en) * 1995-02-24 2003-05-27 Sloan-Kettering Institute For Cancer Research Prostate-specific membrane antigen and uses thereof
US20040253246A1 (en) * 1996-02-23 2004-12-16 Israeli Ron S. Prostate-specific membrane antigen and uses thereof
MXPA03006467A (es) * 2001-01-17 2004-01-29 Guilford Pharm Inc Inibidores de naaladasa a base de tiol.
CA2436408A1 (en) 2001-02-07 2002-12-12 Beth Israel Deaconess Medical Center Modified psma ligands and uses related thereto
US7148250B2 (en) * 2001-12-28 2006-12-12 Guilford Pharmaceuticals Inc. Indoles as NAALADase inhibitors
DE602004021476D1 (de) * 2003-03-03 2009-07-23 Eisai Corp North America THIOLACTONE ALS NAALADase INHIBITOREN
US20040186081A1 (en) * 2003-03-03 2004-09-23 Guilford Pharmaceuticals Inc. Naaladase inhibitors for treating opioid tolerance
JP2008505884A (ja) 2004-07-08 2008-02-28 エヌエスティー・ニューロサバイバル・テクノロジーズ・リミテッド 疾患を検出する方法および化合物
US8023934B2 (en) * 2008-03-28 2011-09-20 Ianywhere Solutions, Inc. Synchronizing communications and data between mobile devices and servers
US8019863B2 (en) 2008-03-28 2011-09-13 Ianywhere Solutions, Inc. Synchronizing events between mobile devices and servers
US20110093619A1 (en) * 2009-10-16 2011-04-21 Ianywhere Solutions, Inc. Synchronizing Tasks between Mobile Devices and Servers
US8434097B2 (en) * 2009-12-30 2013-04-30 Sybase, Inc. Dynamic data binding for MBOs for container based application
KR102722949B1 (ko) * 2015-06-15 2024-10-28 엔엠디 파마 에이/에스 신경근 장애의 치료에 사용하기 위한 화합물
US11591284B2 (en) 2017-12-14 2023-02-28 Nmd Pharma A/S Compounds for the treatment of neuromuscular disorders
US11147788B2 (en) 2017-12-14 2021-10-19 Nmd Pharma A/S Compounds for the treatment of neuromuscular disorders
US12440477B2 (en) 2017-12-14 2025-10-14 Nmd Pharma A/S Compounds for the treatment of neuromuscular disorders
US11730714B2 (en) 2017-12-14 2023-08-22 Nmd Pharma A/S Compounds for the treatment of neuromuscular disorders
US10385028B2 (en) 2017-12-14 2019-08-20 Nmd Pharma A/S Compounds for the treatment of neuromuscular disorders

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0994707A4 (en) * 1997-05-27 2001-11-14 Guilford Pharm Inc INHIBITORS OF NAALADASE ENZYME ACTIVITY
MXPA01000144A (es) * 1998-07-06 2002-10-17 Guilford Pharm Inc Inhibidores de naaladasa utiles como composiciones y compuestos farmaceuticos.
US20020013295A1 (en) 2000-05-30 2002-01-31 Slusher Barbara S. Naaladase inhibitors for treating amyotrophic lateral sclerosis
WO2001092274A2 (en) * 2000-05-30 2001-12-06 Guilford Pharmaceuticals Inc. Naaladase inhibitors for treating retinal disorders and glaucoma
AU2001265111A1 (en) * 2000-05-30 2001-12-11 Guilford Pharmaceuticals Inc. Benzenedicarboxylic acid derivatives
MXPA03006467A (es) * 2001-01-17 2004-01-29 Guilford Pharm Inc Inibidores de naaladasa a base de tiol.

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JP2009051854A (ja) 2009-03-12
US20050085503A1 (en) 2005-04-21
JP2004524294A (ja) 2004-08-12
US20030105088A1 (en) 2003-06-05
MXPA03006467A (es) 2004-01-29
EP1353903A2 (en) 2003-10-22
US6586623B2 (en) 2003-07-01
AU2002245271B2 (en) 2008-01-31
WO2002057222A2 (en) 2002-07-25
US6812364B2 (en) 2004-11-02
US20030216468A1 (en) 2003-11-20
WO2002057222A3 (en) 2002-12-19
CA2435273A1 (en) 2002-07-25
US20060135812A1 (en) 2006-06-22
WO2002057222A9 (en) 2004-05-06
US6992215B2 (en) 2006-01-31

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