JP2022519301A5 - - Google Patents

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Publication number
JP2022519301A5
JP2022519301A5 JP2021545808A JP2021545808A JP2022519301A5 JP 2022519301 A5 JP2022519301 A5 JP 2022519301A5 JP 2021545808 A JP2021545808 A JP 2021545808A JP 2021545808 A JP2021545808 A JP 2021545808A JP 2022519301 A5 JP2022519301 A5 JP 2022519301A5
Authority
JP
Japan
Prior art keywords
pyridine
sulfamoyl
trifluoromethyl
amino
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2021545808A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022519301A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2020/050884 external-priority patent/WO2020161623A1/en
Publication of JP2022519301A publication Critical patent/JP2022519301A/ja
Publication of JP2022519301A5 publication Critical patent/JP2022519301A5/ja
Withdrawn legal-status Critical Current

Links

JP2021545808A 2019-02-06 2020-02-04 N-(ピリジン-2-イル)ピリジン-スルホンアミド誘導体及び疾患の処置におけるそれらの使用 Withdrawn JP2022519301A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962801717P 2019-02-06 2019-02-06
US62/801,717 2019-02-06
PCT/IB2020/050884 WO2020161623A1 (en) 2019-02-06 2020-02-04 N-(pyridin-2-yl)pyridine-sulfonamide derivatives and their use in the treatment of disease

Publications (2)

Publication Number Publication Date
JP2022519301A JP2022519301A (ja) 2022-03-22
JP2022519301A5 true JP2022519301A5 (https=) 2023-02-13

Family

ID=69528901

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021545808A Withdrawn JP2022519301A (ja) 2019-02-06 2020-02-04 N-(ピリジン-2-イル)ピリジン-スルホンアミド誘導体及び疾患の処置におけるそれらの使用

Country Status (5)

Country Link
US (1) US20220127247A1 (https=)
EP (1) EP3921313A1 (https=)
JP (1) JP2022519301A (https=)
CN (1) CN113423702A (https=)
WO (1) WO2020161623A1 (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2019222758B2 (en) 2018-02-15 2022-07-07 Vertex Pharmaceuticals Incorporated Macrocycles as modulators of cystic fibrosis transmembrane conductance regulator, pharmaceutical compositions thereof, their use in the treatment of cystic fibrosis, and process for making them
TWI848092B (zh) 2019-04-03 2024-07-11 美商維泰克斯製藥公司 囊腫纖維化跨膜傳導調節蛋白調節劑
CA3150162A1 (en) 2019-08-14 2021-02-18 Vertex Pharmaceuticals Incorporated Crystalline forms of cftr modulators
TWI867024B (zh) 2019-08-14 2024-12-21 美商維泰克斯製藥公司 囊腫纖維化跨膜傳導調節蛋白之調節劑
TWI899097B (zh) 2019-08-14 2025-10-01 美商維泰克斯製藥公司 製備cftr調節劑之方法
IL300413A (en) 2020-08-13 2023-04-01 Vertex Pharma Crystal forms of CFTR modulators
EP4225762A1 (en) 2020-10-07 2023-08-16 Vertex Pharmaceuticals Incorporated Modulators of cystic fibrosis transmembrane conductance regulator
AU2021397294A1 (en) 2020-12-10 2023-07-06 Vertex Pharmaceuticals Incorporated Methods of treatment for cystic fibrosis

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0301654D0 (sv) * 2003-06-05 2003-06-05 Astrazeneca Ab Novel compounds
WO2015138934A1 (en) * 2014-03-13 2015-09-17 Proteostasis Therapeutics, Inc. Compounds, compositions, and methods for increasing cftr activity
KR20180029204A (ko) * 2015-06-02 2018-03-20 애브비 에스.에이.알.엘. 치환된 피리딘 및 사용 방법
TW201811766A (zh) * 2016-08-29 2018-04-01 瑞士商諾華公司 N-(吡啶-2-基)吡啶-磺醯胺衍生物及其用於疾病治療之用途

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