JP2021511351A5 - - Google Patents
Info
- Publication number
- JP2021511351A5 JP2021511351A5 JP2020540565A JP2020540565A JP2021511351A5 JP 2021511351 A5 JP2021511351 A5 JP 2021511351A5 JP 2020540565 A JP2020540565 A JP 2020540565A JP 2020540565 A JP2020540565 A JP 2020540565A JP 2021511351 A5 JP2021511351 A5 JP 2021511351A5
- Authority
- JP
- Japan
- Prior art keywords
- diazaspiro
- cyclopropane
- bicyclo
- octane
- oxo
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN2018074185 | 2018-01-25 | ||
| CNPCT/CN2018/074185 | 2018-01-25 | ||
| PCT/CN2019/073000 WO2019144912A1 (zh) | 2018-01-25 | 2019-01-24 | β-内酰胺酶抑制剂及其用途 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021511351A JP2021511351A (ja) | 2021-05-06 |
| JP2021511351A5 true JP2021511351A5 (https=) | 2023-03-13 |
| JP7273420B2 JP7273420B2 (ja) | 2023-05-15 |
Family
ID=67394549
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020540565A Active JP7273420B2 (ja) | 2018-01-25 | 2019-01-24 | β－ラクタマーゼ阻害剤及びその用途 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US11078202B2 (https=) |
| EP (1) | EP3744722A4 (https=) |
| JP (1) | JP7273420B2 (https=) |
| KR (1) | KR102769880B1 (https=) |
| CN (1) | CN111670187B (https=) |
| AU (1) | AU2019211693B2 (https=) |
| CA (1) | CA3089150A1 (https=) |
| WO (1) | WO2019144912A1 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR102769880B1 (ko) | 2018-01-25 | 2025-02-20 | 쑤저우 시노벤트 파마슈티칼즈 씨오., 엘티디. | β-락타마제 억제제 및 그 용도 |
| CA3238268A1 (en) | 2021-11-17 | 2023-05-25 | Xufan WANG | ?-lactamase inhibitor intermediate and preparation method therefor |
| CN117186107A (zh) * | 2022-05-31 | 2023-12-08 | 成都先导药物开发股份有限公司 | 一种制备2-取代-5,7-二羰基-2,6-二氮杂螺[3,4]辛烷中间体的方法 |
| EP4659750A1 (en) | 2023-02-02 | 2025-12-10 | Evopoint Biosciences Co., Ltd. | PHARMACEUTICAL COMPOSITION CONTAINING ß-LACTAMASE INHIBITOR AND USE THEREOF |
| CN116730941B (zh) * | 2023-06-15 | 2024-07-02 | 广东省科学院微生物研究所(广东省微生物分析检测中心) | 5-苯基-1,3,4-恶二唑类化合物及其制备方法和应用 |
| CN118453513B (zh) * | 2024-05-23 | 2025-06-17 | 苏州信诺维医药科技股份有限公司 | 一种β-内酰胺酶抑制剂液体制剂的制备工艺 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US1098129A (en) | 1910-04-05 | 1914-05-26 | John Thomas Simpson | Aeroplane. |
| US1033000A (en) | 1910-12-14 | 1912-07-16 | Joseph Leslie Forster | Pneumatic piano-player. |
| US1337809A (en) | 1917-06-22 | 1920-04-20 | Winton Alexander | Protecting means for vessels |
| ES2533826T3 (es) * | 2008-01-18 | 2015-04-15 | Merck Sharp & Dohme Corp. | Inhibidores de beta-lactamasa |
| MX340533B (es) * | 2011-08-30 | 2016-07-13 | Wockhardt Ltd | Derivados de 1,6- diazabiciclo [3,2,1] octan-7-ona y su uso en el tratamiento de infecciones bacterianas. |
| TW201343645A (zh) | 2012-03-30 | 2013-11-01 | Cubist Pharm Inc | １，３，４－□二唑及１，３，４－噻二唑β－內醯胺酶抑制劑 |
| KR20150003777A (ko) * | 2012-03-30 | 2015-01-09 | 큐비스트 파마슈티컬즈 인코포레이티드 | 이속사졸 β-락타마제 억제제 |
| WO2014141132A1 (en) * | 2013-03-14 | 2014-09-18 | Naeja Pharmaceutical Inc. | NEW HETEROCYCLIC COMPOUNDS AND THEIR USE AS ANTIBACTERIAL AGENTS AND β-LACTAMASE INHIBITORS |
| US9822115B2 (en) | 2014-01-21 | 2017-11-21 | Wockhardt Limited | Nitrogen containing compounds and their use as antibacterial agents |
| IN2014MU01196A (https=) * | 2014-03-29 | 2015-10-02 | Wockhardt Ltd | |
| EP3131583A1 (en) | 2014-04-18 | 2017-02-22 | The Wockhardt Limited | Pharmaceutical compositions comprising antibacterial agents |
| WO2015173663A1 (en) | 2014-05-14 | 2015-11-19 | Wockhardt Limited | A process for preparation of trans-sulfuric acid mono-{2-[5-(2-methylamino-ethyl)-[1,3,4]-oxadiazol-2-yl]-7-oxo-1,6-diaza-bicyclo [3.2.1]oct-6-yl} ester |
| WO2015173665A1 (en) | 2014-05-14 | 2015-11-19 | Wockhardt Limited | A process for preparation of trans-sulfuric acid mono-{2-[5-(3-azetidinylamino)-methyl-[1,3,4]- oxadiazol-2-yl]-7-oxo-1,6-diazabicyclo[3.2.1] oct-6-yl} ester trifluoroacetate |
| CA3000087A1 (en) | 2015-10-02 | 2017-04-06 | Legochem Biosciences, Inc. | Compositions and methods for inhibiting beta-lactamase |
| KR102769880B1 (ko) | 2018-01-25 | 2025-02-20 | 쑤저우 시노벤트 파마슈티칼즈 씨오., 엘티디. | β-락타마제 억제제 및 그 용도 |
-
2019
- 2019-01-24 KR KR1020207024397A patent/KR102769880B1/ko active Active
- 2019-01-24 AU AU2019211693A patent/AU2019211693B2/en active Active
- 2019-01-24 CN CN201980010129.1A patent/CN111670187B/zh active Active
- 2019-01-24 EP EP19743504.3A patent/EP3744722A4/en active Pending
- 2019-01-24 CA CA3089150A patent/CA3089150A1/en active Pending
- 2019-01-24 JP JP2020540565A patent/JP7273420B2/ja active Active
- 2019-01-24 WO PCT/CN2019/073000 patent/WO2019144912A1/zh not_active Ceased
-
2020
- 2020-08-20 US US16/998,577 patent/US11078202B2/en active Active
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