JP2021091671A - 多環性ピリドン誘導体を含有する医薬組成物 - Google Patents
多環性ピリドン誘導体を含有する医薬組成物 Download PDFInfo
- Publication number
- JP2021091671A JP2021091671A JP2020196447A JP2020196447A JP2021091671A JP 2021091671 A JP2021091671 A JP 2021091671A JP 2020196447 A JP2020196447 A JP 2020196447A JP 2020196447 A JP2020196447 A JP 2020196447A JP 2021091671 A JP2021091671 A JP 2021091671A
- Authority
- JP
- Japan
- Prior art keywords
- substituted
- unsubstituted
- alkyl
- aromatic
- ring
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
- 0 CC(*C(C(C(O)=C12)=O)=CN1N(CCCCC1)[C@@]1(*1CC1)N(*)C2=O)C(CC1)=CCC1(C)NC Chemical compound CC(*C(C(C(O)=C12)=O)=CN1N(CCCCC1)[C@@]1(*1CC1)N(*)C2=O)C(CC1)=CCC1(C)NC 0.000 description 4
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2019214867 | 2019-11-28 | ||
| JP2019214867 | 2019-11-28 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2021091671A true JP2021091671A (ja) | 2021-06-17 |
| JP2021091671A5 JP2021091671A5 (https=) | 2023-11-29 |
Family
ID=76312248
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020196447A Ceased JP2021091671A (ja) | 2019-11-28 | 2020-11-27 | 多環性ピリドン誘導体を含有する医薬組成物 |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JP2021091671A (https=) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US12564595B2 (en) | 2019-11-28 | 2026-03-03 | Shionogi & Co., Ltd. | Prophylactic and therapeutic pharmaceutical agent for HIV infectious diseases characterized by comprising combination of integrase inhibitor and anti-HIV agent |
| US12577241B2 (en) | 2019-11-28 | 2026-03-17 | Shionogi & Co., Ltd. | Polycyclic pyridopyrazine derivative |
Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2011129095A1 (ja) * | 2010-04-12 | 2011-10-20 | 塩野義製薬株式会社 | インテグラーゼ阻害活性を有するピリドン誘導体 |
| WO2016027879A1 (ja) * | 2014-08-22 | 2016-02-25 | 塩野義製薬株式会社 | インテグラーゼ阻害活性を有する多環性ピリドン誘導体 |
| WO2017087257A1 (en) * | 2015-11-17 | 2017-05-26 | Merck Sharp & Dohme Corp. | Amido-substituted pyridotriazine derivatives useful as hiv integrase inhibitors |
| WO2017087256A1 (en) * | 2015-11-17 | 2017-05-26 | Merck Sharp & Dohme Corp. | Spirocyclic pyridotriazine derivatives useful as hiv integrase inhibitors |
| WO2019160783A1 (en) * | 2018-02-15 | 2019-08-22 | Merck Sharp & Dohme Corp. | Tricyclic heterocycle compounds useful as hiv integrase inhibitors |
| JP7353707B2 (ja) * | 2018-05-31 | 2023-10-02 | 塩野義製薬株式会社 | 多環性ピリドン誘導体 |
-
2020
- 2020-11-27 JP JP2020196447A patent/JP2021091671A/ja not_active Ceased
Patent Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2011129095A1 (ja) * | 2010-04-12 | 2011-10-20 | 塩野義製薬株式会社 | インテグラーゼ阻害活性を有するピリドン誘導体 |
| WO2016027879A1 (ja) * | 2014-08-22 | 2016-02-25 | 塩野義製薬株式会社 | インテグラーゼ阻害活性を有する多環性ピリドン誘導体 |
| WO2017087257A1 (en) * | 2015-11-17 | 2017-05-26 | Merck Sharp & Dohme Corp. | Amido-substituted pyridotriazine derivatives useful as hiv integrase inhibitors |
| WO2017087256A1 (en) * | 2015-11-17 | 2017-05-26 | Merck Sharp & Dohme Corp. | Spirocyclic pyridotriazine derivatives useful as hiv integrase inhibitors |
| WO2019160783A1 (en) * | 2018-02-15 | 2019-08-22 | Merck Sharp & Dohme Corp. | Tricyclic heterocycle compounds useful as hiv integrase inhibitors |
| JP7353707B2 (ja) * | 2018-05-31 | 2023-10-02 | 塩野義製薬株式会社 | 多環性ピリドン誘導体 |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US12564595B2 (en) | 2019-11-28 | 2026-03-03 | Shionogi & Co., Ltd. | Prophylactic and therapeutic pharmaceutical agent for HIV infectious diseases characterized by comprising combination of integrase inhibitor and anti-HIV agent |
| US12577241B2 (en) | 2019-11-28 | 2026-03-17 | Shionogi & Co., Ltd. | Polycyclic pyridopyrazine derivative |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP7353707B2 (ja) | 多環性ピリドン誘導体 | |
| JP7679427B2 (ja) | 多環性カルバモイルピリドン誘導体 | |
| JP7776335B2 (ja) | 多環性ピリドピラジン誘導体 | |
| WO2021107066A1 (ja) | インテグラーゼ阻害剤及び抗hiv薬を組み合わせることを特徴とするhiv感染症の予防及び治療用医薬 | |
| JP2023182723A (ja) | 多環性カルバモイルピリドン誘導体を含有する医薬組成物 | |
| JP2021091671A (ja) | 多環性ピリドン誘導体を含有する医薬組成物 | |
| TWI820141B (zh) | 衍生物 | |
| EA047250B1 (ru) | Полициклическое производное карбамоилпиридона | |
| HK40043566A (en) | Polycyclic pyridone derivative | |
| EA042593B1 (ru) | Полициклическое производное пиридона, полезное для лечения вич-инфекции, его фармацевтическая композиция и применение | |
| EA053268B1 (ru) | Полициклическое производное карбамоилпиридона | |
| WO2023033018A1 (ja) | Hiv複製阻害作用を有する縮合複素環誘導体 | |
| BR122025006471A2 (pt) | Derivado de carbamoilpiridona policíclica e composição farmacêutica compreendendo o mesmo |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RD03 | Notification of appointment of power of attorney |
Free format text: JAPANESE INTERMEDIATE CODE: A7423 Effective date: 20231019 |
|
| A521 | Request for written amendment filed |
Free format text: JAPANESE INTERMEDIATE CODE: A523 Effective date: 20231120 |
|
| A621 | Written request for application examination |
Free format text: JAPANESE INTERMEDIATE CODE: A621 Effective date: 20231120 |
|
| RD04 | Notification of resignation of power of attorney |
Free format text: JAPANESE INTERMEDIATE CODE: A7424 Effective date: 20240122 |
|
| A131 | Notification of reasons for refusal |
Free format text: JAPANESE INTERMEDIATE CODE: A131 Effective date: 20241022 |
|
| A521 | Request for written amendment filed |
Free format text: JAPANESE INTERMEDIATE CODE: A523 Effective date: 20241203 |
|
| A131 | Notification of reasons for refusal |
Free format text: JAPANESE INTERMEDIATE CODE: A131 Effective date: 20250218 |
|
| A521 | Request for written amendment filed |
Free format text: JAPANESE INTERMEDIATE CODE: A523 Effective date: 20250418 |
|
| A01 | Written decision to grant a patent or to grant a registration (utility model) |
Free format text: JAPANESE INTERMEDIATE CODE: A01 Effective date: 20250708 |
|
| A045 | Written measure of dismissal of application [lapsed due to lack of payment] |
Free format text: JAPANESE INTERMEDIATE CODE: A045 Effective date: 20251125 |