JP2018002699A5 - - Google Patents
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- Publication number
- JP2018002699A5 JP2018002699A5 JP2016256790A JP2016256790A JP2018002699A5 JP 2018002699 A5 JP2018002699 A5 JP 2018002699A5 JP 2016256790 A JP2016256790 A JP 2016256790A JP 2016256790 A JP2016256790 A JP 2016256790A JP 2018002699 A5 JP2018002699 A5 JP 2018002699A5
- Authority
- JP
- Japan
- Prior art keywords
- carmellose
- tablet
- combination
- drug substance
- combination tablet
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 239000003826 tablet Substances 0.000 claims 6
- 229920002134 Carboxymethyl cellulose Polymers 0.000 claims 4
- VJHCJDRQFCCTHL-UHFFFAOYSA-N acetic acid 2,3,4,5,6-pentahydroxyhexanal Chemical compound CC(O)=O.OCC(O)C(O)C(O)C(O)C=O VJHCJDRQFCCTHL-UHFFFAOYSA-N 0.000 claims 4
- 235000010948 carboxy methyl cellulose Nutrition 0.000 claims 4
- 229950008138 carmellose Drugs 0.000 claims 4
- OYPRJOBELJOOCE-UHFFFAOYSA-N Calcium Chemical compound [Ca] OYPRJOBELJOOCE-UHFFFAOYSA-N 0.000 claims 2
- 239000008186 active pharmaceutical agent Substances 0.000 claims 2
- 239000011575 calcium Substances 0.000 claims 2
- 229910052791 calcium Inorganic materials 0.000 claims 2
- 239000007884 disintegrant Substances 0.000 claims 2
- 229940088679 drug related substance Drugs 0.000 claims 2
- 239000002947 C09CA04 - Irbesartan Substances 0.000 claims 1
- DPXJVFZANSGRMM-UHFFFAOYSA-N acetic acid;2,3,4,5,6-pentahydroxyhexanal;sodium Chemical compound [Na].CC(O)=O.OCC(O)C(O)C(O)C(O)C=O DPXJVFZANSGRMM-UHFFFAOYSA-N 0.000 claims 1
- ZPBWCRDSRKPIDG-UHFFFAOYSA-N amlodipine benzenesulfonate Chemical group OS(=O)(=O)C1=CC=CC=C1.CCOC(=O)C1=C(COCCN)NC(C)=C(C(=O)OC)C1C1=CC=CC=C1Cl ZPBWCRDSRKPIDG-UHFFFAOYSA-N 0.000 claims 1
- 229960004005 amlodipine besylate Drugs 0.000 claims 1
- 239000007941 film coated tablet Substances 0.000 claims 1
- 239000007888 film coating Substances 0.000 claims 1
- 238000009501 film coating Methods 0.000 claims 1
- YCPOHTHPUREGFM-UHFFFAOYSA-N irbesartan Chemical group O=C1N(CC=2C=CC(=CC=2)C=2C(=CC=CC=2)C=2[N]N=NN=2)C(CCCC)=NC21CCCC2 YCPOHTHPUREGFM-UHFFFAOYSA-N 0.000 claims 1
- 229960002198 irbesartan Drugs 0.000 claims 1
- 239000010410 layer Substances 0.000 claims 1
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2016025015 | 2016-02-12 | ||
| JP2016025015 | 2016-02-12 | ||
| JP2016128121 | 2016-06-28 | ||
| JP2016128121 | 2016-06-28 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2018002699A JP2018002699A (ja) | 2018-01-11 |
| JP2018002699A5 true JP2018002699A5 (enExample) | 2018-02-22 |
| JP6321131B2 JP6321131B2 (ja) | 2018-05-09 |
Family
ID=60945772
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016256790A Active JP6321131B2 (ja) | 2016-02-12 | 2016-12-28 | アムロジピン含有配合錠の溶出性改善方法 |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JP6321131B2 (enExample) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP7425560B2 (ja) * | 2018-08-10 | 2024-01-31 | アリナミン製薬株式会社 | 固形製剤の製造方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5421945B2 (ja) * | 2010-03-10 | 2014-02-19 | 大日本住友製薬株式会社 | イルベサルタンとアムロジピンまたはその塩を含有する医薬組成物 |
| JP6041591B2 (ja) * | 2011-09-13 | 2016-12-14 | 大日本住友製薬株式会社 | イルベサルタンとアムロジピンまたはその塩を含有する安定化された医薬組成物 |
| JP6245677B2 (ja) * | 2012-01-20 | 2017-12-13 | ニプロ株式会社 | 口腔内崩壊錠 |
| JP6199922B2 (ja) * | 2015-03-20 | 2017-09-20 | 大原薬品工業株式会社 | 化学的な安定性が向上したイルベサルタン含有錠剤 |
-
2016
- 2016-12-28 JP JP2016256790A patent/JP6321131B2/ja active Active
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