JP2013520428A5 - - Google Patents

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Publication number
JP2013520428A5
JP2013520428A5 JP2012553986A JP2012553986A JP2013520428A5 JP 2013520428 A5 JP2013520428 A5 JP 2013520428A5 JP 2012553986 A JP2012553986 A JP 2012553986A JP 2012553986 A JP2012553986 A JP 2012553986A JP 2013520428 A5 JP2013520428 A5 JP 2013520428A5
Authority
JP
Japan
Prior art keywords
sulfonamido
acetic acid
methyl
dimethylchroman
biphenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP2012553986A
Other languages
English (en)
Japanese (ja)
Other versions
JP2013520428A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2011/025041 external-priority patent/WO2011103156A1/en
Publication of JP2013520428A publication Critical patent/JP2013520428A/ja
Publication of JP2013520428A5 publication Critical patent/JP2013520428A5/ja
Ceased legal-status Critical Current

Links

JP2012553986A 2010-02-19 2011-02-16 ジアシルグリセロールリパーゼの阻害剤として使用するためのグリシンクロマン−6−スルホンアミド Ceased JP2013520428A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US30602310P 2010-02-19 2010-02-19
US61/306,023 2010-02-19
PCT/US2011/025041 WO2011103156A1 (en) 2010-02-19 2011-02-16 Glycine chroman-6-sulfonamides for use as inhibitors of diacylglycerol lipase

Publications (2)

Publication Number Publication Date
JP2013520428A JP2013520428A (ja) 2013-06-06
JP2013520428A5 true JP2013520428A5 (cg-RX-API-DMAC10.html) 2014-04-03

Family

ID=43743459

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012553986A Ceased JP2013520428A (ja) 2010-02-19 2011-02-16 ジアシルグリセロールリパーゼの阻害剤として使用するためのグリシンクロマン−6−スルホンアミド

Country Status (5)

Country Link
US (1) US8354548B2 (cg-RX-API-DMAC10.html)
EP (1) EP2536704B1 (cg-RX-API-DMAC10.html)
JP (1) JP2013520428A (cg-RX-API-DMAC10.html)
CN (1) CN102858760A (cg-RX-API-DMAC10.html)
WO (1) WO2011103156A1 (cg-RX-API-DMAC10.html)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3095787A1 (en) * 2015-05-22 2016-11-23 Universiteit Leiden Pharmaceutically active compounds as dag-lipase inhibitors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5614649A (en) * 1994-11-14 1997-03-25 Cephalon, Inc. Multicatalytic protease inhibitors
CZ20012294A3 (cs) * 1998-12-22 2001-12-12 F. Hoffmann-La Roche Ag Sulfonamidové hydroxamáty
EP1160248A1 (en) * 2000-05-31 2001-12-05 Pfizer Inc. N-(Isoxazol-5-yl)-sulfonamide derivatives and their use as endothelin antagonists
JP4114859B2 (ja) * 2002-01-09 2008-07-09 松下電器産業株式会社 動きベクトル符号化方法および動きベクトル復号化方法
WO2006066756A1 (en) * 2004-12-21 2006-06-29 F. Hoffmann-La Roche Ag Chroman derivatives and uses thereof in the treatment of cns disorders
CN101300246A (zh) * 2005-11-03 2008-11-05 弗·哈夫曼-拉罗切有限公司 作为5-ht6抑制剂的芳基磺酰基色满类化合物作为蛋白激酶抑制剂的吲哚基马来酰亚胺衍生物

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