JP2013520428A5 - - Google Patents
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- Publication number
- JP2013520428A5 JP2013520428A5 JP2012553986A JP2012553986A JP2013520428A5 JP 2013520428 A5 JP2013520428 A5 JP 2013520428A5 JP 2012553986 A JP2012553986 A JP 2012553986A JP 2012553986 A JP2012553986 A JP 2012553986A JP 2013520428 A5 JP2013520428 A5 JP 2013520428A5
- Authority
- JP
- Japan
- Prior art keywords
- sulfonamido
- acetic acid
- methyl
- dimethylchroman
- biphenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US30602310P | 2010-02-19 | 2010-02-19 | |
| US61/306,023 | 2010-02-19 | ||
| PCT/US2011/025041 WO2011103156A1 (en) | 2010-02-19 | 2011-02-16 | Glycine chroman-6-sulfonamides for use as inhibitors of diacylglycerol lipase |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013520428A JP2013520428A (ja) | 2013-06-06 |
| JP2013520428A5 true JP2013520428A5 (cg-RX-API-DMAC10.html) | 2014-04-03 |
Family
ID=43743459
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012553986A Ceased JP2013520428A (ja) | 2010-02-19 | 2011-02-16 | ジアシルグリセロールリパーゼの阻害剤として使用するためのグリシンクロマン−6−スルホンアミド |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US8354548B2 (cg-RX-API-DMAC10.html) |
| EP (1) | EP2536704B1 (cg-RX-API-DMAC10.html) |
| JP (1) | JP2013520428A (cg-RX-API-DMAC10.html) |
| CN (1) | CN102858760A (cg-RX-API-DMAC10.html) |
| WO (1) | WO2011103156A1 (cg-RX-API-DMAC10.html) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3095787A1 (en) * | 2015-05-22 | 2016-11-23 | Universiteit Leiden | Pharmaceutically active compounds as dag-lipase inhibitors |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5614649A (en) * | 1994-11-14 | 1997-03-25 | Cephalon, Inc. | Multicatalytic protease inhibitors |
| CZ20012294A3 (cs) * | 1998-12-22 | 2001-12-12 | F. Hoffmann-La Roche Ag | Sulfonamidové hydroxamáty |
| EP1160248A1 (en) * | 2000-05-31 | 2001-12-05 | Pfizer Inc. | N-(Isoxazol-5-yl)-sulfonamide derivatives and their use as endothelin antagonists |
| JP4114859B2 (ja) * | 2002-01-09 | 2008-07-09 | 松下電器産業株式会社 | 動きベクトル符号化方法および動きベクトル復号化方法 |
| WO2006066756A1 (en) * | 2004-12-21 | 2006-06-29 | F. Hoffmann-La Roche Ag | Chroman derivatives and uses thereof in the treatment of cns disorders |
| CN101300246A (zh) * | 2005-11-03 | 2008-11-05 | 弗·哈夫曼-拉罗切有限公司 | 作为5-ht6抑制剂的芳基磺酰基色满类化合物作为蛋白激酶抑制剂的吲哚基马来酰亚胺衍生物 |
-
2011
- 2011-02-11 US US13/025,674 patent/US8354548B2/en active Active
- 2011-02-16 CN CN2011800198854A patent/CN102858760A/zh active Pending
- 2011-02-16 EP EP11705776.0A patent/EP2536704B1/en not_active Not-in-force
- 2011-02-16 JP JP2012553986A patent/JP2013520428A/ja not_active Ceased
- 2011-02-16 WO PCT/US2011/025041 patent/WO2011103156A1/en not_active Ceased
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