JP2011509296A5 - - Google Patents
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- JP2011509296A5 JP2011509296A5 JP2010542280A JP2010542280A JP2011509296A5 JP 2011509296 A5 JP2011509296 A5 JP 2011509296A5 JP 2010542280 A JP2010542280 A JP 2010542280A JP 2010542280 A JP2010542280 A JP 2010542280A JP 2011509296 A5 JP2011509296 A5 JP 2011509296A5
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- carboxylic acid
- amide
- ethyl
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| US12424008P | 2008-04-14 | 2008-04-14 | |
| PCT/US2009/000150 WO2009089057A1 (en) | 2008-01-09 | 2009-01-09 | Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same |
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| JP5699090B2 (ja) | 2008-12-30 | 2015-04-08 | バーテックス ファーマシューティカルズ インコーポレイテッドＶｅｒｔｅｘ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｉｎｃｏｒｐｏｒａｔｅｄ | 嚢胞性線維症膜コンダクタンス調節因子のモジュレーター |
| EP2447263A1 (en) | 2010-09-27 | 2012-05-02 | Bioprojet | Benzazole derivatives as histamine H4 receptor ligands |
| FI3609868T3 (fi) | 2017-03-13 | 2023-11-22 | Raqualia Pharma Inc | Tetrahydrokinoliinijohdannaisia P2X7-reseptorin antagonisteina |
| JP6994061B2 (ja) | 2019-02-15 | 2022-01-14 | ノバルティス アーゲー | ４－（７－ヒドロキシ－２－イソプロピル－４－オキソ－４ｈ－キナゾリン－３－イル）－ベンゾニトリルの製剤 |
| KR20210129677A (ko) | 2019-02-15 | 2021-10-28 | 노파르티스 아게 | 안구 표면 통증의 치료 방법 |
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| WO2004110986A1 (ja) * | 2003-06-12 | 2004-12-23 | Astellas Pharma Inc. | ベンズアミド誘導体又はその塩 |
| FR2880625B1 (fr) * | 2005-01-07 | 2007-03-09 | Sanofi Aventis Sa | Derives de n-(heteroaryl)-1h-indole-2-carboxamides, leur preparation et leur application en therapeutique |
| BRPI0709596A2 (pt) | 2006-03-16 | 2011-07-19 | Renovis Inc | compostos bicicloeteroarila como moduladores de p2x7 e seus usos |
| WO2007133637A2 (en) * | 2006-05-10 | 2007-11-22 | Renovis, Inc. | Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same |
| WO2008007211A1 (en) * | 2006-07-11 | 2008-01-17 | Pfizer Japan Inc. | Substituted n-bicyclicalkyl bicyclic carboxyamide compounds |
| WO2008090434A1 (en) | 2007-01-25 | 2008-07-31 | Pfizer Japan Inc. | Substituted n-bicyclicalkyl bicyclic carboxyamide compounds |
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- 2009-01-09 CA CA2707441A patent/CA2707441A1/en not_active Abandoned
- 2009-01-09 EP EP09700264A patent/EP2240467B1/en not_active Not-in-force
- 2009-01-09 WO PCT/US2009/000150 patent/WO2009089057A1/en not_active Ceased
- 2009-01-09 US US12/811,972 patent/US8163901B2/en not_active Expired - Fee Related
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2012
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