JP2008514563A5 - - Google Patents

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Publication number
JP2008514563A5
JP2008514563A5 JP2007532823A JP2007532823A JP2008514563A5 JP 2008514563 A5 JP2008514563 A5 JP 2008514563A5 JP 2007532823 A JP2007532823 A JP 2007532823A JP 2007532823 A JP2007532823 A JP 2007532823A JP 2008514563 A5 JP2008514563 A5 JP 2008514563A5
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JP
Japan
Prior art keywords
mic
test results
table below
antibacterial test
typical antibacterial
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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JP2007532823A
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Japanese (ja)
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JP4887297B2 (en
JP2008514563A (en
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Priority claimed from PCT/EP2005/010154 external-priority patent/WO2006032466A2/en
Publication of JP2008514563A publication Critical patent/JP2008514563A/en
Publication of JP2008514563A5 publication Critical patent/JP2008514563A5/ja
Application granted granted Critical
Publication of JP4887297B2 publication Critical patent/JP4887297B2/en
Expired - Fee Related legal-status Critical Current
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Description

典型的な抗菌性の試験結果を以下の表に示してある（ｍｇ／ｌでのＭＩＣ）。

Figure 2008514563
Typical antibacterial test results are shown in the table below (MIC in mg / l).
Figure 2008514563
JP2007532823A 2004-09-24 2005-09-20 New bicyclic antibiotics Expired - Fee Related JP4887297B2 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP2004010762 2004-09-24
EPPCT/EP2004/010762 2004-09-24
EP2005007731 2005-07-15
EPPCT/EP2005/007731 2005-07-15
PCT/EP2005/010154 WO2006032466A2 (en) 2004-09-24 2005-09-20 New bicyclic antibiotics

Publications (3)

Publication Number Publication Date
JP2008514563A JP2008514563A (en) 2008-05-08
JP2008514563A5 true JP2008514563A5 (en) 2011-12-08
JP4887297B2 JP4887297B2 (en) 2012-02-29

Family

ID=36090370

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007532823A Expired - Fee Related JP4887297B2 (en) 2004-09-24 2005-09-20 New bicyclic antibiotics

Country Status (5)

Country Link
JP (1) JP4887297B2 (en)
AR (1) AR050958A1 (en)
CA (1) CA2580621A1 (en)
TW (1) TW200615267A (en)
WO (1) WO2006032466A2 (en)

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CL2008001003A1 (en) 2007-04-11 2008-10-17 Actelion Pharmaceuticals Ltd COMPOUNDS DERIVED FROM OXAZOLIDINONA; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; AND ITS USE TO PREPARE A MEDICINAL PRODUCT TO TREAT A BACTERIAL INFECTION.
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US8012961B2 (en) 2008-04-15 2011-09-06 Actelion Pharmaceutical Ltd. Tricyclic antibiotics
KR101658681B1 (en) 2008-06-03 2016-09-21 액테리온 파마슈티칼 리미티드 [4-(1-amino-ethyl)-cyclohexyl]-methyl-amine and [6-(1-amino-ethyl)-tetrahydro-pyran-3-yl]-methyl-amine derivatives as antibacterials
US8466168B2 (en) 2008-08-04 2013-06-18 Actellon Pharmaceuticals Ltd. Tricyclic alkylaminomethyloxazolidinone derivatives
PT2344495E (en) 2008-10-07 2015-04-01 Actelion Pharmaceuticals Ltd Tricyclic oxazolidinone antibiotic compounds
EP2352734A1 (en) 2008-10-17 2011-08-10 Glaxo Group Limited Tricyclic nitrogen compounds used as antibacterials
NZ591914A (en) 2008-11-17 2013-04-26 Hoffmann La Roche Naphthylacetic acids
US8211890B2 (en) 2008-12-12 2012-07-03 Actelion Pharmaceuticals 5-amino-2-(1-hydroxy-ethyl)-tetrahydropyran derivatives
ES2561631T3 (en) 2009-01-15 2016-02-29 Glaxo Group Limited Naphthyridine-2 (1H) -one compounds useful as antibacterial agents
CN102361863B (en) 2009-01-21 2014-12-03 巴斯利尔药物股份公司 Novel bicyclic antibiotics
AR076222A1 (en) 2009-04-09 2011-05-26 Actelion Pharmaceuticals Ltd DERIVATIVES 2-HYDROXIETIL-1H-QUINOLIN-ONA AND ITS AZAISOTHERAL ANALOGS WITH ANTIBACTERIAL ACTIVITY AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
WO2012042539A2 (en) 2010-09-28 2012-04-05 Panacea Biotec Ltd Novel bicyclic compounds
RU2612534C2 (en) 2011-03-10 2017-03-09 Дайити Санкио Компани, Лимитед Dispiropyrrolidine derivatives
EP2685828A4 (en) * 2011-03-17 2014-08-13 Merck Sharp & Dohme Substituted 3-azabicyclo[3.1.0]hexane derivatives useful as ccr2 antagonists
JP6023800B2 (en) * 2011-06-17 2016-11-09 アストラゼネカ アクチボラグ Process for producing a heterocyclic compound containing trans-7-oxo-6- (sulfooxy) -1,6-diazabicyclo [3,2,1] octane-2-carboxamide and a salt thereof
EP2723737A1 (en) * 2011-06-27 2014-04-30 Kyorin Pharmaceutical Co., Ltd. Bridged bicyclic compounds for the treatment of bacterial infections
US8470884B2 (en) 2011-11-09 2013-06-25 Hoffmann-La Roche Inc. Alkenyl naphthylacetic acids
EP2785721A1 (en) 2011-11-30 2014-10-08 Actelion Pharmaceuticals Ltd. 3,7-disubstituted octahydro-2h-pyrido[4,3-e][1,3]oxazin-2-one antibiotics
SG11201700566SA (en) 2014-08-22 2017-03-30 Glaxosmithkline Ip Dev Ltd Tricyclic nitrogen containing compounds for treating neisseria gonorrhoea infection
UY36851A (en) 2015-08-16 2017-03-31 Glaxosmithkline Ip Dev Ltd COMPOUNDS FOR USE IN ANTIBACTERIAL APPLICATIONS
JP7382308B2 (en) * 2017-09-01 2023-11-16 デナリ セラピューティクス インコーポレイテッド Compounds, compositions and methods
UA126589C2 (en) 2017-09-14 2022-11-02 Даїті Санкіо Компані, Лімітед Compound having cyclic structure
CN109082280B (en) * 2018-11-05 2020-07-28 宁夏中星显示材料有限公司 Preparation method of liquid crystal material

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DE10316081A1 (en) * 2003-04-08 2004-10-21 Morphochem AG Aktiengesellschaft für kombinatorische Chemie New compounds with antibacterial activity
EP1778688A1 (en) * 2004-07-22 2007-05-02 Glaxo Group Limited Antibacterial agents
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