JP2007526291A - アデノシン受容体アゴニスト - Google Patents
アデノシン受容体アゴニスト Download PDFInfo
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- JP2007526291A JP2007526291A JP2007501345A JP2007501345A JP2007526291A JP 2007526291 A JP2007526291 A JP 2007526291A JP 2007501345 A JP2007501345 A JP 2007501345A JP 2007501345 A JP2007501345 A JP 2007501345A JP 2007526291 A JP2007526291 A JP 2007526291A
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Applications Claiming Priority (10)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/GB2004/000902 WO2004079329A2 (en) | 2003-03-07 | 2004-03-05 | Identification of therapeutic compounds |
| GB0405012A GB0405012D0 (en) | 2004-03-05 | 2004-03-05 | Therapeutic compounds |
| GBGB0405009.2A GB0405009D0 (en) | 2004-03-05 | 2004-03-05 | Analgesics |
| GB0412262A GB0412262D0 (en) | 2004-06-02 | 2004-06-02 | Use of compounds for the treatment of pain |
| GB0412261A GB0412261D0 (en) | 2004-06-02 | 2004-06-02 | Analgesics |
| GB0413627A GB0413627D0 (en) | 2004-06-18 | 2004-06-18 | Analgesics |
| GB0419718A GB0419718D0 (en) | 2004-09-06 | 2004-09-06 | Therapeutic compounds |
| GB0420063A GB0420063D0 (en) | 2004-09-09 | 2004-09-09 | Therapeutic compounds |
| GB0420615A GB0420615D0 (en) | 2004-09-16 | 2004-09-16 | Therapeutic compounds |
| PCT/GB2005/000800 WO2005084653A2 (en) | 2004-03-05 | 2005-03-04 | Adenosine receptor agonists |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2011280200A Division JP2012102114A (ja) | 2004-03-05 | 2011-12-21 | アデノシン受容体アゴニスト |
Publications (2)
| Publication Number | Publication Date |
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| JP2007526291A true JP2007526291A (ja) | 2007-09-13 |
| JP2007526291A5 JP2007526291A5 (enExample) | 2008-04-17 |
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| Application Number | Title | Priority Date | Filing Date |
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| JP2007501345A Pending JP2007526291A (ja) | 2004-03-05 | 2005-03-04 | アデノシン受容体アゴニスト |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20080221060A1 (enExample) |
| EP (1) | EP1749016A2 (enExample) |
| JP (1) | JP2007526291A (enExample) |
| KR (1) | KR20070004792A (enExample) |
| AU (1) | AU2005218997B2 (enExample) |
| BR (1) | BRPI0508488A (enExample) |
| CA (1) | CA2557285A1 (enExample) |
| EA (2) | EA014425B1 (enExample) |
| MX (1) | MXPA06010075A (enExample) |
| NO (1) | NO20064365L (enExample) |
| SG (1) | SG144146A1 (enExample) |
| WO (1) | WO2005084653A2 (enExample) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2011509305A (ja) * | 2008-01-09 | 2011-03-24 | ピージーエックスヘルス、リミテッド、ライアビリティー、カンパニー | Ａ２ａｒアゴニストによる神経障害性疼痛の髄腔内治療 |
| JP2014532636A (ja) * | 2011-10-24 | 2014-12-08 | ユニヴエルシテ・ピエール・エ・マリー・キユリー・パリ・シス | ウイルス感染の処置のためのヌクレオシドアナログおよび該処置に対する感受性を評価するための方法 |
Families Citing this family (32)
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|---|---|---|---|---|
| EP1434782A2 (en) | 2001-10-01 | 2004-07-07 | University of Virginia Patent Foundation | 2-propynyl adenosine analogs having a2a agonist activity and compositions thereof |
| GB0228723D0 (en) | 2002-12-09 | 2003-01-15 | Cambridge Biotechnology Ltd | Treatment of pain |
| EP1746885A4 (en) * | 2004-05-03 | 2010-09-08 | Univ Virginia | AGONISTS OF A2A ADENOSINE RECEPTORS FOR THE TREATMENT OF NEEDLE INJURY IN DIABETES |
| GT200500281A (es) | 2004-10-22 | 2006-04-24 | Novartis Ag | Compuestos organicos. |
| CA2586845A1 (en) * | 2004-11-08 | 2006-05-11 | Can-Fite Biopharma Ltd. | Therapeutic treatment of accelerated bone resorption |
| GB0500785D0 (en) | 2005-01-14 | 2005-02-23 | Novartis Ag | Organic compounds |
| CN1947717B (zh) * | 2005-10-14 | 2012-09-26 | 卓敏 | 选择性抑制腺苷酸环化酶1的化合物在制备用于治疗神经性疼痛和炎性疼痛的药物中的应用 |
| US20070183995A1 (en) * | 2006-02-09 | 2007-08-09 | Conopco, Inc., D/B/A Unilever | Compounds useful as agonists of A2A adenosine receptors, cosmetic compositions with A2A agonists and a method for using the same |
| US8178509B2 (en) | 2006-02-10 | 2012-05-15 | University Of Virginia Patent Foundation | Method to treat sickle cell disease |
| GB0607950D0 (en) | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| GB0607953D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| PE20080361A1 (es) | 2006-04-21 | 2008-06-03 | Novartis Ag | Compuestos derivados de purina como activadores del receptor de adenosina a2a |
| US8188063B2 (en) | 2006-06-19 | 2012-05-29 | University Of Virginia Patent Foundation | Use of adenosine A2A modulators to treat spinal cord injury |
| JP2009541438A (ja) * | 2006-06-27 | 2009-11-26 | ビオヴィトルム・アクチボラゲット（プブリクト） | 治療用化合物 |
| EP2081932A2 (en) | 2006-06-27 | 2009-07-29 | BIOVITRUM AB (publ) | 2-o'-methyladenosine derivatives and their use as agonists or antagonists of an adenosine receptor |
| CA2657973A1 (en) | 2006-06-27 | 2008-01-03 | Biovitrum Ab (Publ) | Therapeutic compounds |
| EP1889846A1 (en) | 2006-07-13 | 2008-02-20 | Novartis AG | Purine derivatives as A2a agonists |
| EP1903044A1 (en) | 2006-09-14 | 2008-03-26 | Novartis AG | Adenosine Derivatives as A2A Receptor Agonists |
| WO2009061516A1 (en) * | 2007-11-08 | 2009-05-14 | New York University School Of Medicine | Medical implants containing adenosine receptor agonists and methods for inhibiting medical implant loosening |
| US8058259B2 (en) | 2007-12-20 | 2011-11-15 | University Of Virginia Patent Foundation | Substituted 4-{3-[6-amino-9-(3,4-dihydroxy-tetrahydro-furan-2-yl)-9H-purin-2-yl]-prop-2-ynyl}-piperidine-1-carboxylic acid esters as A2AR agonists |
| US20100160351A1 (en) * | 2008-12-19 | 2010-06-24 | Nuon Therapeutics, Inc. | Pharmaceutical compositions and methods for treating hyperuricemia and related disorders |
| WO2010071865A1 (en) | 2008-12-19 | 2010-06-24 | Nuon Therapeutics, Inc. | Pharmaceutical compositions and methods for treating hyperuricemia and related disorders |
| CA2766937A1 (en) * | 2009-07-09 | 2011-01-13 | Cbt Development Limited | Combined preparation for use as a medicament |
| WO2011032175A1 (en) | 2009-09-14 | 2011-03-17 | Nuon Therapeutics, Inc. | Combination formulations of tranilast and allopurinol and methods related thereto |
| CA2783859A1 (en) * | 2009-12-10 | 2011-06-16 | Institute Of Materia Medica, Chinese Academy Of Medical Sciences | N6-substituted adenosine derivatives and n6-substituted adenine derivatives and uses thereof |
| US20130109645A1 (en) * | 2010-03-31 | 2013-05-02 | The united States of America,as represented by Secretary,Dept.,of Health and Human Services | Adenosine receptor agonists for the treatment and prevention of vascular or joint capsule calcification disorders |
| KR20140059246A (ko) * | 2011-09-22 | 2014-05-15 | 화이자 인코포레이티드 | 피롤로피리미딘 및 퓨린 유도체 |
| US20160038526A1 (en) * | 2012-08-16 | 2016-02-11 | Thomas Jefferson University | Treatment of prostate cancer |
| US20150209379A1 (en) * | 2012-08-16 | 2015-07-30 | Thomas Jefferson University | Treatment of prostate cancer and hematologic neoplasms |
| EP2711008A1 (en) | 2012-09-19 | 2014-03-26 | Institut Univ. de Ciència i Tecnologia, S.A. | N6,N6-dimethyladenosine for use in treating or preventing primary and metastatic breast cancer |
| US9771390B2 (en) * | 2013-12-10 | 2017-09-26 | Scinopharm Taiwan, Ltd. | Process for the preparation of regadenoson |
| WO2018140734A1 (en) | 2017-01-27 | 2018-08-02 | Academia Sinica | Compound with analgesic effect for use in prevention and treatment of pain |
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| US5877180A (en) * | 1994-07-11 | 1999-03-02 | University Of Virginia Patent Foundation | Method for treating inflammatory diseases with A2a adenosine receptor agonists |
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| BE792155A (fr) * | 1971-12-01 | 1973-05-30 | Takeda Chemical Industries Ltd | Nouveaux derives de l'adenosine et leur procede de production |
| DE2359536C2 (de) * | 1972-12-08 | 1984-08-02 | Takeda Chemical Industries, Ltd., Osaka | 2,6-Diaminonebularinderivate |
| US4705758A (en) * | 1984-06-19 | 1987-11-10 | Warner-Lambert Company | Adenosine receptor assay and kit |
| US5013829A (en) * | 1989-04-26 | 1991-05-07 | University Of Iowa Research Foundation | Stable congener of 2',3'-dideoxyadenosine |
| US5679650A (en) * | 1993-11-24 | 1997-10-21 | Fukunaga; Atsuo F. | Pharmaceutical compositions including mixtures of an adenosine compound and a catecholamine |
| US5677290A (en) * | 1990-05-10 | 1997-10-14 | Fukunaga; Atsuo F. | Therapeutic use of adenosine compounds as surgical anesthetics |
| US6174873B1 (en) * | 1998-11-04 | 2001-01-16 | Supergen, Inc. | Oral administration of adenosine analogs |
| GB0228723D0 (en) * | 2002-12-09 | 2003-01-15 | Cambridge Biotechnology Ltd | Treatment of pain |
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| GB0305149D0 (en) * | 2003-03-07 | 2003-04-09 | Cambridge Biotechnology Ltd | Compounds for the treatment of pain |
| GB0305153D0 (en) * | 2003-03-07 | 2003-04-09 | Cambridge Biotechnology Ltd | Identification of therapeutic compounds |
| GB0328323D0 (en) * | 2003-12-05 | 2004-01-07 | Cambridge Biotechnology Ltd | Synthesis of 2-substituted adenosines |
| US20090131651A1 (en) * | 2003-12-05 | 2009-05-21 | Giles Albert Brown | Synthesis of 2-substituted adenosines |
| GB0401292D0 (en) * | 2004-01-21 | 2004-02-25 | Cambridge Biotechnology Ltd | Synthesis of spongosine |
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- 2005-03-04 WO PCT/GB2005/000800 patent/WO2005084653A2/en not_active Ceased
- 2005-03-04 US US10/598,520 patent/US20080221060A1/en not_active Abandoned
- 2005-03-04 EA EA200800538A patent/EA014425B1/ru not_active IP Right Cessation
- 2005-03-04 AU AU2005218997A patent/AU2005218997B2/en not_active Expired - Fee Related
- 2005-03-04 SG SG200804350-7A patent/SG144146A1/en unknown
- 2005-03-04 MX MXPA06010075A patent/MXPA06010075A/es unknown
- 2005-03-04 CA CA002557285A patent/CA2557285A1/en not_active Abandoned
- 2005-03-04 EP EP05717878A patent/EP1749016A2/en not_active Withdrawn
- 2005-03-04 JP JP2007501345A patent/JP2007526291A/ja active Pending
- 2005-03-04 BR BRPI0508488-1A patent/BRPI0508488A/pt not_active IP Right Cessation
- 2005-03-04 KR KR1020067020304A patent/KR20070004792A/ko not_active Ceased
- 2005-03-04 EA EA200601642A patent/EA011099B1/ru not_active IP Right Cessation
-
2006
- 2006-09-26 NO NO20064365A patent/NO20064365L/no not_active Application Discontinuation
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2011509305A (ja) * | 2008-01-09 | 2011-03-24 | ピージーエックスヘルス、リミテッド、ライアビリティー、カンパニー | Ａ２ａｒアゴニストによる神経障害性疼痛の髄腔内治療 |
| JP2014532636A (ja) * | 2011-10-24 | 2014-12-08 | ユニヴエルシテ・ピエール・エ・マリー・キユリー・パリ・シス | ウイルス感染の処置のためのヌクレオシドアナログおよび該処置に対する感受性を評価するための方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| SG144146A1 (en) | 2008-07-29 |
| EA200601642A1 (ru) | 2006-12-29 |
| EA200800538A1 (ru) | 2008-06-30 |
| CA2557285A1 (en) | 2005-09-15 |
| AU2005218997A1 (en) | 2005-09-15 |
| WO2005084653A2 (en) | 2005-09-15 |
| EA011099B1 (ru) | 2008-12-30 |
| US20080221060A1 (en) | 2008-09-11 |
| KR20070004792A (ko) | 2007-01-09 |
| BRPI0508488A (pt) | 2007-07-31 |
| EA014425B1 (ru) | 2010-12-30 |
| EP1749016A2 (en) | 2007-02-07 |
| NO20064365L (no) | 2006-11-22 |
| MXPA06010075A (es) | 2007-04-10 |
| AU2005218997B2 (en) | 2012-05-10 |
| WO2005084653A3 (en) | 2006-05-18 |
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