JP2002534996A - アルファ−コノトキシン・ペプチド - Google Patents
アルファ−コノトキシン・ペプチドInfo
- Publication number
- JP2002534996A JP2002534996A JP2000596032A JP2000596032A JP2002534996A JP 2002534996 A JP2002534996 A JP 2002534996A JP 2000596032 A JP2000596032 A JP 2000596032A JP 2000596032 A JP2000596032 A JP 2000596032A JP 2002534996 A JP2002534996 A JP 2002534996A
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- JP
- Japan
- Prior art keywords
- xaa
- lys
- tyr
- halo
- pro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
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- SRBFZHDQGSBBOR-UHFFFAOYSA-N beta-D-Pyranose-Lyxose Natural products OC1COC(O)C(O)C1O SRBFZHDQGSBBOR-UHFFFAOYSA-N 0.000 description 1
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- MGJXBDMLVWIYOQ-UHFFFAOYSA-N methylazanide Chemical compound [NH-]C MGJXBDMLVWIYOQ-UHFFFAOYSA-N 0.000 description 1
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- 125000002950 monocyclic group Chemical group 0.000 description 1
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- 244000062645 predators Species 0.000 description 1
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/43504—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from invertebrates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biophysics (AREA)
- Gastroenterology & Hepatology (AREA)
- Zoology (AREA)
- Biochemistry (AREA)
- Toxicology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Tropical Medicine & Parasitology (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US11838199P | 1999-01-29 | 1999-01-29 | |
| US60/118,381 | 1999-01-29 | ||
| PCT/US2000/001979 WO2000044776A1 (en) | 1999-01-29 | 2000-01-28 | Alpha-conotoxin peptides |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2002534996A true JP2002534996A (ja) | 2002-10-22 |
| JP2002534996A5 JP2002534996A5 (https=) | 2007-03-29 |
Family
ID=22378229
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2000596032A Pending JP2002534996A (ja) | 1999-01-29 | 2000-01-28 | アルファ−コノトキシン・ペプチド |
Country Status (5)
| Country | Link |
|---|---|
| EP (1) | EP1147130A4 (https=) |
| JP (1) | JP2002534996A (https=) |
| AU (1) | AU770076B2 (https=) |
| CA (2) | CA2743116C (https=) |
| WO (1) | WO2000044776A1 (https=) |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2009545526A (ja) * | 2006-07-18 | 2009-12-24 | ユニバーシティ・オブ・ユタ・リサーチ・ファウンデーション | 痛みの処置方法および鎮痛化合物のスクリーニング方法 |
| JP2015532637A (ja) * | 2012-08-07 | 2015-11-12 | ハイナン ユニバーシティ | α−コノトキシンペプチド、その医薬組成物及びそれらの使用 |
| US9284358B2 (en) | 2006-07-18 | 2016-03-15 | University Of Utah Research Foundation | Conotoxin peptides |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2002245934B2 (en) * | 2001-03-29 | 2008-05-01 | John Down | Alpha conotoxin peptides with analgesic properties |
| AUPR409401A0 (en) | 2001-03-29 | 2001-04-26 | University Of Melbourne, The | Analgesic compound |
| CA2661014A1 (en) * | 2006-08-17 | 2008-02-21 | Eribis Pharmaceuticals Ab | Cardioprotective compounds |
| CN103483439B (zh) | 2012-06-15 | 2015-09-16 | 海南大学 | αO-超家族芋螺毒素肽、其药物组合物及用途 |
| CN121471320B (zh) * | 2026-01-12 | 2026-03-17 | 中国海洋大学 | 一种靶向trpv1的多肽及其应用 |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH10509415A (ja) * | 1993-10-19 | 1998-09-14 | ユニバーシティ オブ ユタ リサーチ ファウンデーション | コノトキシン（ｃｏｎｏｔｏｘｉｎ）ペプチド |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5595972A (en) * | 1993-06-29 | 1997-01-21 | University Of Utah Research Foundation | Conotoxin peptides |
| US5432155A (en) * | 1993-06-29 | 1995-07-11 | The Salk Institute For Biological Studies | Conotoxins I |
| US5739276A (en) * | 1994-10-07 | 1998-04-14 | University Of Utah Research Foundation | Conotoxin peptides |
| US5719264A (en) * | 1994-10-07 | 1998-02-17 | Univ. Of Utah Research Foundation | Conotoxin peptides |
| US5670622A (en) * | 1996-02-15 | 1997-09-23 | University Of Utah Research Foundation | Conotoxin peptide PIIIA |
| US5672682A (en) * | 1996-03-18 | 1997-09-30 | University Of Utah Research Foundation | Conotoxin peptide PVIIA |
| WO1998022126A1 (en) * | 1996-11-18 | 1998-05-28 | University Of Utah Research Foundation | USE OF CONOTOXIN PEPTIDES ImI AND MII AS CARDIOVASCULAR AGENTS |
| US5780433A (en) * | 1996-12-06 | 1998-07-14 | University Of Utah Research Foundation | Use of α-conotoxin MII to treat disorders resulting from nicotine stimulated dopamine release |
| US5889147A (en) * | 1997-01-17 | 1999-03-30 | University Of Utah Research Foundation | Bromo-tryptophan conopeptides |
| US5866682A (en) * | 1997-05-15 | 1999-02-02 | University Of Utah Research Foundation | Conopeptides AuIA, AuIB and AuIC |
| US5969096A (en) * | 1998-06-26 | 1999-10-19 | The Salk Institute For Biological Studies | Conotoxin peptides |
-
2000
- 2000-01-28 JP JP2000596032A patent/JP2002534996A/ja active Pending
- 2000-01-28 WO PCT/US2000/001979 patent/WO2000044776A1/en not_active Ceased
- 2000-01-28 CA CA2743116A patent/CA2743116C/en not_active Expired - Fee Related
- 2000-01-28 EP EP00908382A patent/EP1147130A4/en not_active Withdrawn
- 2000-01-28 AU AU29735/00A patent/AU770076B2/en not_active Ceased
- 2000-01-28 CA CA2361534A patent/CA2361534C/en not_active Expired - Fee Related
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH10509415A (ja) * | 1993-10-19 | 1998-09-14 | ユニバーシティ オブ ユタ リサーチ ファウンデーション | コノトキシン（ｃｏｎｏｔｏｘｉｎ）ペプチド |
Non-Patent Citations (2)
| Title |
|---|
| JPN6009054683, Ｊ． Ｂｉｏｌ． Ｃｈｅｍ． （１９９８） ｖｏｌ．２７３， ｎｏ．２５， ｐ．１５６６７−１５６７４ * |
| JPN6009054685, Ｊ． Ｂｉｏｌ． Ｃｈｅｍ． （１９９６） ｖｏｌ．２７１， ｎｏ．１３， ｐ．７５２２−７５２８ * |
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2009545526A (ja) * | 2006-07-18 | 2009-12-24 | ユニバーシティ・オブ・ユタ・リサーチ・ファウンデーション | 痛みの処置方法および鎮痛化合物のスクリーニング方法 |
| US9284358B2 (en) | 2006-07-18 | 2016-03-15 | University Of Utah Research Foundation | Conotoxin peptides |
| US9717775B2 (en) | 2006-07-18 | 2017-08-01 | University Of Utah Research Foundation | Methods for treating pain and screening analgesic compounds |
| JP2015532637A (ja) * | 2012-08-07 | 2015-11-12 | ハイナン ユニバーシティ | α−コノトキシンペプチド、その医薬組成物及びそれらの使用 |
Also Published As
| Publication number | Publication date |
|---|---|
| CA2743116C (en) | 2016-06-21 |
| WO2000044776A1 (en) | 2000-08-03 |
| CA2361534A1 (en) | 2000-08-03 |
| EP1147130A4 (en) | 2004-09-29 |
| AU2973500A (en) | 2000-08-18 |
| AU770076B2 (en) | 2004-02-12 |
| CA2361534C (en) | 2011-08-30 |
| EP1147130A1 (en) | 2001-10-24 |
| CA2743116A1 (en) | 2000-08-03 |
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