ITSA20110014A1 - Sintesi e attività biologica di derivati n-alchilcarbazoli come inibitori di stat3 - Google Patents

Sintesi e attività biologica di derivati n-alchilcarbazoli come inibitori di stat3

Info

Publication number
ITSA20110014A1
ITSA20110014A1 IT000014A ITSA20110014A ITSA20110014A1 IT SA20110014 A1 ITSA20110014 A1 IT SA20110014A1 IT 000014 A IT000014 A IT 000014A IT SA20110014 A ITSA20110014 A IT SA20110014A IT SA20110014 A1 ITSA20110014 A1 IT SA20110014A1
Authority
IT
Italy
Prior art keywords
alchilcarbazol
derivatives
biological activity
stat3 inhibitors
stat3
Prior art date
Application number
IT000014A
Other languages
English (en)
Inventor
Longo Pasquale
Carmela Saturnino
Original Assignee
Univ Degli Studi Salerno
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Degli Studi Salerno filed Critical Univ Degli Studi Salerno
Priority to IT000014A priority Critical patent/ITSA20110014A1/it
Publication of ITSA20110014A1 publication Critical patent/ITSA20110014A1/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/80—[b, c]- or [b, d]-condensed
    • C07D209/82—Carbazoles; Hydrogenated carbazoles
    • C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
IT000014A 2011-06-16 2011-06-16 Sintesi e attività biologica di derivati n-alchilcarbazoli come inibitori di stat3 ITSA20110014A1 (it)

Priority Applications (1)

Application Number Priority Date Filing Date Title
IT000014A ITSA20110014A1 (it) 2011-06-16 2011-06-16 Sintesi e attività biologica di derivati n-alchilcarbazoli come inibitori di stat3

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT000014A ITSA20110014A1 (it) 2011-06-16 2011-06-16 Sintesi e attività biologica di derivati n-alchilcarbazoli come inibitori di stat3

Publications (1)

Publication Number Publication Date
ITSA20110014A1 true ITSA20110014A1 (it) 2012-12-17

Family

ID=44898331

Family Applications (1)

Application Number Title Priority Date Filing Date
IT000014A ITSA20110014A1 (it) 2011-06-16 2011-06-16 Sintesi e attività biologica di derivati n-alchilcarbazoli come inibitori di stat3

Country Status (1)

Country Link
IT (1) ITSA20110014A1 (it)

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6468996B1 (en) * 1998-10-21 2002-10-22 Novo Nordisk A/S Substituted hetero-polycyclic compounds as PPARα and PPARγ activators
WO2008021745A2 (en) * 2006-08-16 2008-02-21 Itherx Pharmaceuticals, Inc. Hepatitis c virus entry inhibitors

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6468996B1 (en) * 1998-10-21 2002-10-22 Novo Nordisk A/S Substituted hetero-polycyclic compounds as PPARα and PPARγ activators
WO2008021745A2 (en) * 2006-08-16 2008-02-21 Itherx Pharmaceuticals, Inc. Hepatitis c virus entry inhibitors

Non-Patent Citations (5)

* Cited by examiner, † Cited by third party
Title
ARBISER JACK L ET AL: "Carbazole is a naturally occurring inhibitor of angiogenesis and inflammation isolated from antipsoriatic coal tar", JOURNAL OF INVESTIGATIVE DERMATOLOGY, NATURE PUBLISHING GROUP, GB, vol. 126, no. 6, 1 June 2006 (2006-06-01), pages 1396 - 1402, XP008125101, ISSN: 0022-202X, [retrieved on 20060413] *
JIANFENG PAN ET AL: "Synthesis of Carrier-Transporting Dendrimers with Perylenebis(dicarboximide)s as a Luminescent Core", EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, vol. 2006, no. 4, 1 February 2006 (2006-02-01), pages 986 - 1001, XP055011866, ISSN: 1434-193X, DOI: 10.1002/ejoc.200500642 *
LI S ET AL: "Antenna-functionalized dendritic beta-diketonates and europium complexes: synthetic approaches to generation growth", TETRAHEDRON, ELSEVIER SCIENCE PUBLISHERS, AMSTERDAM, NL, vol. 62, no. 21, 22 May 2006 (2006-05-22), pages 5035 - 5048, XP025001960, ISSN: 0040-4020, [retrieved on 20060522], DOI: 10.1016/J.TET.2006.03.052 *
TAE WOO KIM ET AL: "Molecular Tripods Showing Fluorescence Enhancement upon Binding to Streptavidin", ORGANIC LETTERS, vol. 7, no. 1, 1 January 2005 (2005-01-01), pages 111 - 114, XP055011892, ISSN: 1523-7060, DOI: 10.1021/ol047801h *
YOUXUAN ZHENG ET AL: "Synthesis and Photoluminescence Properties of Heteroleptic Europium(III) Complexes with Appended Carbazole Units", EUROPEAN JOURNAL OF INORGANIC CHEMISTRY, vol. 2008, no. 12, 1 April 2008 (2008-04-01), pages 2075 - 2080, XP055011889, ISSN: 1434-1948, DOI: 10.1002/ejic.200701257 *

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