ITMI962385A0 - Diaril-ciclometilenpirazoli farmacologicamente attivi procedimento per prepararli e composizioni farmaceutiche che li contengono - Google Patents

Diaril-ciclometilenpirazoli farmacologicamente attivi procedimento per prepararli e composizioni farmaceutiche che li contengono

Info

Publication number
ITMI962385A0
ITMI962385A0 IT96MI002385A ITMI962385A ITMI962385A0 IT MI962385 A0 ITMI962385 A0 IT MI962385A0 IT 96MI002385 A IT96MI002385 A IT 96MI002385A IT MI962385 A ITMI962385 A IT MI962385A IT MI962385 A0 ITMI962385 A0 IT MI962385A0
Authority
IT
Italy
Prior art keywords
cyclomethylenpyrazoles
preparing
procedure
contain
pharmaceutical compositions
Prior art date
Application number
IT96MI002385A
Other languages
English (en)
Inventor
Marilena Giannangeli
Mauro Tomaselli
Mario Pinza
Original Assignee
Angelini Ricerche Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Angelini Ricerche Spa filed Critical Angelini Ricerche Spa
Priority to IT96MI002385A priority Critical patent/IT1287174B1/it
Publication of ITMI962385A0 publication Critical patent/ITMI962385A0/it
Priority to PCT/EP1997/006398 priority patent/WO1998022442A2/en
Priority to AU55526/98A priority patent/AU5552698A/en
Priority to ZA9710272A priority patent/ZA9710272B/xx
Priority to ARP970105365A priority patent/AR009612A1/es
Publication of ITMI962385A1 publication Critical patent/ITMI962385A1/it
Application granted granted Critical
Publication of IT1287174B1 publication Critical patent/IT1287174B1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D303/00Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02Compounds containing oxirane rings
    • C07D303/12Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
    • C07D303/32Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by aldehydo- or ketonic radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00Sulfones; Sulfoxides
    • C07C317/24Sulfones; Sulfoxides having sulfone or sulfoxide groups and doubly-bound oxygen atoms bound to the same carbon skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IT96MI002385A 1996-11-15 1996-11-15 Diaril-ciclometilenpirazoli farmacologicamente attivi,procedimento per prepararli e composizioni farmaceutiche che li contengono IT1287174B1 (it)

Priority Applications (5)

Application Number Priority Date Filing Date Title
IT96MI002385A IT1287174B1 (it) 1996-11-15 1996-11-15 Diaril-ciclometilenpirazoli farmacologicamente attivi,procedimento per prepararli e composizioni farmaceutiche che li contengono
PCT/EP1997/006398 WO1998022442A2 (en) 1996-11-15 1997-11-12 Pharmaceutical compositions comprising diaryl-cyclomethylenpyrazole compounds and their use as cyclooxygenase i (cox 1) inhibitors
AU55526/98A AU5552698A (en) 1996-11-15 1997-11-12 Pharmaceutical compositions comprising diaryl-cyclomethylenpyrazole compounds and their use as cyclooxygenase i (cox i) inhibitors
ZA9710272A ZA9710272B (en) 1996-11-15 1997-11-13 Pharmaceutical compositions comprising diaryl-cyclomethylenpyrazole compounds.
ARP970105365A AR009612A1 (es) 1996-11-15 1997-11-17 Una composicion farmaceutica, un diaril-ciclometilenpirazol, un procedimiento para preparar un diaril-ciclometilenpirazol y comuestosintermedios

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT96MI002385A IT1287174B1 (it) 1996-11-15 1996-11-15 Diaril-ciclometilenpirazoli farmacologicamente attivi,procedimento per prepararli e composizioni farmaceutiche che li contengono

Publications (3)

Publication Number Publication Date
ITMI962385A0 true ITMI962385A0 (it) 1996-11-15
ITMI962385A1 ITMI962385A1 (it) 1998-05-15
IT1287174B1 IT1287174B1 (it) 1998-08-04

Family

ID=11375225

Family Applications (1)

Application Number Title Priority Date Filing Date
IT96MI002385A IT1287174B1 (it) 1996-11-15 1996-11-15 Diaril-ciclometilenpirazoli farmacologicamente attivi,procedimento per prepararli e composizioni farmaceutiche che li contengono

Country Status (5)

Country Link
AR (1) AR009612A1 (it)
AU (1) AU5552698A (it)
IT (1) IT1287174B1 (it)
WO (1) WO1998022442A2 (it)
ZA (1) ZA9710272B (it)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TNSN99111A1 (fr) * 1998-06-11 2005-11-10 Pfizer Derives de sulfonylbenzene nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant.
US6727238B2 (en) 1998-06-11 2004-04-27 Pfizer Inc. Sulfonylbenzene compounds as anti-inflammatory/analgesic agents
US6294558B1 (en) 1999-05-31 2001-09-25 Pfizer Inc. Sulfonylbenzene compounds as anti-inflammatory/analgesic agents
WO2000066562A1 (en) * 1999-05-03 2000-11-09 Dr. Reddy's Research Foundation Pyrazoles having antiinflammatory activity
US6506784B1 (en) 1999-07-01 2003-01-14 3-Dimensional Pharmaceuticals, Inc. Use of 1,3-substituted pyrazol-5-yl sulfonates as pesticides
US6409988B1 (en) 1999-07-01 2002-06-25 3-Dimensional Pharmaceuticals, Inc. Radiolabeled 1-aryl pyrazoles, the synthesis thereof and the use thereof as pest GABA receptor ligands
WO2001007413A1 (en) 1999-07-22 2001-02-01 3-Dimensional Pharmaceuticals, Inc. 1-aryl-3-thioalkyl pyrazoles, the synthesis thereof and the use thereof as insecticides
US6545033B1 (en) 1999-10-06 2003-04-08 3-Dimensional Pharmaceuticals, Inc. Fused 1-(2,6-dichloro-4-trifluoromethylphenyl)-pyrazoles, the synthesis thereof and the use thereof as pesticides
US6083969A (en) * 1999-10-20 2000-07-04 Ortho-Mcneil Pharaceutical, Inc. 1,3- and 2,3-diarylcycloalkano and cycloalkeno pyrazoles as selective inhibitors of cyclooxygenase-2 and antiinflammatory agents
ES2159479B1 (es) * 1999-10-25 2002-05-01 Menarini Lab Nuevos indazoles como inhibidores de la ciclooxigenasa-ii
AU2001296542B2 (en) 2000-10-02 2007-10-25 Emory University Triptolide analogs for the treatment of autoimmune and inflammatory disorders
US6673818B2 (en) 2001-04-20 2004-01-06 Pharmacia Corporation Fluoro-substituted benzenesulfonyl compounds for the treatment of inflammation
PL1745791T3 (pl) 2003-05-07 2013-11-29 Osteologix As Leczenie chorób chrząstki/kości za pomocą rozpuszczalnych w wodzie soli strontu
AU2013302468B2 (en) 2012-08-16 2017-08-24 Janssen Pharmaceutica Nv Substituted pyrazoles as N-type calcium channel blockers
PE20151137A1 (es) * 2012-08-16 2015-08-07 Janssen Pharmaceutica Nv Ciclopentilpirazoles como bloqueadores del canal de calcio tipo n
BR112015003359A2 (pt) * 2012-08-16 2017-07-04 Janssen Pharmaceutica Nv pirrolopirazóis como bloqueadores de canal de cálcio de tipo-n
US9453002B2 (en) 2013-08-16 2016-09-27 Janssen Pharmaceutica Nv Substituted imidazoles as N-type calcium channel blockers
CA3209491A1 (en) 2021-03-15 2022-09-22 Saul Yedgar Hyaluronic acid-conjugated dipalmitoyl phosphatidyl ethanolamine in combination with non-steroidal anti-inflammatory drugs (nsaids) for treating or alleviating inflammatory disease

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3928378A (en) * 1974-01-30 1975-12-23 Hoechst Co American Fused bicyclic aminopyrazoles
FR2315924A1 (fr) * 1975-07-03 1977-01-28 Enzypha Nouveaux polymethylene-4,5 pyrazoles, leur procede de preparation et leur application en therapeutique
US4173634A (en) * 1979-02-23 1979-11-06 E. R. Squibb & Sons, Inc. Basically-substituted tricyclic pyrazoles useful as antiinflammatory agents
DK0924201T3 (da) * 1993-11-30 2002-05-21 Searle & Co Tricyclisk substitueret pyrazolylbenzensulfonamider og deres anvendelse som cyclooxygenase II-inhibitorer

Also Published As

Publication number Publication date
WO1998022442A3 (en) 1998-07-30
IT1287174B1 (it) 1998-08-04
AR009612A1 (es) 2000-04-26
WO1998022442A2 (en) 1998-05-28
ZA9710272B (en) 1998-06-10
ITMI962385A1 (it) 1998-05-15
AU5552698A (en) 1998-06-10

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Legal Events

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