ITMI962385A0 - Diaril-ciclometilenpirazoli farmacologicamente attivi procedimento per prepararli e composizioni farmaceutiche che li contengono - Google Patents
Diaril-ciclometilenpirazoli farmacologicamente attivi procedimento per prepararli e composizioni farmaceutiche che li contengonoInfo
- Publication number
- ITMI962385A0 ITMI962385A0 IT96MI002385A ITMI962385A ITMI962385A0 IT MI962385 A0 ITMI962385 A0 IT MI962385A0 IT 96MI002385 A IT96MI002385 A IT 96MI002385A IT MI962385 A ITMI962385 A IT MI962385A IT MI962385 A0 ITMI962385 A0 IT MI962385A0
- Authority
- IT
- Italy
- Prior art keywords
- cyclomethylenpyrazoles
- preparing
- procedure
- contain
- pharmaceutical compositions
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/12—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
- C07D303/32—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by aldehydo- or ketonic radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
- C07C317/24—Sulfones; Sulfoxides having sulfone or sulfoxide groups and doubly-bound oxygen atoms bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Priority Applications (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT96MI002385A IT1287174B1 (it) | 1996-11-15 | 1996-11-15 | Diaril-ciclometilenpirazoli farmacologicamente attivi,procedimento per prepararli e composizioni farmaceutiche che li contengono |
PCT/EP1997/006398 WO1998022442A2 (en) | 1996-11-15 | 1997-11-12 | Pharmaceutical compositions comprising diaryl-cyclomethylenpyrazole compounds and their use as cyclooxygenase i (cox 1) inhibitors |
AU55526/98A AU5552698A (en) | 1996-11-15 | 1997-11-12 | Pharmaceutical compositions comprising diaryl-cyclomethylenpyrazole compounds and their use as cyclooxygenase i (cox i) inhibitors |
ZA9710272A ZA9710272B (en) | 1996-11-15 | 1997-11-13 | Pharmaceutical compositions comprising diaryl-cyclomethylenpyrazole compounds. |
ARP970105365A AR009612A1 (es) | 1996-11-15 | 1997-11-17 | Una composicion farmaceutica, un diaril-ciclometilenpirazol, un procedimiento para preparar un diaril-ciclometilenpirazol y comuestosintermedios |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT96MI002385A IT1287174B1 (it) | 1996-11-15 | 1996-11-15 | Diaril-ciclometilenpirazoli farmacologicamente attivi,procedimento per prepararli e composizioni farmaceutiche che li contengono |
Publications (3)
Publication Number | Publication Date |
---|---|
ITMI962385A0 true ITMI962385A0 (it) | 1996-11-15 |
ITMI962385A1 ITMI962385A1 (it) | 1998-05-15 |
IT1287174B1 IT1287174B1 (it) | 1998-08-04 |
Family
ID=11375225
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT96MI002385A IT1287174B1 (it) | 1996-11-15 | 1996-11-15 | Diaril-ciclometilenpirazoli farmacologicamente attivi,procedimento per prepararli e composizioni farmaceutiche che li contengono |
Country Status (5)
Country | Link |
---|---|
AR (1) | AR009612A1 (it) |
AU (1) | AU5552698A (it) |
IT (1) | IT1287174B1 (it) |
WO (1) | WO1998022442A2 (it) |
ZA (1) | ZA9710272B (it) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TNSN99111A1 (fr) * | 1998-06-11 | 2005-11-10 | Pfizer | Derives de sulfonylbenzene nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant. |
US6727238B2 (en) | 1998-06-11 | 2004-04-27 | Pfizer Inc. | Sulfonylbenzene compounds as anti-inflammatory/analgesic agents |
US6294558B1 (en) | 1999-05-31 | 2001-09-25 | Pfizer Inc. | Sulfonylbenzene compounds as anti-inflammatory/analgesic agents |
WO2000066562A1 (en) * | 1999-05-03 | 2000-11-09 | Dr. Reddy's Research Foundation | Pyrazoles having antiinflammatory activity |
US6506784B1 (en) | 1999-07-01 | 2003-01-14 | 3-Dimensional Pharmaceuticals, Inc. | Use of 1,3-substituted pyrazol-5-yl sulfonates as pesticides |
US6409988B1 (en) | 1999-07-01 | 2002-06-25 | 3-Dimensional Pharmaceuticals, Inc. | Radiolabeled 1-aryl pyrazoles, the synthesis thereof and the use thereof as pest GABA receptor ligands |
WO2001007413A1 (en) | 1999-07-22 | 2001-02-01 | 3-Dimensional Pharmaceuticals, Inc. | 1-aryl-3-thioalkyl pyrazoles, the synthesis thereof and the use thereof as insecticides |
US6545033B1 (en) | 1999-10-06 | 2003-04-08 | 3-Dimensional Pharmaceuticals, Inc. | Fused 1-(2,6-dichloro-4-trifluoromethylphenyl)-pyrazoles, the synthesis thereof and the use thereof as pesticides |
US6083969A (en) * | 1999-10-20 | 2000-07-04 | Ortho-Mcneil Pharaceutical, Inc. | 1,3- and 2,3-diarylcycloalkano and cycloalkeno pyrazoles as selective inhibitors of cyclooxygenase-2 and antiinflammatory agents |
ES2159479B1 (es) * | 1999-10-25 | 2002-05-01 | Menarini Lab | Nuevos indazoles como inhibidores de la ciclooxigenasa-ii |
AU2001296542B2 (en) | 2000-10-02 | 2007-10-25 | Emory University | Triptolide analogs for the treatment of autoimmune and inflammatory disorders |
US6673818B2 (en) | 2001-04-20 | 2004-01-06 | Pharmacia Corporation | Fluoro-substituted benzenesulfonyl compounds for the treatment of inflammation |
PL1745791T3 (pl) | 2003-05-07 | 2013-11-29 | Osteologix As | Leczenie chorób chrząstki/kości za pomocą rozpuszczalnych w wodzie soli strontu |
AU2013302468B2 (en) | 2012-08-16 | 2017-08-24 | Janssen Pharmaceutica Nv | Substituted pyrazoles as N-type calcium channel blockers |
PE20151137A1 (es) * | 2012-08-16 | 2015-08-07 | Janssen Pharmaceutica Nv | Ciclopentilpirazoles como bloqueadores del canal de calcio tipo n |
BR112015003359A2 (pt) * | 2012-08-16 | 2017-07-04 | Janssen Pharmaceutica Nv | pirrolopirazóis como bloqueadores de canal de cálcio de tipo-n |
US9453002B2 (en) | 2013-08-16 | 2016-09-27 | Janssen Pharmaceutica Nv | Substituted imidazoles as N-type calcium channel blockers |
CA3209491A1 (en) | 2021-03-15 | 2022-09-22 | Saul Yedgar | Hyaluronic acid-conjugated dipalmitoyl phosphatidyl ethanolamine in combination with non-steroidal anti-inflammatory drugs (nsaids) for treating or alleviating inflammatory disease |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3928378A (en) * | 1974-01-30 | 1975-12-23 | Hoechst Co American | Fused bicyclic aminopyrazoles |
FR2315924A1 (fr) * | 1975-07-03 | 1977-01-28 | Enzypha | Nouveaux polymethylene-4,5 pyrazoles, leur procede de preparation et leur application en therapeutique |
US4173634A (en) * | 1979-02-23 | 1979-11-06 | E. R. Squibb & Sons, Inc. | Basically-substituted tricyclic pyrazoles useful as antiinflammatory agents |
DK0924201T3 (da) * | 1993-11-30 | 2002-05-21 | Searle & Co | Tricyclisk substitueret pyrazolylbenzensulfonamider og deres anvendelse som cyclooxygenase II-inhibitorer |
-
1996
- 1996-11-15 IT IT96MI002385A patent/IT1287174B1/it active IP Right Grant
-
1997
- 1997-11-12 AU AU55526/98A patent/AU5552698A/en not_active Abandoned
- 1997-11-12 WO PCT/EP1997/006398 patent/WO1998022442A2/en active Application Filing
- 1997-11-13 ZA ZA9710272A patent/ZA9710272B/xx unknown
- 1997-11-17 AR ARP970105365A patent/AR009612A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
WO1998022442A3 (en) | 1998-07-30 |
IT1287174B1 (it) | 1998-08-04 |
AR009612A1 (es) | 2000-04-26 |
WO1998022442A2 (en) | 1998-05-28 |
ZA9710272B (en) | 1998-06-10 |
ITMI962385A1 (it) | 1998-05-15 |
AU5552698A (en) | 1998-06-10 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
0001 | Granted |