IT1293525B1 - Bis-acridincarbossiammidi aventi attivita' antitumorale - Google Patents

Bis-acridincarbossiammidi aventi attivita' antitumorale

Info

Publication number
IT1293525B1
IT1293525B1 IT97MI001852A ITMI971852A IT1293525B1 IT 1293525 B1 IT1293525 B1 IT 1293525B1 IT 97MI001852 A IT97MI001852 A IT 97MI001852A IT MI971852 A ITMI971852 A IT MI971852A IT 1293525 B1 IT1293525 B1 IT 1293525B1
Authority
IT
Italy
Prior art keywords
acridincarbossiamidi
bis
cancer activity
cancer
activity
Prior art date
Application number
IT97MI001852A
Other languages
English (en)
Italian (it)
Inventor
Ippolito Antonini
Sante Martelli
Paolo Polucci
Original Assignee
Uni Degli Studi Camerino
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Uni Degli Studi Camerino filed Critical Uni Degli Studi Camerino
Priority to IT97MI001852A priority Critical patent/IT1293525B1/it
Priority to AU88080/98A priority patent/AU8808098A/en
Priority to JP2000505131A priority patent/JP2001512104A/ja
Priority to EP98939644A priority patent/EP1001936A1/fr
Priority to PCT/EP1998/004755 priority patent/WO1999006372A1/fr
Publication of ITMI971852A1 publication Critical patent/ITMI971852A1/it
Application granted granted Critical
Publication of IT1293525B1 publication Critical patent/IT1293525B1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D219/00Heterocyclic compounds containing acridine or hydrogenated acridine ring systems
    • C07D219/04Heterocyclic compounds containing acridine or hydrogenated acridine ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • C07D219/08Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IT97MI001852A 1997-08-01 1997-08-01 Bis-acridincarbossiammidi aventi attivita' antitumorale IT1293525B1 (it)

Priority Applications (5)

Application Number Priority Date Filing Date Title
IT97MI001852A IT1293525B1 (it) 1997-08-01 1997-08-01 Bis-acridincarbossiammidi aventi attivita' antitumorale
AU88080/98A AU8808098A (en) 1997-08-01 1998-07-30 Bis-acridinecarboxamides having antitumor activity
JP2000505131A JP2001512104A (ja) 1997-08-01 1998-07-30 抗腫瘍活性を有するビス−アクリジンカルボキサミド
EP98939644A EP1001936A1 (fr) 1997-08-01 1998-07-30 Bis-acridinecarboxamides ayant une activite antitumorale
PCT/EP1998/004755 WO1999006372A1 (fr) 1997-08-01 1998-07-30 Bis-acridinecarboxamides ayant une activite antitumorale

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT97MI001852A IT1293525B1 (it) 1997-08-01 1997-08-01 Bis-acridincarbossiammidi aventi attivita' antitumorale

Publications (2)

Publication Number Publication Date
ITMI971852A1 ITMI971852A1 (it) 1999-02-01
IT1293525B1 true IT1293525B1 (it) 1999-03-01

Family

ID=11377699

Family Applications (1)

Application Number Title Priority Date Filing Date
IT97MI001852A IT1293525B1 (it) 1997-08-01 1997-08-01 Bis-acridincarbossiammidi aventi attivita' antitumorale

Country Status (5)

Country Link
EP (1) EP1001936A1 (fr)
JP (1) JP2001512104A (fr)
AU (1) AU8808098A (fr)
IT (1) IT1293525B1 (fr)
WO (1) WO1999006372A1 (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9621795D0 (en) * 1996-10-18 1996-12-11 Xenova Ltd Pharmaceutical compounds
FR2879598B1 (fr) * 2004-12-17 2007-03-30 Sod Conseils Rech Applic Inhibiteurs de phosphatases cdc25
EP3070078B1 (fr) * 2015-03-20 2017-10-04 Politechnika Gdanska Bisacridines asymmetriques at leur utilisation en tant qu`agents anti-tumorales

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9104548D0 (en) * 1991-03-05 1991-04-17 Cholody Wienlaw M Antineoplastic modified imidazoacridines
US5508289A (en) * 1994-03-14 1996-04-16 The United States America As Represented By The Department Of Health And Human Services Bis-acridone chemotherapeutic derivatives
EP0892801B1 (fr) * 1996-04-12 2002-01-02 THE GOVERNMENT OF THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES Composes derives de l'acridone utiles en tant qu'agents antineoplasiques et antiretroviraux

Also Published As

Publication number Publication date
EP1001936A1 (fr) 2000-05-24
JP2001512104A (ja) 2001-08-21
WO1999006372A1 (fr) 1999-02-11
AU8808098A (en) 1999-02-22
ITMI971852A1 (it) 1999-02-01

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