IT1250626B - ESERIDIN DERIVATIVES USEFUL FOR THE TREATMENT OF DISEASES ASSOCIATED WITH CHOLINERGIC DISORDERS, PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM. - Google Patents
ESERIDIN DERIVATIVES USEFUL FOR THE TREATMENT OF DISEASES ASSOCIATED WITH CHOLINERGIC DISORDERS, PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM.Info
- Publication number
- IT1250626B IT1250626B ITMI911842A ITMI911842A IT1250626B IT 1250626 B IT1250626 B IT 1250626B IT MI911842 A ITMI911842 A IT MI911842A IT MI911842 A ITMI911842 A IT MI911842A IT 1250626 B IT1250626 B IT 1250626B
- Authority
- IT
- Italy
- Prior art keywords
- preparation
- pharmaceutical compositions
- eseridin
- procedure
- contain
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title 2
- CNBHDDBNEKKMJH-ZFWWWQNUSA-N Eseridine Chemical class O1N(C)CC[C@@]2(C)C3=CC(OC(=O)NC)=CC=C3N(C)[C@H]21 CNBHDDBNEKKMJH-ZFWWWQNUSA-N 0.000 title 1
- 230000001713 cholinergic effect Effects 0.000 title 1
- 201000010099 disease Diseases 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- 125000004432 carbon atom Chemical group C* 0.000 abstract 2
- 230000000694 effects Effects 0.000 abstract 1
- 150000007522 mineralic acids Chemical class 0.000 abstract 1
- 150000007524 organic acids Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invenzione riguarda i derivati dell'eseridina ad attività anticoline sterasi di formula (I) (FORMULA I) in cui R è un alchile saturo, lineare o ramificato, avente da 1 a 20 atomi di carbonio, oppure un alchile lineare o ramificato, contenente una o più insaturazioni, avente da 1 a 20 atomi di carbonio, R1 e R2, uguali o diversi fra loro, sono H o alchile lineare o ramificato, n è 0, 1, 2 oppure 3 e HA è un acido organico o inorganico farmaceuticamente accettabile, il procedimento per la loro preparazione e le composizioni farmaceutiche che li contengono.The present invention relates to derivatives of hexeridine with anticoline sterase activity of formula (I) (FORMULA I) wherein R is a saturated alkyl, linear or branched, having from 1 to 20 carbon atoms, or a linear or branched alkyl, containing one or more unsaturations, having from 1 to 20 carbon atoms, R1 and R2, equal or different from each other, are H or linear or branched alkyl, n is 0, 1, 2 or 3 and HA is an organic or inorganic acid pharmaceutically acceptable, the process for their preparation and the pharmaceutical compositions containing them.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITMI911842A IT1250626B (en) | 1991-07-04 | 1991-07-04 | ESERIDIN DERIVATIVES USEFUL FOR THE TREATMENT OF DISEASES ASSOCIATED WITH CHOLINERGIC DISORDERS, PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM. |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITMI911842A IT1250626B (en) | 1991-07-04 | 1991-07-04 | ESERIDIN DERIVATIVES USEFUL FOR THE TREATMENT OF DISEASES ASSOCIATED WITH CHOLINERGIC DISORDERS, PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM. |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| ITMI911842A0 ITMI911842A0 (en) | 1991-07-04 |
| ITMI911842A1 ITMI911842A1 (en) | 1993-01-05 |
| IT1250626B true IT1250626B (en) | 1995-04-21 |
Family
ID=11360273
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ITMI911842A IT1250626B (en) | 1991-07-04 | 1991-07-04 | ESERIDIN DERIVATIVES USEFUL FOR THE TREATMENT OF DISEASES ASSOCIATED WITH CHOLINERGIC DISORDERS, PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM. |
Country Status (1)
| Country | Link |
|---|---|
| IT (1) | IT1250626B (en) |
-
1991
- 1991-07-04 IT ITMI911842A patent/IT1250626B/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| ITMI911842A1 (en) | 1993-01-05 |
| ITMI911842A0 (en) | 1991-07-04 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| UY26143A1 (en) | USEFUL HETEROCYCLIC DERIVATIVES AS ANTI-CANCER AGENTS | |
| MX9603593A (en) | 4-heterocyclyl-substituted quinazoline derivatives, processes for their preparation and their use as anti-cancer agents. | |
| ES2160693T3 (en) | STABLE FORMULATION OF 10-HYDROXY-7-ETHYL-CAMPTOTECHINE IN THE LACTONE FORM. | |
| TR200003478T2 (en) | Isothiazole derivatives useful as anticancer agents | |
| IT1254915B (en) | ADENOSINE DERIVATIVES FOR ACTIVITY A2 AGONIST | |
| IL99926A0 (en) | Cyclo imino derivatives,their preparation and pharmaceutical compositions containing them | |
| HUT70426A (en) | Pyrazolo-pyrimidine derivatives, process for preparing them and pharmaceutical compositions containing them as active agents | |
| HUT49612A (en) | Process for producing new 3-alkenyl-1-azabicyclo/3.2.0/ hept-2-ene-2-carboxylic acid derivatives and pharmaceutical compositions comprising same | |
| ES2132101T3 (en) | PROCEDURE FOR THE PREPARATION OF A MEDICINE INTENDED FOR ADMINISTRATION BY ORAL OR TOPIC IN THE TREATMENT OF LEISHMANIASIS. | |
| NO307688B1 (en) | Use of terfenadine derivatives as antihistamine agents in a pharmaceutical composition | |
| HU9401161D0 (en) | Oxazolidone derivatives, process for producing them and pharmaceutical compositions containing them | |
| AU3623299A (en) | Benzofuroxan derivatives and their use in treating angina pectoris | |
| TW343975B (en) | New phospholipid derivatives of phosphonocarboxylic acids, the production thereof as well as their use as antiviral pharmaceutical agents | |
| AR003456A1 (en) | AN ANALOGUE COMPOUND OF DISTAMICINE AND ITS SALTS, PROCEDURE FOR ITS PREPARATION, PHARMACEUTICAL COMPOSITION THAT CONTAINS IT AND USES OF THE SAME. | |
| IT1256178B (en) | COMPOUNDS WITH THERAPEUTIC ACTIVITIES USEFUL FOR THE TREATMENT OF DISEASES CONNECTED WITH A GLUTATION DEFICIENCY, PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM. | |
| EP0546177A4 (en) | Benzopyran derivative, production thereof, and pharmaceutical composition containing the same. | |
| IT1250626B (en) | ESERIDIN DERIVATIVES USEFUL FOR THE TREATMENT OF DISEASES ASSOCIATED WITH CHOLINERGIC DISORDERS, PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM. | |
| GR3017599T3 (en) | Thiochromane derivatives, process for their preparation and pharmaceutical compositions containing them. | |
| IT1250625B (en) | DERIVATIVES OF HESERIDINE USEFUL FOR THE TREATMENT OF DISEASES ASSOCIATED WITH COLINERGIC DISORDERS, PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM. | |
| ITMI932193A1 (en) | COMPOUNDS WITH ANTIHISTAMIN ACTIVITY PROCEDURE FOR THEIR PREPERATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
| AU7424394A (en) | 3- or 4-glycosyloxybenzopyran derivatives and antiallergic agents containing the derivatives as active ingredients | |
| FI892685A0 (en) | Method for the preparation of new cytostatically active anthracycline derivatives | |
| AU686104B2 (en) | Substituted amidinonaphthyl ester derivatives | |
| ES2121058T3 (en) | CARBAPENEM ANTIBIOTIC COMPOUNDS. | |
| MX9804752A (en) | Covalent lipid-phosphono-carboxylic acid conjugates and application thereof as antiviral medicaments. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 0001 | Granted |