IT1219567B - FORSKOLINA DERIVATIVES, THEIR PROCEDURE AND PREPARATION INTERMEDIATES, THEIR APPLICATION AS MEDICATIONS AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM - Google Patents

FORSKOLINA DERIVATIVES, THEIR PROCEDURE AND PREPARATION INTERMEDIATES, THEIR APPLICATION AS MEDICATIONS AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM

Info

Publication number
IT1219567B
IT1219567B IT47912/88A IT4791288A IT1219567B IT 1219567 B IT1219567 B IT 1219567B IT 47912/88 A IT47912/88 A IT 47912/88A IT 4791288 A IT4791288 A IT 4791288A IT 1219567 B IT1219567 B IT 1219567B
Authority
IT
Italy
Prior art keywords
forskolina
medications
derivatives
procedure
contain
Prior art date
Application number
IT47912/88A
Other languages
Italian (it)
Other versions
IT8847912A0 (en
Inventor
Bernard Delpech
Robert Lett
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of IT8847912A0 publication Critical patent/IT8847912A0/en
Application granted granted Critical
Publication of IT1219567B publication Critical patent/IT1219567B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78Ring systems having three or more relevant rings
    • C07D311/92Naphthopyrans; Hydrogenated naphthopyrans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrane Compounds (AREA)
IT47912/88A 1987-05-04 1988-05-03 FORSKOLINA DERIVATIVES, THEIR PROCEDURE AND PREPARATION INTERMEDIATES, THEIR APPLICATION AS MEDICATIONS AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM IT1219567B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8706242A FR2614891B1 (en) 1987-05-04 1987-05-04 NOVEL FORSKOLINE DERIVATIVES, THEIR PREPARATION PROCESS, THEIR APPLICATION AS MEDICAMENTS, THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AS WELL AS INTERMEDIATES OF THEIR PREPARATION PROCESS

Publications (2)

Publication Number Publication Date
IT8847912A0 IT8847912A0 (en) 1988-05-03
IT1219567B true IT1219567B (en) 1990-05-18

Family

ID=9350729

Family Applications (1)

Application Number Title Priority Date Filing Date
IT47912/88A IT1219567B (en) 1987-05-04 1988-05-03 FORSKOLINA DERIVATIVES, THEIR PROCEDURE AND PREPARATION INTERMEDIATES, THEIR APPLICATION AS MEDICATIONS AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM

Country Status (7)

Country Link
JP (1) JPS63284169A (en)
CH (1) CH676598A5 (en)
DE (1) DE3815213A1 (en)
FR (1) FR2614891B1 (en)
GB (1) GB2205564A (en)
IT (1) IT1219567B (en)
NL (1) NL8801174A (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5268471A (en) * 1990-07-24 1993-12-07 Hoechst Aktiengesellschaft Process for the preparation of 6-acyl, 7-acyl, and 6,7-diacyl analogues of forskolin and intermediates thereof
KR920002575A (en) * 1990-07-24 1992-02-28 이젠브루크, 라피체 Method for preparing 6-acyl, 7-acyl and 6,7-diacyl analogs of forskolin and intermediates thereof
FI913506A (en) * 1990-07-24 1992-01-25 Hoechst Ag FOERFARANDE FOER FRAMSTAELLNING AV 6- (SUBSTITUERAT AMINOPROPIONYL) -DERIVAT AV FORSKOLIN.
CN1089092C (en) * 1997-10-30 2002-08-14 中国科学院动物研究所 Diterpene-kind compound anticancer drug capable of promoting differentiation and depressing proliferation and preparation method and use thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1083589A (en) * 1975-09-06 1980-08-12 Sujata V. Bhat Effective substance from plants belonging to the labiatae family
AU2717777A (en) * 1976-07-21 1979-01-25 Hoechst Ag Pharmacologically effective substance from plants belonging to the family of labiatae
US4517200A (en) * 1982-12-27 1985-05-14 Schering-Plough Corporation Method for treating allergic reactions with forskolin

Also Published As

Publication number Publication date
FR2614891A1 (en) 1988-11-10
CH676598A5 (en) 1991-02-15
FR2614891B1 (en) 1991-05-24
NL8801174A (en) 1988-12-01
IT8847912A0 (en) 1988-05-03
JPS63284169A (en) 1988-11-21
GB2205564A (en) 1988-12-14
GB8810463D0 (en) 1988-06-08
DE3815213A1 (en) 1988-11-17

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Legal Events

Date Code Title Description
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19960419