IT1173443B - Compsns. for topical application to eyes - Google Patents
Compsns. for topical application to eyesInfo
- Publication number
- IT1173443B IT1173443B IT20060/84A IT2006084A IT1173443B IT 1173443 B IT1173443 B IT 1173443B IT 20060/84 A IT20060/84 A IT 20060/84A IT 2006084 A IT2006084 A IT 2006084A IT 1173443 B IT1173443 B IT 1173443B
- Authority
- IT
- Italy
- Prior art keywords
- soln
- cornea
- compsns
- topical application
- eyes
- Prior art date
Links
- 230000000699 topical effect Effects 0.000 title abstract 2
- 210000004087 cornea Anatomy 0.000 abstract 3
- HEDRZPFGACZZDS-UHFFFAOYSA-N Chloroform Chemical compound ClC(Cl)Cl HEDRZPFGACZZDS-UHFFFAOYSA-N 0.000 abstract 2
- RTZKZFJDLAIYFH-UHFFFAOYSA-N Diethyl ether Chemical compound CCOCC RTZKZFJDLAIYFH-UHFFFAOYSA-N 0.000 abstract 2
- FDDDEECHVMSUSB-UHFFFAOYSA-N sulfanilamide Chemical compound NC1=CC=C(S(N)(=O)=O)C=C1 FDDDEECHVMSUSB-UHFFFAOYSA-N 0.000 abstract 2
- 229940124530 sulfonamide Drugs 0.000 abstract 2
- 229940122072 Carbonic anhydrase inhibitor Drugs 0.000 abstract 1
- 102000003846 Carbonic anhydrases Human genes 0.000 abstract 1
- 108090000209 Carbonic anhydrases Proteins 0.000 abstract 1
- 241000283973 Oryctolagus cuniculus Species 0.000 abstract 1
- 239000003489 carbonate dehydratase inhibitor Substances 0.000 abstract 1
- 238000010494 dissociation reaction Methods 0.000 abstract 1
- 230000005593 dissociations Effects 0.000 abstract 1
- 230000035515 penetration Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cosmetics (AREA)
Abstract
Compsns. for topical application to the eyes contain a sulphonamide as carbonic anhydrase inhibitor, the sulphonamide being pharmaceutically acceptable and having the following properties: (a) either a pKa baove 7.0 and below 7.3 or sufficient solubility inter to form an at least 3mM soln. at pH 8.2, but insufficient to form a 1% by wt. soln., (b) a sepn. coefft. with ether of at least 1.0; (c) a sepn. coeffnt. with chloroform of at least 0.01; (d) a dissociation constant with carbonic anhydrase not exceeding 3 x 10 to the 8th power molar; (e) a first order penetration constant across a live rabbit cornea of at least 0.005 per hour; (f) harmlessness to the cornea; (g) stability in soln. and in contact with the cornea.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT20060/84A IT1173443B (en) | 1984-03-15 | 1984-03-15 | Compsns. for topical application to eyes |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT20060/84A IT1173443B (en) | 1984-03-15 | 1984-03-15 | Compsns. for topical application to eyes |
Publications (2)
Publication Number | Publication Date |
---|---|
IT8420060A0 IT8420060A0 (en) | 1984-03-15 |
IT1173443B true IT1173443B (en) | 1987-06-24 |
Family
ID=11163493
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT20060/84A IT1173443B (en) | 1984-03-15 | 1984-03-15 | Compsns. for topical application to eyes |
Country Status (1)
Country | Link |
---|---|
IT (1) | IT1173443B (en) |
-
1984
- 1984-03-15 IT IT20060/84A patent/IT1173443B/en active
Also Published As
Publication number | Publication date |
---|---|
IT8420060A0 (en) | 1984-03-15 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
TA | Fee payment date (situation as of event date), data collected since 19931001 |
Effective date: 19970325 |