IT1160853B - PHENYLETHANOLAMINE DERIVATIVES, PARTICULARLY USEFUL IN THERAPY, AND PROCEDURE FOR THEIR PREPARATION - Google Patents
PHENYLETHANOLAMINE DERIVATIVES, PARTICULARLY USEFUL IN THERAPY, AND PROCEDURE FOR THEIR PREPARATIONInfo
- Publication number
- IT1160853B IT1160853B IT69350/78A IT6935078A IT1160853B IT 1160853 B IT1160853 B IT 1160853B IT 69350/78 A IT69350/78 A IT 69350/78A IT 6935078 A IT6935078 A IT 6935078A IT 1160853 B IT1160853 B IT 1160853B
- Authority
- IT
- Italy
- Prior art keywords
- therapy
- procedure
- preparation
- particularly useful
- phenylethanolamine derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
- C07D317/62—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
- C07D317/64—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C43/00—Ethers; Compounds having groups, groups or groups
- C07C43/02—Ethers
- C07C43/20—Ethers having an ether-oxygen atom bound to a carbon atom of a six-membered aromatic ring
- C07C43/23—Ethers having an ether-oxygen atom bound to a carbon atom of a six-membered aromatic ring containing hydroxy or O-metal groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/34—Compounds containing oxirane rings with hydrocarbon radicals, substituted by sulphur, selenium or tellurium atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D319/10—1,4-Dioxanes; Hydrogenated 1,4-dioxanes
- C07D319/14—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
- C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D319/20—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring with substituents attached to the hetero ring
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP12203477A JPS5473751A (en) | 1977-10-12 | 1977-10-12 | Phenyl ethanolamine derivatives and their preparation |
| JP12843677A JPS5463048A (en) | 1977-10-26 | 1977-10-26 | Novel phenyl ethanolamine derivatives and their preparation |
| JP15535277A JPS5495544A (en) | 1977-12-23 | 1977-12-23 | Phenylethanolamine derivative and its preparation |
| JP7496478A JPS552639A (en) | 1978-06-21 | 1978-06-21 | Phenylethanolamine derivative and its preparation |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IT7869350A0 IT7869350A0 (en) | 1978-10-11 |
| IT1160853B true IT1160853B (en) | 1987-03-11 |
Family
ID=27465764
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT69350/78A IT1160853B (en) | 1977-10-12 | 1978-10-11 | PHENYLETHANOLAMINE DERIVATIVES, PARTICULARLY USEFUL IN THERAPY, AND PROCEDURE FOR THEIR PREPARATION |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US4217305A (en) |
| AT (1) | AT363457B (en) |
| AU (1) | AU526715B2 (en) |
| CA (1) | CA1147342A (en) |
| CH (1) | CH639948A5 (en) |
| DE (1) | DE2843016A1 (en) |
| DK (1) | DK168484B1 (en) |
| ES (2) | ES474149A1 (en) |
| FR (1) | FR2405931A1 (en) |
| GB (1) | GB2006772B (en) |
| GR (1) | GR65337B (en) |
| IT (1) | IT1160853B (en) |
| NO (1) | NO147148C (en) |
| PT (1) | PT68624A (en) |
| SE (1) | SE448232B (en) |
| SU (2) | SU982537A3 (en) |
Families Citing this family (35)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS55124742A (en) * | 1979-03-20 | 1980-09-26 | Kyowa Hakko Kogyo Co Ltd | Novel aminoalcohol derivative |
| US4206125A (en) * | 1979-05-04 | 1980-06-03 | Richardson-Merrell Inc. | 5-[2-[(2,3-Dihydro-1,4-benzodioxan-2-ylmethyl)amino]-1-hydroxyethyl]-2-hydroxybenzoic acid derivatives |
| DD202692A5 (en) * | 1979-12-04 | 1983-09-28 | Ciba Geigy | PROCESS FOR THE PREPARATION OF NEW DERIVATIVES OF 2-AMINO-AETHANOL |
| US4558156A (en) * | 1980-02-08 | 1985-12-10 | Yamanouchi Pharmaceutical Co., Ltd. | Sulfamoyl-substituted phenethylamine derivatives |
| JPS56110665A (en) * | 1980-02-08 | 1981-09-01 | Yamanouchi Pharmaceut Co Ltd | Sulfamoyl-substituted phenetylamine derivative and its preparation |
| US5391825A (en) * | 1980-02-08 | 1995-02-21 | Yamanouchi Pharmaceutical Co., Ltd. | Sulfamoyl substituted phenethylamine intermediates |
| DE3128117A1 (en) * | 1980-07-29 | 1982-03-11 | Yamanouchi Pharmaceutical Co., Ltd., Tokyo | NEW PHENYL-AETHYLAMINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF |
| CA1219865A (en) * | 1982-05-14 | 1987-03-31 | Leo Alig | Aziridine phenethanolamine derivatives |
| PT78388B (en) * | 1983-04-12 | 1986-09-15 | Smithkline Beckman Corp | Dopamine-beta-hydroxylase inhibitors |
| JPS6051106A (en) * | 1983-08-31 | 1985-03-22 | Yamanouchi Pharmaceut Co Ltd | Long acting pharmaceutical preparation of amosulalol hydrochloride |
| EP0162404B1 (en) * | 1984-05-15 | 1988-08-24 | Seitetsu Kagaku Co., Ltd. | Process for preparing 2-alkyl-5-haloacetylbenzenesulfonamide |
| US4678855A (en) * | 1985-10-09 | 1987-07-07 | Merck & Co., Inc. | Substituted benzenesulfonamides |
| JPS62114952A (en) * | 1985-11-13 | 1987-05-26 | Yamanouchi Pharmaceut Co Ltd | Production of substituted phenethylamine derivative |
| AU609209B2 (en) * | 1987-11-13 | 1991-04-26 | Glaxo Group Limited | Phenethanolamine derivatives |
| ATE185070T1 (en) * | 1992-05-22 | 1999-10-15 | Senju Pharma Co | DRUGS FOR GLAUCOMA |
| FR2737494B1 (en) * | 1995-08-04 | 1997-08-29 | Synthelabo | BENZENESULFONAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
| CA2242351C (en) * | 1996-01-10 | 2003-03-11 | Asahi Kasei Kogyo Kabushiki Kaisha | Novel tricyclic compounds and drug compositions containing the same |
| WO1999057131A1 (en) * | 1998-05-06 | 1999-11-11 | Duke University | Method of treating bladder and lower urinary tract syndromes |
| FR2791675B1 (en) * | 1999-03-30 | 2001-05-04 | Synthelabo | DERIVATIVES OF N- [2- (4-AMINOPHENYL) ETHYL] -2,3-DIHYDRO-1,4- BENZODIOXINNE-2-METHANAMINE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
| US6835853B2 (en) | 2001-10-31 | 2004-12-28 | Synthon Bv | Process for resolution of tamsulosin and compounds, compositions, and processes associated therewith |
| ATE502635T1 (en) | 2002-08-19 | 2011-04-15 | Pfizer | COMBINATION THERAPY AGAINST HYPERPROLIFERATIVE DISEASES |
| EP2319843B1 (en) | 2003-05-30 | 2013-04-03 | Ranbaxy Laboratories Limited | Substituted pyrrole derivatives and their use as HMG-CO inhibitors |
| US7329780B2 (en) * | 2003-12-09 | 2008-02-12 | Cj Corporation | Method of preparing optically pure phenethylamine derivatives |
| CA2590533C (en) * | 2004-11-23 | 2010-09-07 | Warner-Lambert Company Llc | 7-(2h-pyrazol-3-yl)-3,5-dihydroxy-heptanoic acid derivatives as hmg co-a reductase inhibitors for the treatment of lipidemia |
| GT200600381A (en) | 2005-08-25 | 2007-03-28 | ORGANIC COMPOUNDS | |
| US7741317B2 (en) | 2005-10-21 | 2010-06-22 | Bristol-Myers Squibb Company | LXR modulators |
| BRPI0618379A2 (en) | 2005-11-08 | 2011-08-30 | Ranbaxy Lab Ltd | (3r, 5r) -7- [2- (4-fluorophenyl) -5-isopropyl-3-phenyl-4 - [(4-hydroxymethylphenylamino) carbonyl] -pyrroleic acid 1-yl] -3,5-dihydroxy heptanoic |
| US7888376B2 (en) | 2005-11-23 | 2011-02-15 | Bristol-Myers Squibb Company | Heterocyclic CETP inhibitors |
| WO2007131804A1 (en) | 2006-05-17 | 2007-11-22 | Synthon B.V. | Tablet composition with a prolonged release of tamsulosin |
| WO2008070496A2 (en) | 2006-12-01 | 2008-06-12 | Bristol-Myers Squibb Company | N- ( (3-benzyl) -2, 2- (bis-phenyl) -propan-1-amine derivatives as cetp inhibitors for the treatment of atherosclerosis and cardiovascular diseases |
| US8465770B2 (en) * | 2008-12-24 | 2013-06-18 | Synthon Bv | Low dose controlled release tablet |
| CN102050766B (en) * | 2009-11-03 | 2013-08-07 | 安徽省新星药物开发有限责任公司 | Synthesis method for amosulalol hydrochloride |
| WO2014170786A1 (en) | 2013-04-17 | 2014-10-23 | Pfizer Inc. | N-piperidin-3-ylbenzamide derivatives for treating cardiovascular diseases |
| WO2016055901A1 (en) | 2014-10-08 | 2016-04-14 | Pfizer Inc. | Substituted amide compounds |
| CN113574055A (en) | 2019-01-18 | 2021-10-29 | 阿斯利康(瑞典)有限公司 | PCSK9 inhibitors and methods of use thereof |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3701808A (en) * | 1967-12-21 | 1972-10-31 | Allen & Hanburys Ltd | Phenylethanolamines |
| GB1266058A (en) | 1969-07-08 | 1972-03-08 | ||
| GB1321701A (en) | 1969-10-01 | 1973-06-27 | Continental Pharma | Amino-alcohols their salts and process for prepairing the same |
| US3711545A (en) * | 1971-02-23 | 1973-01-16 | Smith Kline French Lab | Alpha-aminoalkyl-4-hydroxy-3-sulfamoylaminobenzyl alcohols |
| DE2115926C3 (en) * | 1971-04-01 | 1978-05-03 | C.H. Boehringer Sohn, 6507 Ingelheim | 1 - (4-Hydroxy-3-dimethylaminosulfamidophenyI) -2-aminoether derivatives, process for their preparation and compositions containing them |
| US4034112A (en) * | 1973-06-22 | 1977-07-05 | Imperial Chemical Industries Limited | Ethanolamine derivatives having β-adrenergic blocking activity |
| US3860647A (en) * | 1973-08-20 | 1975-01-14 | Smithkline Corp | {60 -Aminomethyl-4-hydroxy-3-sulfamyl-benzyl alcohols and 4-hydroxy-3-sulfamyl phenethylamines |
| DK31578A (en) * | 1977-02-03 | 1978-08-04 | Allen & Hanburys Ltd | PROCEDURE FOR THE PRODUCTION OF BENZENE DERIVATIVES |
| GB1593651A (en) * | 1977-02-03 | 1981-07-22 | Allen & Hanburys Ltd | Amides |
-
1978
- 1978-09-22 CA CA000311934A patent/CA1147342A/en not_active Expired
- 1978-09-25 GR GR57301A patent/GR65337B/en unknown
- 1978-09-27 US US05/946,192 patent/US4217305A/en not_active Expired - Lifetime
- 1978-10-02 CH CH1021878A patent/CH639948A5/en not_active IP Right Cessation
- 1978-10-03 DE DE19782843016 patent/DE2843016A1/en active Granted
- 1978-10-06 PT PT68624A patent/PT68624A/en unknown
- 1978-10-09 FR FR7828743A patent/FR2405931A1/en active Granted
- 1978-10-11 SU SU782673556A patent/SU982537A3/en active
- 1978-10-11 IT IT69350/78A patent/IT1160853B/en active
- 1978-10-11 AT AT0731778A patent/AT363457B/en not_active IP Right Cessation
- 1978-10-11 NO NO783442A patent/NO147148C/en unknown
- 1978-10-11 DK DK452178A patent/DK168484B1/en active
- 1978-10-11 ES ES474149A patent/ES474149A1/en not_active Expired
- 1978-10-11 SE SE7810613A patent/SE448232B/en not_active IP Right Cessation
- 1978-10-12 GB GB7840390A patent/GB2006772B/en not_active Expired
- 1978-10-12 AU AU40642/78A patent/AU526715B2/en not_active Expired
-
1979
- 1979-06-13 ES ES481549A patent/ES481549A1/en not_active Expired
- 1979-10-18 SU SU792835396A patent/SU932982A3/en active
Also Published As
| Publication number | Publication date |
|---|---|
| NO147148B (en) | 1982-11-01 |
| SE448232B (en) | 1987-02-02 |
| AU526715B2 (en) | 1983-01-27 |
| NO783442L (en) | 1979-04-18 |
| FR2405931A1 (en) | 1979-05-11 |
| ES474149A1 (en) | 1979-10-16 |
| DE2843016C2 (en) | 1988-10-13 |
| AU4064278A (en) | 1980-04-17 |
| DK168484B1 (en) | 1994-04-05 |
| PT68624A (en) | 1978-11-01 |
| AT363457B (en) | 1981-08-10 |
| IT7869350A0 (en) | 1978-10-11 |
| GB2006772B (en) | 1982-02-03 |
| ATA731778A (en) | 1981-01-15 |
| SU982537A3 (en) | 1982-12-15 |
| SU932982A3 (en) | 1982-05-30 |
| US4217305A (en) | 1980-08-12 |
| GR65337B (en) | 1980-08-18 |
| NO147148C (en) | 1983-02-09 |
| GB2006772A (en) | 1979-05-10 |
| DK452178A (en) | 1979-04-13 |
| ES481549A1 (en) | 1980-04-01 |
| SE7810613L (en) | 1979-04-12 |
| FR2405931B1 (en) | 1982-11-19 |
| CH639948A5 (en) | 1983-12-15 |
| DE2843016A1 (en) | 1979-04-26 |
| CA1147342A (en) | 1983-05-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| TA | Fee payment date (situation as of event date), data collected since 19931001 |
Effective date: 19951031 |