IT1147340B - PROCEDURE FOR THE PREPARATION OF 5- (3,4,5-TRIMETOSSIBENZIL) -2,4-DIAMINO-PIRIMIDINA - Google Patents

PROCEDURE FOR THE PREPARATION OF 5- (3,4,5-TRIMETOSSIBENZIL) -2,4-DIAMINO-PIRIMIDINA

Info

Publication number
IT1147340B
IT1147340B IT21209/80A IT2120980A IT1147340B IT 1147340 B IT1147340 B IT 1147340B IT 21209/80 A IT21209/80 A IT 21209/80A IT 2120980 A IT2120980 A IT 2120980A IT 1147340 B IT1147340 B IT 1147340B
Authority
IT
Italy
Prior art keywords
trimetossibenzil
pirimidina
diamino
procedure
preparation
Prior art date
Application number
IT21209/80A
Other languages
Italian (it)
Other versions
IT8021209A0 (en
Inventor
Masini Wanda Molina
Original Assignee
Pharnova Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharnova Sa filed Critical Pharnova Sa
Publication of IT8021209A0 publication Critical patent/IT8021209A0/en
Priority to NL8101676A priority Critical patent/NL8101676A/en
Priority to DK153681A priority patent/DK153681A/en
Application granted granted Critical
Publication of IT1147340B publication Critical patent/IT1147340B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
IT21209/80A 1980-02-20 1980-04-04 PROCEDURE FOR THE PREPARATION OF 5- (3,4,5-TRIMETOSSIBENZIL) -2,4-DIAMINO-PIRIMIDINA IT1147340B (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
NL8101676A NL8101676A (en) 1980-04-04 1981-04-03 Prepn. of trimethoprim from 3,4,5-tri:methoxy-benzoyl chloride - via new 5-tri:methoxy:benzoyl-2,4-di:amino pyrimidine
DK153681A DK153681A (en) 1980-04-04 1981-04-03 METHOD FOR PREPARING 5- (3,4,5-TRIMETHOXYBENZYL) -2,4-DIAMINOPYRIDINE

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH136980 1980-02-20

Publications (2)

Publication Number Publication Date
IT8021209A0 IT8021209A0 (en) 1980-04-04
IT1147340B true IT1147340B (en) 1986-11-19

Family

ID=4208803

Family Applications (1)

Application Number Title Priority Date Filing Date
IT21209/80A IT1147340B (en) 1980-02-20 1980-04-04 PROCEDURE FOR THE PREPARATION OF 5- (3,4,5-TRIMETOSSIBENZIL) -2,4-DIAMINO-PIRIMIDINA

Country Status (6)

Country Link
CA (1) CA1141381A (en)
DE (1) DE3014412A1 (en)
FR (1) FR2476080A1 (en)
GB (1) GB2070602A (en)
IT (1) IT1147340B (en)
YU (1) YU105780A (en)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1497933A (en) * 1965-10-28 1967-10-13 Wellcome Found Preparation of cyanoacetals and pyrimidines
LU67232A1 (en) * 1973-03-16 1973-05-22

Also Published As

Publication number Publication date
IT8021209A0 (en) 1980-04-04
CA1141381A (en) 1983-02-15
DE3014412A1 (en) 1981-09-10
FR2476080A1 (en) 1981-08-21
GB2070602A (en) 1981-09-09
YU105780A (en) 1983-01-21

Similar Documents

Publication Publication Date Title
IT8223705A0 (en) PROCEDURE FOR THE PREPARATION OF CYANOETEROCYCLIC COMPOUNDS.
IT8124141A0 (en) PROCEDURE FOR THE PREPARATION OF 4'-DEOXY-DAUNORUBICIN 4'-DEOXY-DOXORUBICIN.
ES499299A0 (en) PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF TRIMETOXY- 3,4,5 CINAMOYLPIPERACINE
AR227697A1 (en) PROCEDURE FOR THE PREPARATION OF 3,4-BIS-SUBSTITUTED 1,2,5, -OXADIAZOL-2-OXIDES
ES500618A0 (en) PROCEDURE FOR THE PREPARATION OF 2,3-DICHLORO-2-TRIFLUO- ROMETIL-1,1,1,3,4,4,5,5,5, -NONAFLUOROPENTANO
MX7052E (en) PROCEDURE FOR THE PREPARATION OF 2-METOXI-4-AMINO-5-ALKYL SULFONYL-N- (3-BETA-8-AZABICICLO- (3,2,1) OCTIL) -BENZAMIDES
IT1172073B (en) PROCEDURE FOR THE PREPARATION OF BUSPIRONE
ES516597A0 (en) "PROCEDURE FOR THE PREPARATION OF NEW LACTAMA COMPOUNDS".
IT8125157A0 (en) PROCEDURE FOR THE PREPARATION OF 2-AMINOETHANOLS.
IT1123731B (en) PROCEDURE FOR THE PREPARATION OF 1,2,3-TIADIAZOL-5-IL-UREE
IT1147340B (en) PROCEDURE FOR THE PREPARATION OF 5- (3,4,5-TRIMETOSSIBENZIL) -2,4-DIAMINO-PIRIMIDINA
IT8021231A0 (en) PROCEDURE FOR THE PREPARATION OF SUBSTITUTED 2-AMINOPYRAZINES.
IT8224818A0 (en) PROCEDURE FOR THE PREPARATION OF 7-METHYL-3-METHYLENE-7-OTTEN-1-IL-PROPIONATE.
ES505478A0 (en) PROCEDURE FOR THE PREPARATION OF 2,5-DIMETILHEXADIENO-2,4
IT1227791B (en) PROCEDURE FOR THE PREPARATION OF 7,8 DICHLORO-TETRAIDRO-ISOCHINOLINA
ES512697A0 (en) "METHOD OF PREPARING METHYLQUINOXALIN-1,4-DIOXIDIC COMPOUNDS".
IT8026859A0 (en) PROCEDURE FOR THE PREPARATION OF CHOLESTERIN-DERIVATIVES.
IT1148828B (en) PROCEDURE FOR THE PREPARATION OF 1,2-EPOXYCICLOHEXANE
IT8024829A0 (en) PROCEDURE FOR THE PREPARATION OF 2, 4-DIAMINO-5-BENZYLPYRYMIDINES.
IT8223632A0 (en) PROCEDURE FOR THE PREPARATION OF 2,2-DIALKYLAMINO-1-NITROETHENES.
ES509619A0 (en) "PROCEDURE FOR THE PREPARATION OF SUBSTITUTED ALCOHILTIOACILAMINOACIDOS".
ES503907A0 (en) PROCEDURE FOR THE PREPARATION OF 1,2-BENZOTIACINOPIRAZO-LES
IT1151010B (en) METHOD FOR THE PREPARATION OF NI-2-5-DIMETHYLAMINE-METHYL-2-FURANYL-METHYL-THIO-ETHYL-N'-ALCHIL-2-NITRO-1,1-ETHYDIAMINE
FI804018L (en) PROCEDURE FOR FRAMSTATION OF 7,8-DIHYDROXY-1- (SULFAMYLPHENYL) -2,3,4,5-TETRAHYDRO-1H-3-BENZAZEPINDERIVAT
IT8025874A0 (en) PROCEDURE FOR THE PREPARATION OF ISOPHTHALONITRILE.