IT1081511B - PEPTIDE DERIVATIVES AND THEIR PREPARATION - Google Patents

PEPTIDE DERIVATIVES AND THEIR PREPARATION

Info

Publication number
IT1081511B
IT1081511B IT25208/77A IT2520877A IT1081511B IT 1081511 B IT1081511 B IT 1081511B IT 25208/77 A IT25208/77 A IT 25208/77A IT 2520877 A IT2520877 A IT 2520877A IT 1081511 B IT1081511 B IT 1081511B
Authority
IT
Italy
Prior art keywords
preparation
peptide derivatives
peptide
derivatives
Prior art date
Application number
IT25208/77A
Other languages
Italian (it)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of IT1081511B publication Critical patent/IT1081511B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/30Phosphinic acids R2P(=O)(OH); Thiophosphinic acids, i.e. R2P(=X)(XH) (X = S, Se)
    • C07F9/301Acyclic saturated acids which can have further substituents on alkyl
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids RP(=O)(OH)2; Thiophosphonic acids, i.e. RP(=X)(XH)2 (X = S, Se)
    • C07F9/3804Phosphonic acids RP(=O)(OH)2; Thiophosphonic acids, i.e. RP(=X)(XH)2 (X = S, Se) not used, see subgroups
    • C07F9/3808Acyclic saturated acids which can have further substituents on alkyl
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06191Dipeptides containing heteroatoms different from O, S, or N
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
IT25208/77A 1976-07-13 1977-06-29 PEPTIDE DERIVATIVES AND THEIR PREPARATION IT1081511B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB2910176 1976-07-13

Publications (1)

Publication Number Publication Date
IT1081511B true IT1081511B (en) 1985-05-21

Family

ID=10286172

Family Applications (1)

Application Number Title Priority Date Filing Date
IT25208/77A IT1081511B (en) 1976-07-13 1977-06-29 PEPTIDE DERIVATIVES AND THEIR PREPARATION

Country Status (13)

Country Link
JP (1) JPS539720A (en)
AU (1) AU2684777A (en)
BE (1) BE856724A (en)
DE (1) DE2730524A1 (en)
DK (1) DK317177A (en)
FR (1) FR2358414A1 (en)
IL (1) IL52469A0 (en)
IT (1) IT1081511B (en)
LU (1) LU77725A1 (en)
NL (1) NL7707736A (en)
NZ (1) NZ184603A (en)
SE (1) SE7708120L (en)
ZA (1) ZA774073B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GR73085B (en) * 1977-12-20 1984-01-31 Hoffmann La Roche
CA1108125A (en) * 1977-12-23 1981-09-01 Frank R. Atherton Olgiopeptide derivatives of phosphonic acid
DE2901843A1 (en) * 1979-01-18 1980-07-31 Hoechst Ag METHOD FOR PRODUCING CARBONIC ACID AMIDES AND PEPTIDES
DE3368418D1 (en) * 1982-09-17 1987-01-29 Kyowa Hakko Kogyo Kk Phosphorus-containing peptide derivative
EP1585751A4 (en) * 2002-11-14 2008-08-13 Celmed Oncology Usa Inc Peptide deformylase activated prodrugs

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL48835A (en) * 1975-01-27 1979-05-31 Sparamedica Ag Amino acyl and peptidyl derivatives of phophonic acids, their preparation and pharmaceutical compositions containingthem

Also Published As

Publication number Publication date
IL52469A0 (en) 1977-10-31
BE856724A (en) 1978-01-12
JPS539720A (en) 1978-01-28
NL7707736A (en) 1978-01-17
ZA774073B (en) 1978-05-30
FR2358414B1 (en) 1979-06-01
FR2358414A1 (en) 1978-02-10
DE2730524A1 (en) 1978-01-19
DK317177A (en) 1978-01-14
LU77725A1 (en) 1978-09-14
AU2684777A (en) 1979-01-11
SE7708120L (en) 1978-01-14
NZ184603A (en) 1980-03-05

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