IT1080679B - Derivati di dipeptidi - Google Patents

Derivati di dipeptidi

Info

Publication number
IT1080679B
IT1080679B IT24908/77A IT2490877A IT1080679B IT 1080679 B IT1080679 B IT 1080679B IT 24908/77 A IT24908/77 A IT 24908/77A IT 2490877 A IT2490877 A IT 2490877A IT 1080679 B IT1080679 B IT 1080679B
Authority
IT
Italy
Prior art keywords
dipeptides
derivatives
dipeptides derivatives
Prior art date
Application number
IT24908/77A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB26662/76A external-priority patent/GB1564317A/en
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of IT1080679B publication Critical patent/IT1080679B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06008Dipeptides with the first amino acid being neutral
    • C07K5/06017Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06026Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Rheumatology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IT24908/77A 1976-06-25 1977-06-21 Derivati di dipeptidi IT1080679B (it)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB26662/76A GB1564317A (en) 1976-06-25 1976-06-25 Dipeptide derivatives
GB3284776 1976-08-06
GB1065777 1977-03-14

Publications (1)

Publication Number Publication Date
IT1080679B true IT1080679B (it) 1985-05-16

Family

ID=27256556

Family Applications (1)

Application Number Title Priority Date Filing Date
IT24908/77A IT1080679B (it) 1976-06-25 1977-06-21 Derivati di dipeptidi

Country Status (17)

Country Link
US (1) US4187216A (it)
JP (1) JPS532417A (it)
AT (4) AT355742B (it)
AU (1) AU510722B2 (it)
CA (1) CA1092097A (it)
CH (1) CH627735A5 (it)
DE (1) DE2728593A1 (it)
DK (1) DK283177A (it)
FR (1) FR2360561A1 (it)
IE (1) IE45517B1 (it)
IL (1) IL52337A (it)
IT (1) IT1080679B (it)
LU (1) LU77603A1 (it)
NL (1) NL7706967A (it)
NZ (1) NZ184428A (it)
PH (1) PH14141A (it)
SE (1) SE7707339L (it)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5255593A (en) * 1975-10-30 1977-05-07 Ajinomoto Kk Measuring method of enzyme activity
US4309342A (en) * 1980-07-03 1982-01-05 Abbott Laboratories Antibacterial peptides
US4462943A (en) * 1980-11-24 1984-07-31 E. R. Squibb & Sons, Inc. Carboxyalkyl amino acid derivatives of various substituted prolines
US4906615A (en) * 1980-12-18 1990-03-06 Schering Corporation Substituted dipeptides as inhibitors of enkephalinases
US4610816A (en) * 1980-12-18 1986-09-09 Schering Corporation Substituted dipeptides as inhibitors of enkephalinases
US4820729A (en) * 1981-03-30 1989-04-11 Rorer Pharmaceutical Corporation N-substituted-amido-amino acids
CS226907B1 (en) * 1981-08-07 1984-04-16 Kasafirek Evzen Alkylamides of carboxyalkanoylpeptides
CS231228B1 (en) * 1982-10-01 1984-10-15 Evzen Kasafirek Biologically effective tri and tetrapeptide alkylamide derivatives and their processing method
WO1986003746A1 (en) * 1984-12-14 1986-07-03 La Trobe University Amino acid and peptide inhibitors of human leucocytic elastase
EP0190852A3 (en) * 1985-01-31 1988-11-02 Ajinomoto Co., Inc. Dipeptide derivatives and antihypertensive drugs containing them
FR2646847B1 (fr) * 1989-05-12 1991-07-12 Rhone Poulenc Sante N-phenyl amides, leurs procedes de preparation et les medicaments les contenant
JPH05345754A (ja) * 1992-06-15 1993-12-27 Suntory Ltd ジペプチド誘導体およびそれを有効成分とする骨疾患の予防または治療剤
FR2733995B1 (fr) * 1995-05-09 1997-07-25 Inst Nat Sante Rech Med Inhibiteurs de l'inactivation de neuropeptides endogenes notamment la cholecystokinine, leurs procedes de preparation leur utilisation comme medicaments et procede de criblage de medicaments
US7855181B2 (en) * 1999-08-13 2010-12-21 University Of Florida Research Foundation, Inc. Dipeptides for prevention of muscle breakdown and microbial infection
JP6288588B2 (ja) * 2012-11-21 2018-03-07 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング N−スルフィニル−α−アミノアミドの製造方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5255593A (en) * 1975-10-30 1977-05-07 Ajinomoto Kk Measuring method of enzyme activity

Also Published As

Publication number Publication date
IE45517B1 (en) 1982-09-22
PH14141A (en) 1981-03-05
JPS532417A (en) 1978-01-11
NL7706967A (nl) 1977-12-28
DE2728593A1 (de) 1978-01-05
IL52337A (en) 1980-11-30
FR2360561B1 (it) 1980-04-25
ATA300579A (de) 1980-12-15
SE7707339L (sv) 1977-12-26
CA1092097A (en) 1980-12-23
NZ184428A (en) 1980-08-26
CH627735A5 (de) 1982-01-29
AT363205B (de) 1981-07-27
ATA300479A (de) 1981-01-15
FR2360561A1 (fr) 1978-03-03
AU2624377A (en) 1979-01-04
ATA448177A (de) 1979-08-15
ATA300379A (de) 1980-12-15
IL52337A0 (en) 1977-08-31
AT363206B (de) 1981-07-27
AU510722B2 (en) 1980-07-10
IE45517L (en) 1977-12-25
DK283177A (da) 1977-12-26
US4187216A (en) 1980-02-05
AT363626B (de) 1981-08-25
LU77603A1 (it) 1978-07-11
AT355742B (de) 1980-03-25

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