IN2014DN07384A - - Google Patents

Info

Publication number
IN2014DN07384A
IN2014DN07384A IN7384DEN2014A IN2014DN07384A IN 2014DN07384 A IN2014DN07384 A IN 2014DN07384A IN 7384DEN2014 A IN7384DEN2014 A IN 7384DEN2014A IN 2014DN07384 A IN2014DN07384 A IN 2014DN07384A
Authority
IN
India
Prior art keywords
compounds
disclosed
mediated
pyrimidinebased
pyrazolo
Prior art date
Application number
Inventor
Yingzhi Bi
Kenneth Gordon Carson
Giovanni Cianchetta
Michael Alan Green
Godwin Kumi
Alan Main
Yulian Zhang
Glenn Gregory Zipp
Original Assignee
Lexicon Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lexicon Pharmaceuticals Inc filed Critical Lexicon Pharmaceuticals Inc
Publication of IN2014DN07384A publication Critical patent/IN2014DN07384A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/05Isotopically modified compounds, e.g. labelled
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B59/00Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
    • C07B59/002Heterocyclic compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Pyrazolo[l,5-a]pyrimidinebased compounds of the formula: are disclosed, wherein Ri, R2 and R3 are defined herein. Compositions comprising the compounds and methods of their use to treat, manage and/or prevent diseases and disorders mediated by mediated by adaptor associated kinase 1 activity are also disclosed.
IN7384DEN2014 2012-03-09 2013-03-05 IN2014DN07384A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261608765P 2012-03-09 2012-03-09
PCT/US2013/029056 WO2013134228A1 (en) 2012-03-09 2013-03-05 PYRAZOLO[1,5-a]PYRIMIDINE-BASED COMPOUNDS, COMPOSITIONS COMPRISING THEM, AND METHODS OF THEIR USE

Publications (1)

Publication Number Publication Date
IN2014DN07384A true IN2014DN07384A (en) 2015-04-24

Family

ID=47892052

Family Applications (1)

Application Number Title Priority Date Filing Date
IN7384DEN2014 IN2014DN07384A (en) 2012-03-09 2013-03-05

Country Status (25)

Country Link
US (3) US8946415B2 (en)
EP (1) EP2834243B1 (en)
JP (1) JP6418950B2 (en)
KR (1) KR101965025B1 (en)
CN (1) CN104302649B (en)
AR (1) AR090292A1 (en)
AU (1) AU2013230128B2 (en)
BR (1) BR112014022000A8 (en)
CA (1) CA2866143C (en)
DK (1) DK2834243T3 (en)
ES (1) ES2676224T3 (en)
HU (1) HUE038786T2 (en)
IL (1) IL234486A (en)
IN (1) IN2014DN07384A (en)
MX (2) MX381849B (en)
NZ (1) NZ630721A (en)
PL (1) PL2834243T3 (en)
PT (1) PT2834243T (en)
RU (1) RU2014140735A (en)
SG (1) SG11201405561RA (en)
TR (1) TR201808280T4 (en)
TW (1) TW201341386A (en)
UY (1) UY34668A (en)
WO (1) WO2013134228A1 (en)
ZA (1) ZA201406149B (en)

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TW201542550A (en) 2013-09-06 2015-11-16 Lexicon Pharmaceuticals Inc Pyrazolo[1,5-a]pyrimidinyl compound, composition comprising the same, and method of using the same
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TW201620911A (en) * 2014-03-17 2016-06-16 雷西肯製藥股份有限公司 Inhibitors of adapter associated kinase 1, compositions comprising them, and methods of their use
WO2016053794A1 (en) * 2014-09-30 2016-04-07 Bristol-Myers Squibb Company Quinazoline-based kinase inhibitors
HRP20240937T1 (en) * 2014-12-15 2024-10-25 Cmg Pharmaceutical Co., Ltd. Fused ring heteroaryl compounds and their use as trk inhibitors
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CN109890824B (en) 2016-11-02 2022-05-24 詹森药业有限公司 [1,2,4]Triazolo[1,5-A]pyrimidine compounds as PDE2 inhibitors
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JP7321183B2 (en) * 2017-12-15 2023-08-04 ピラミッド バイオサイエンシズ インコーポレイテッド 5-(2-(2,5-difluorophenyl)pyrrolidin-1-yl)-3-(1H-pyrazol-1-yl)pyrazolo[1,5] as TRK kinase inhibitors for treating cancer -A] pyrimidine derivatives and related compounds
CN111511746B (en) 2017-12-19 2024-01-09 特普医药公司 Macrocyclic compounds for the treatment of diseases
EP3730492A4 (en) * 2017-12-22 2021-08-11 Shenzhen TargetRx, Inc. Substituted pyrazolo[1,5-a]pyrimidine compound and pharmaceutical composition and use thereof
JP7162915B2 (en) 2018-01-23 2022-10-31 深▲チェン▼市塔吉瑞生物医薬有限公司 Substituted pyrazolo[1,5-a]pyrimidine macrocycles
JP2022503932A (en) * 2018-09-27 2022-01-12 フォチョン・ファーマシューティカルズ・リミテッド Substituted imidazole [1,2-A] pyridine and [1,2,4] triazolo [1,5-A] pyridine compounds as RET kinase inhibitors
WO2020081508A1 (en) * 2018-10-15 2020-04-23 Nimbus Lakshmi, Inc. Tyk2 inhibitors and uses thereof
WO2021216441A1 (en) 2020-04-21 2021-10-28 Lexicon Pharmaceuticals, Inc. Aak1 inhibitors for use in treating viral infections
WO2021216454A1 (en) * 2020-04-21 2021-10-28 Lexicon Pharmaceuticals, Inc. 4-(3-(pyridin-3-yl)pyrazolo[1,5-a]pyrimidin-5-yl)piperazine for use in the the treatment of cov-229e or cov-oc43 coronaviruses infections
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Also Published As

Publication number Publication date
BR112014022000A2 (en) 2017-06-20
CA2866143A1 (en) 2013-09-12
EP2834243B1 (en) 2018-04-25
NZ630721A (en) 2016-12-23
AR090292A1 (en) 2014-11-05
CN104302649A (en) 2015-01-21
ES2676224T3 (en) 2018-07-17
AU2013230128B2 (en) 2017-08-17
DK2834243T3 (en) 2018-07-23
UY34668A (en) 2013-10-31
JP2015509535A (en) 2015-03-30
JP6418950B2 (en) 2018-11-07
US20150183792A1 (en) 2015-07-02
BR112014022000A8 (en) 2021-06-15
KR101965025B1 (en) 2019-04-02
US8946415B2 (en) 2015-02-03
PL2834243T3 (en) 2018-09-28
US9403832B2 (en) 2016-08-02
WO2013134228A1 (en) 2013-09-12
EP2834243A1 (en) 2015-02-11
SG11201405561RA (en) 2014-10-30
ZA201406149B (en) 2016-06-29
MX381849B (en) 2025-03-13
TR201808280T4 (en) 2018-07-23
AU2013230128A1 (en) 2014-09-25
HK1201257A1 (en) 2015-08-28
RU2014140735A (en) 2016-04-27
PT2834243T (en) 2018-08-01
TW201341386A (en) 2013-10-16
US20170129896A1 (en) 2017-05-11
CN104302649B (en) 2017-06-23
HUE038786T2 (en) 2018-11-28
CA2866143C (en) 2020-08-04
MX345830B (en) 2017-02-17
US20130253194A1 (en) 2013-09-26
MX2014010589A (en) 2014-09-18
KR20140138864A (en) 2014-12-04
IL234486A (en) 2016-10-31

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