IN2014DN07129A - - Google Patents

Info

Publication number
IN2014DN07129A
IN2014DN07129A IN7129DEN2014A IN2014DN07129A IN 2014DN07129 A IN2014DN07129 A IN 2014DN07129A IN 7129DEN2014 A IN7129DEN2014 A IN 7129DEN2014A IN 2014DN07129 A IN2014DN07129 A IN 2014DN07129A
Authority
IN
India
Prior art keywords
fluoroalkyl
bis
pyrazol
carboxylic acid
acid derivatives
Prior art date
Application number
Inventor
Sergii Pazenok
Norbert Lui
Jean Pierre Vors
Frédéric Leroux
Florence Giornal
Original Assignee
Bayer Cropscience Ag
Centre Nat Rech Scient
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag, Centre Nat Rech Scient filed Critical Bayer Cropscience Ag
Publication of IN2014DN07129A publication Critical patent/IN2014DN07129A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/30—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and unsaturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

The invention relates to novel 3 5 bis(fluoroalkyl) pyrazol 4 carboxylic acid derivatives and to a method for producing 3 5 bis(fluoroalkyl) pyrazol 4 carboxylic acid derivatives and 3 5 bis(fluoroalkyl) pyrazoles.
IN7129DEN2014 2012-02-01 2013-01-31 IN2014DN07129A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12356001.3A EP2623496A1 (en) 2012-02-01 2012-02-01 Method for producing 3,5-bis(fluoralkyl)-pyrazol-4-carboxylic acid derivatives and 3,5-bis(fluoralkyl)-pyrazoles
PCT/EP2013/051930 WO2013113829A1 (en) 2012-02-01 2013-01-31 Method for producing 3,5-bis(fluoroalkyl)-pyrazol-4-carboxylic acid derivatives and 3,5-bis(fluoroalkyl)-pyrazoles

Publications (1)

Publication Number Publication Date
IN2014DN07129A true IN2014DN07129A (en) 2015-04-24

Family

ID=47624109

Family Applications (1)

Application Number Title Priority Date Filing Date
IN7129DEN2014 IN2014DN07129A (en) 2012-02-01 2013-01-31

Country Status (13)

Country Link
US (2) US9309202B2 (en)
EP (2) EP2623496A1 (en)
JP (1) JP6155283B2 (en)
KR (1) KR101861116B1 (en)
CN (1) CN104245676B (en)
BR (1) BR112014019036B1 (en)
DK (1) DK2809653T3 (en)
ES (1) ES2647348T3 (en)
IL (1) IL233926B (en)
IN (1) IN2014DN07129A (en)
MX (1) MX362689B (en)
TW (1) TWI609006B (en)
WO (1) WO2013113829A1 (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112015027707B1 (en) 2013-05-22 2021-02-09 Bayer Cropscience Aktiengesellschaft method of preparing 3,5-bis (fluoroalkyl) pyrazole derivatives and intermediate compounds involved in this method
TWI647215B (en) * 2013-11-11 2019-01-11 德商拜耳作物科學股份有限公司 Method for preparing 3,5-dihaloalkylpyrazole derivatives from α,α-dihalamine
CN106164049B (en) * 2014-03-24 2019-04-12 拜耳作物科学股份公司 Process for the preparation of 3, 5-di (haloalkyl) pyrazole derivatives from α -dihaloamines and ketimines
EP3015458A1 (en) * 2014-11-03 2016-05-04 Bayer CropScience AG Process for preparing 3,5-bis(haloalkyl)pyrazole derivatives from a,a-dihaloamines and ketimines
BR112016028700B1 (en) * 2014-06-11 2021-03-23 Bayer Cropscience Aktiengesellschaft PROCESS FOR THE PREPARATION OF 3,5-BIS (HALOALKYL) PIRAZÓIS VIA ACETION OF CETIMINES
EP3154946B1 (en) * 2014-06-11 2018-04-18 Bayer CropScience Aktiengesellschaft Process for preparing 3,5-bis(haloalkyl)pyrazole derivatives via acylation of hydrazones
MX2017010401A (en) 2015-02-11 2017-12-07 Basf Se Pesticidal mixture comprising a pyrazole compound, an insecticide and a fungicide.
EP3313820A1 (en) * 2015-06-26 2018-05-02 Bayer CropScience Aktiengesellschaft Process for preparing substituted pyrazoles containing haloalkoxy- and haloalkylthio groups from , -dihaloalkylamines and ketimines
CN112351972A (en) 2018-06-18 2021-02-09 拜耳公司 Disubstituted 5(3) -pyrazole carboxylic acid esters and methods of making same from enol esters and Fluoroalkylamino (FAR) reagents
WO2020210174A2 (en) * 2019-04-06 2020-10-15 Trinapco, Inc. Sulfonyldiazoles and n-(fluorosulfonyl)azoles, and methods of making the same

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2004460A6 (en) * 1987-07-29 1989-01-01 Consejo Superior Investigacion 3,5-Di:halomethyl pyrazole deriv. prepn.
JP3533134B2 (en) * 1999-02-15 2004-05-31 三井化学株式会社 Fluorinating agents and their production and use
JP2001192369A (en) * 2000-01-12 2001-07-17 Mitsui Chemicals Inc Method of producing fluorine-containing heterocyclic aromatic compound and novel pyrazole ping compound
DE10215292A1 (en) 2002-02-19 2003-08-28 Bayer Cropscience Ag New N-biphenylyl-1-methyl-3-(di- or trifluoromethyl)-1H-pyrazole-4-carboxamides, useful as microbicides, especially fungicides and bactericides for protection of plants or materials such as wood
US7842693B2 (en) * 2002-06-12 2010-11-30 Chemocentryx, Inc. Substituted piperazines
DE10349500A1 (en) 2003-10-23 2005-06-02 Bayer Cropscience Ag A process for producing 2-dihaloacyl-3-amino-acrylic acid esters and 3-dihalomethyl-pyrazole-4-carboxylic acid esters
TW200738701A (en) 2005-07-26 2007-10-16 Du Pont Fungicidal carboxamides
GB0526044D0 (en) * 2005-12-21 2006-02-01 Syngenta Ltd Novel herbicides
WO2008013622A2 (en) 2006-07-27 2008-01-31 E. I. Du Pont De Nemours And Company Fungicidal azocyclic amides
DE102006039909A1 (en) 2006-08-25 2008-03-13 Bayer Cropscience Ag Process for the preparation of 3-dihalomethyl-pyrazole-4-carboxylic acid derivatives
WO2008091594A2 (en) * 2007-01-24 2008-07-31 E. I. Du Pont De Nemours And Company Fungicidal mixtures
EP2133341A1 (en) 2008-02-25 2009-12-16 Bayer CropScience AG Method for regioselective synthesis of 1-alkyl-3-haloalkyl-1-pyrazol-4-carbonic acid derivatives
EP2100883A1 (en) 2008-03-10 2009-09-16 Bayer CropScience AG Method for regioselective synthesis of 1-alkyl-3-haloalkyl-1-pyrazol-4-carbonic acid derivatives
JP2010083763A (en) * 2008-09-29 2010-04-15 Mitsui Chemicals Inc Pyrazole derivative, method of producing the same, and bactericide

Also Published As

Publication number Publication date
JP2015511227A (en) 2015-04-16
ES2647348T3 (en) 2017-12-21
US20160185731A1 (en) 2016-06-30
KR101861116B1 (en) 2018-05-25
BR112014019036B1 (en) 2019-10-08
DK2809653T3 (en) 2017-11-27
TWI609006B (en) 2017-12-21
CN104245676A (en) 2014-12-24
IL233926A0 (en) 2014-09-30
WO2013113829A1 (en) 2013-08-08
IL233926B (en) 2018-08-30
MX2014009203A (en) 2014-11-12
US20150011779A1 (en) 2015-01-08
MX362689B (en) 2019-02-01
US9309202B2 (en) 2016-04-12
EP2809653B1 (en) 2017-08-16
CN104245676B (en) 2016-09-21
JP6155283B2 (en) 2017-06-28
EP2809653A1 (en) 2014-12-10
US10035773B2 (en) 2018-07-31
BR112014019036A2 (en) 2017-08-22
TW201336826A (en) 2013-09-16
EP2623496A1 (en) 2013-08-07
KR20140128344A (en) 2014-11-05

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