IN2013MU03070A - - Google Patents

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Publication number
IN2013MU03070A
IN2013MU03070A IN3070MU2013A IN2013MU03070A IN 2013MU03070 A IN2013MU03070 A IN 2013MU03070A IN 3070MU2013 A IN3070MU2013 A IN 3070MU2013A IN 2013MU03070 A IN2013MU03070 A IN 2013MU03070A
Authority
IN
India
Prior art keywords
preparation
relates
present
novel process
dimethyl fumarate
Prior art date
Application number
Other languages
English (en)
Inventor
Bhaskar Bhirud Shekhar
Hari Bhushan Kumar
M Veerabhadra Swamy H
Jibhau Patil Dilipkumar
Digambar Dabe Avikumar
Original Assignee
Glenmark Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glenmark Pharmaceuticals Ltd filed Critical Glenmark Pharmaceuticals Ltd
Priority to US15/025,056 priority Critical patent/US9840456B2/en
Priority to IN3070MU2013 priority patent/IN2013MU03070A/en
Priority to PCT/IB2014/064726 priority patent/WO2015044853A2/en
Publication of IN2013MU03070A publication Critical patent/IN2013MU03070A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/52Esters of acyclic unsaturated carboxylic acids having the esterified carboxyl group bound to an acyclic carbon atom
    • C07C69/593Dicarboxylic acid esters having only one carbon-to-carbon double bond
    • C07C69/60Maleic acid esters; Fumaric acid esters
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00Preparation of carboxylic acid esters
    • C07C67/08Preparation of carboxylic acid esters by reacting carboxylic acids or symmetrical anhydrides with the hydroxy or O-metal group of organic compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00Preparation of carboxylic acid esters
    • C07C67/48Separation; Purification; Stabilisation; Use of additives
    • C07C67/60Separation; Purification; Stabilisation; Use of additives by treatment giving rise to chemical modification

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IN3070MU2013 2013-09-25 2014-09-22 IN2013MU03070A (enrdf_load_stackoverflow)

Priority Applications (3)

Application Number Priority Date Filing Date Title
US15/025,056 US9840456B2 (en) 2013-09-25 2014-09-22 Process for preparation of dimethyl fumarate
IN3070MU2013 IN2013MU03070A (enrdf_load_stackoverflow) 2013-09-25 2014-09-22
PCT/IB2014/064726 WO2015044853A2 (en) 2013-09-25 2014-09-22 Process for preparation of dimethyl fumarate

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IN3070MU2013 IN2013MU03070A (enrdf_load_stackoverflow) 2013-09-25 2014-09-22

Publications (1)

Publication Number Publication Date
IN2013MU03070A true IN2013MU03070A (enrdf_load_stackoverflow) 2015-07-17

Family

ID=52744630

Family Applications (1)

Application Number Title Priority Date Filing Date
IN3070MU2013 IN2013MU03070A (enrdf_load_stackoverflow) 2013-09-25 2014-09-22

Country Status (3)

Country Link
US (1) US9840456B2 (enrdf_load_stackoverflow)
IN (1) IN2013MU03070A (enrdf_load_stackoverflow)
WO (1) WO2015044853A2 (enrdf_load_stackoverflow)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10098863B2 (en) 2014-02-28 2018-10-16 Banner Life Sciences Llc Fumarate esters
US9326947B1 (en) 2014-02-28 2016-05-03 Banner Life Sciences Llc Controlled release fumarate esters
US9636318B2 (en) 2015-08-31 2017-05-02 Banner Life Sciences Llc Fumarate ester dosage forms
EP3501510B1 (en) 2014-02-28 2020-07-01 Banner Life Sciences LLC Controlled release enteric soft capsules of fumarate esters
JP2018517735A (ja) * 2015-06-17 2018-07-05 バイオジェン・エムエイ・インコーポレイテッドBiogen MA Inc. フマル酸ジメチル粒子及びそれらの医薬組成物
WO2021142062A1 (en) * 2020-01-10 2021-07-15 Banner Life Sciences Llc Fumarate ester dosage forms with enhanced gastrointestinal tolerability

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI2379063T2 (sl) * 2009-01-09 2021-09-30 Fwp Ip Aps Farmacevtska formulacija, ki obsega enega ali več estrov fumarne kisline v tableti v erozivnem matriksu
KR20150080037A (ko) * 2011-06-08 2015-07-08 바이오젠 엠에이 인코포레이티드 고순도 및 결정질 다이메틸 푸마레이트의 제조 방법
CN102766050A (zh) 2012-08-10 2012-11-07 太仓市运通化工厂 一种富马酸二甲酯的合成方法
AU2014314231A1 (en) * 2013-08-26 2016-03-03 Fwp Ip Aps Pharmaceutical composition containing dimethyl fumarate for administration at a low daily dose

Also Published As

Publication number Publication date
US20160237021A1 (en) 2016-08-18
WO2015044853A2 (en) 2015-04-02
US9840456B2 (en) 2017-12-12
WO2015044853A3 (en) 2015-06-11

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