IN2012DN03310A - - Google Patents

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Publication number
IN2012DN03310A
IN2012DN03310A IN3310DEN2012A IN2012DN03310A IN 2012DN03310 A IN2012DN03310 A IN 2012DN03310A IN 3310DEN2012 A IN3310DEN2012 A IN 3310DEN2012A IN 2012DN03310 A IN2012DN03310 A IN 2012DN03310A
Authority
IN
India
Prior art keywords
moeties
peptiod
tetrapeptide
tripeptide
dipeptide
Prior art date
Application number
Inventor
Guido Franzoso
Albert Andrzej Jaxa-Chamiec
Caroline Minli Rachel Low
Simona Maria Monti
Menotti Ruvo
Laura Tornatore
Catherine Jane Tralau-Stewart
Original Assignee
Imp Innovations Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Imp Innovations Ltd filed Critical Imp Innovations Ltd
Publication of IN2012DN03310A publication Critical patent/IN2012DN03310A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06104—Dipeptides with the first amino acid being acidic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06104—Dipeptides with the first amino acid being acidic
    • C07K5/06113—Asp- or Asn-amino acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0812—Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1016—Tetrapeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)

Abstract

Compounds based around tetrapeptide, tripeptide and dipeptide moeties and corresponding peptiod moeties. Related methods and pharmaceutical compositions for use in treatment of cancer, inflammatory diseases, and other disorders.
IN3310DEN2012 2009-10-22 2010-10-22 IN2012DN03310A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0918579.4A GB0918579D0 (en) 2009-10-22 2009-10-22 Gadd45beta targeting agents
PCT/GB2010/001970 WO2011048390A2 (en) 2009-10-22 2010-10-22 Gadd45beta targeting agents

Publications (1)

Publication Number Publication Date
IN2012DN03310A true IN2012DN03310A (en) 2015-10-23

Family

ID=41426579

Family Applications (1)

Application Number Title Priority Date Filing Date
IN3310DEN2012 IN2012DN03310A (en) 2009-10-22 2010-10-22

Country Status (14)

Country Link
US (2) US8993717B2 (en)
EP (2) EP3178836B1 (en)
JP (2) JP5961113B2 (en)
KR (1) KR20120099440A (en)
CN (1) CN102741269B (en)
AU (1) AU2010309594B2 (en)
BR (1) BR112012011332B1 (en)
CA (2) CA3034860A1 (en)
GB (1) GB0918579D0 (en)
IL (1) IL219325B (en)
IN (1) IN2012DN03310A (en)
MX (1) MX357801B (en)
RU (2) RU2577311C2 (en)
WO (1) WO2011048390A2 (en)

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GB0918579D0 (en) 2009-10-22 2009-12-09 Imp Innovations Ltd Gadd45beta targeting agents
PL219569B1 (en) 2010-02-19 2015-05-29 Peptaderm Spółka Z Ograniczoną Odpowiedzialnością Cyclic tetrapeptides and their application
GB201107118D0 (en) * 2011-04-27 2011-06-08 Imp Innovations Ltd Method of diagnosis and prognosis
WO2013055051A1 (en) * 2011-10-14 2013-04-18 서울대학교산학협력단 Peptide nanostructure and a production method therefor
DK3777876T3 (en) 2011-10-28 2023-10-30 Neostrata Company Inc N-acyl dipeptide derivatives and uses thereof
WO2013142376A1 (en) * 2012-03-19 2013-09-26 Aposignal Bioscience Llc Composition and methods for cell modulation
CN104817616A (en) * 2014-01-30 2015-08-05 陈光健 Oligopeptide CD02, and preparation method and application thereof
CN104817618B (en) * 2014-01-30 2018-07-03 陈光健 Oligopeptides CD01 and its preparation method and application
GB201414542D0 (en) * 2014-08-15 2014-10-01 Imp Innovations Ltd Novel therapy
CN111574585B (en) * 2019-01-30 2021-10-01 浙江省医学科学院 Cod skin oligopeptide and separation and purification method and application thereof
RU2716258C1 (en) * 2019-07-30 2020-03-11 Автономная некоммерческая образовательная организация высшего образования Сколковский институт науки и технологий Peptide antagonist of the nmda receptor
KR102417496B1 (en) * 2019-11-29 2022-07-06 (주)수파드엘릭사 Peptide for inhibiting activity of androgen receptor and Cosmetic composition using the same
WO2021194228A1 (en) * 2020-03-23 2021-09-30 주식회사 엘베이스 Pharmaceutical composition for prevention or treatment of cancer
KR102348728B1 (en) * 2020-03-23 2022-01-12 주식회사 엘베이스 Pharmaceutical Composition for the Prevention or Treatment of Cancer
KR20230038457A (en) 2020-06-10 2023-03-20 알리고스 테라퓨틱스 인코포레이티드 Antiviral compounds for treating coronavirus, picornavirus and norovirus infections
JP2023522311A (en) * 2021-03-22 2023-05-30 エル－ベース カンパニー リミテッド Pharmaceutical composition for cancer prevention or treatment
WO2022203219A1 (en) * 2021-03-22 2022-09-29 주식회사 엘베이스 Pharmaceutical composition for prevention or treatment of cancer
IL309732A (en) 2021-07-09 2024-02-01 Aligos Therapeutics Inc Anti-viral compounds
IT202100023357A1 (en) * 2021-09-09 2023-03-09 Cheirontech S R L Peptides with anti-angiogenic activity
WO2023043269A1 (en) * 2021-09-17 2023-03-23 주식회사 엘베이스 Pharmaceutical composition for modulating immune response
KR102494749B1 (en) * 2021-09-17 2023-02-06 주식회사 엘베이스 Method of characterizing responders to CAGE inhibitors for treatment of cancer
WO2023043261A1 (en) * 2021-09-17 2023-03-23 주식회사 엘베이스 Pharmaceutical composition for enhancing anticancer effect of anticancer drug
CN116350746B (en) * 2023-05-16 2024-03-22 海口桥水联合科技有限责任公司 Application of sardine peptide composition in medicines for treating allergic rhinitis

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Also Published As

Publication number Publication date
BR112012011332A2 (en) 2016-11-22
WO2011048390A3 (en) 2011-11-03
US20150368294A1 (en) 2015-12-24
CN102741269A (en) 2012-10-17
US9518083B2 (en) 2016-12-13
CA2778236A1 (en) 2011-04-28
RU2012120905A (en) 2013-11-27
CA3034860A1 (en) 2011-04-28
AU2010309594B2 (en) 2016-01-07
MX2012004755A (en) 2012-11-22
EP2491051A2 (en) 2012-08-29
JP2013508346A (en) 2013-03-07
WO2011048390A2 (en) 2011-04-28
EP3178836A1 (en) 2017-06-14
KR20120099440A (en) 2012-09-10
US20120277164A1 (en) 2012-11-01
JP2016166211A (en) 2016-09-15
JP5961113B2 (en) 2016-08-02
CN102741269B (en) 2017-08-29
IL219325B (en) 2019-02-28
BR112012011332B1 (en) 2022-07-05
RU2577311C2 (en) 2016-03-20
IL219325A0 (en) 2012-06-28
MX357801B (en) 2018-07-25
EP3178836B1 (en) 2019-12-25
RU2016102083A (en) 2018-11-20
US8993717B2 (en) 2015-03-31
GB0918579D0 (en) 2009-12-09
AU2010309594A1 (en) 2012-05-17

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