IL44068A0 - Process for the preparation of new benzodiazepines and intermediates - Google Patents

Process for the preparation of new benzodiazepines and intermediates

Info

Publication number
IL44068A0
IL44068A0 IL44068A IL4406874A IL44068A0 IL 44068 A0 IL44068 A0 IL 44068A0 IL 44068 A IL44068 A IL 44068A IL 4406874 A IL4406874 A IL 4406874A IL 44068 A0 IL44068 A0 IL 44068A0
Authority
IL
Israel
Prior art keywords
intermediates
preparation
benzodiazepines
new
new benzodiazepines
Prior art date
Application number
IL44068A
Other versions
IL44068A (en
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of IL44068A0 publication Critical patent/IL44068A0/en
Publication of IL44068A publication Critical patent/IL44068A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • C07D215/22Oxygen atoms attached in position 2 or 4
    • C07D215/227Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/18Halogen atoms or nitro radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/101,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
IL44068A 1973-02-14 1974-01-24 Process for the preparation of 6-phenyl-4h-s-triazolo(4,3a)(1,4)benzodiazepines and intermediate 2(2-(methanesulfonyl)methyl)-4h-1,2,4-triazol-4yl)benzophenones IL44068A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US33237773A 1973-02-14 1973-02-14

Publications (2)

Publication Number Publication Date
IL44068A0 true IL44068A0 (en) 1974-05-16
IL44068A IL44068A (en) 1977-05-31

Family

ID=23297958

Family Applications (3)

Application Number Title Priority Date Filing Date
IL44068A IL44068A (en) 1973-02-14 1974-01-24 Process for the preparation of 6-phenyl-4h-s-triazolo(4,3a)(1,4)benzodiazepines and intermediate 2(2-(methanesulfonyl)methyl)-4h-1,2,4-triazol-4yl)benzophenones
IL49503A IL49503A (en) 1973-02-14 1974-01-24 Process for the preparation of 6-phenyl-4h-s-triazolo(4,3-a)(1,4)-benzodiazepines and intermediate 2-(3-(phthalimidomethyl)-4h-1,2,4-triazol-4-yl)benzophenones
IL49503A IL49503A0 (en) 1973-02-14 1976-04-30 Novel benzophenone derivatives and their preparation

Family Applications After (2)

Application Number Title Priority Date Filing Date
IL49503A IL49503A (en) 1973-02-14 1974-01-24 Process for the preparation of 6-phenyl-4h-s-triazolo(4,3-a)(1,4)-benzodiazepines and intermediate 2-(3-(phthalimidomethyl)-4h-1,2,4-triazol-4-yl)benzophenones
IL49503A IL49503A0 (en) 1973-02-14 1976-04-30 Novel benzophenone derivatives and their preparation

Country Status (16)

Country Link
JP (1) JPS49110699A (en)
AU (1) AU471038B2 (en)
BE (1) BE811025A (en)
CA (1) CA999000A (en)
CH (2) CH587263A5 (en)
DE (1) DE2402363A1 (en)
DK (1) DK140803B (en)
ES (2) ES422941A1 (en)
FR (1) FR2217335B1 (en)
GB (3) GB1454684A (en)
HU (1) HU168136B (en)
IL (3) IL44068A (en)
NL (1) NL7400958A (en)
PH (2) PH10784A (en)
SE (2) SE423546B (en)
ZA (1) ZA74466B (en)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3709898A (en) * 1971-02-09 1973-01-09 Upjohn Co Process for the production of triazolobenzodiazepines and intermediates

Also Published As

Publication number Publication date
ES445860A1 (en) 1977-05-01
CA999000A (en) 1976-10-26
GB1454684A (en) 1976-11-03
SE435285B (en) 1984-09-17
GB1454683A (en) 1976-11-03
GB1454682A (en) 1976-11-03
AU471038B2 (en) 1976-04-08
DE2402363A1 (en) 1974-08-22
ES422941A1 (en) 1976-09-16
SE423546B (en) 1982-05-10
CH586704A5 (en) 1977-04-15
ZA74466B (en) 1974-12-24
SE8107017L (en) 1981-11-25
FR2217335A1 (en) 1974-09-06
IL44068A (en) 1977-05-31
DK140803B (en) 1979-11-19
PH10784A (en) 1977-09-06
BE811025A (en) 1974-08-14
IL49503A0 (en) 1976-06-30
PH11789A (en) 1978-07-05
NL7400958A (en) 1974-08-16
JPS49110699A (en) 1974-10-22
AU6478674A (en) 1975-07-24
DK140803C (en) 1980-04-21
IL49503A (en) 1977-05-31
HU168136B (en) 1976-02-28
FR2217335B1 (en) 1977-06-10
CH587263A5 (en) 1977-04-29

Similar Documents

Publication Publication Date Title
IL45289A0 (en) Preparation of benzodiazepines
ZA741608B (en) Method of forming carrier-gels
IL44892A (en) Process for the preparation of triazolo-isoindole derivatives and certain new compounds of this type
EG11496A (en) Process for the preparation of poly-n-alkyliminoalanes
EG11189A (en) Process for preparation of new d-homosteroids
IL45740A0 (en) Process for the preparation of 6-demethyl-6-deoxy-6-methylene-tetracyclines
CH608018A5 (en) Process for the preparation of oligocarboxyalkanephosphonic acids and their use
GB1487929A (en) Process for the preparation of alpha-6-deoxytetra-cycline
CH614930A5 (en) Process for the preparation of novel omega-aminocarboxamides or -aminocarboxypolyamides
EG11639A (en) Process for the preparation of 2-nitrobenzoldehyde
CH608783A5 (en) Process for the preparation of o-diisopropylaminoethoxybutyrophenone
CH614198A5 (en) Process for the preparation of novel 4-oxo-2-imidazolidinylidene-ureas
IL44068A0 (en) Process for the preparation of new benzodiazepines and intermediates
IL45390A (en) Process for the preparation of a-ethynyl benzhydrols and some new compounds prepared thereby
CH610307A5 (en) Process for the preparation of 5-nitroimidazoles
IL44875A0 (en) Process for the 11a-dehalogenation of 11a-halotetracycline
YU306073A (en) Process for the continuous preparation of ethyl benzene
EG11476A (en) Process for the preparation of choleragen
ZA744605B (en) Process for the preparation of benzodiazepine derivatives
CA1001622A (en) Process for new benzodiazepines and intermediates
KR780000404B1 (en) Process for the preparation of chloro-acetanilides
IL45863A0 (en) Process for the preparation of benzodiazepine derivatives
CH608483A5 (en) Process for the preparation of substituted benzoylacrylanilides
CH613863A5 (en) Process for the preparation of an alloantiserum
AU6857974A (en) Method of construction