IL42166A - Drug releasing preparation - Google Patents

Drug releasing preparation

Info

Publication number
IL42166A
IL42166A IL42166A IL4216673A IL42166A IL 42166 A IL42166 A IL 42166A IL 42166 A IL42166 A IL 42166A IL 4216673 A IL4216673 A IL 4216673A IL 42166 A IL42166 A IL 42166A
Authority
IL
Israel
Prior art keywords
plasticiser
weight
releasing preparation
drug releasing
solvent membrane
Prior art date
Application number
IL42166A
Other versions
IL42166A0 (en
Inventor
E Loebel
R Bloch
O Kedem
Original Assignee
Res Prod Rehovot Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Res Prod Rehovot Ltd filed Critical Res Prod Rehovot Ltd
Priority to IL42166A priority Critical patent/IL42166A/en
Publication of IL42166A0 publication Critical patent/IL42166A0/en
Priority to ZA00742682A priority patent/ZA742682B/en
Priority to AU68402/74A priority patent/AU6840274A/en
Priority to FR7415014A priority patent/FR2227875A1/en
Priority to DE2421016A priority patent/DE2421016A1/en
Priority to JP49048382A priority patent/JPS5029731A/ja
Priority to BE143873A priority patent/BE814491A/en
Priority to NL7405903A priority patent/NL7405903A/xx
Publication of IL42166A publication Critical patent/IL42166A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/282Organic compounds, e.g. fats

Landscapes

  • Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The solubility membrane is a plasticiser contg. a thermoplastic polymer esp. PVC or PVA contg. >=40% and pref. 80% plasticiser esp. an adipate, sebacate, phosphate or phthalate digitables is compressed into a tablet with lactose which is then dipped into a soln. of cyclohexanone contg. 8% dioctyl phthalate and 2% PVC and dried. [FR2227875A1]

Claims (26)

Having now particularly described and ascertained the nature of our said invention and in what manner the same is tQ be performed, we declare that what we claim is:
1. Process for the manufacture of a drug releasin preparation, comprising encapsulating or coating a therapeutic agent in or with a solvent membrane, as hereinbefore defined.
2. Process according to claim 1, wherein there is used a solvent membrane comprising at least one plasticiser and at least one polymer reinforcing said plasticiser.
3. 5. Process according to claim 1 or 2, wherein there is used a solvent membrane comprising a plasticiser and a thermoplastic polymer reinforcing said plasticiser.
4. Process according to claim 1, 2 or 3, wherein there is used a solvent membrane wherein the polymer is poly-vinylchloride or pol vinylace ate.
5. Process according to any one of claims 1 to 4, wherein there is used a solvent membrane wherein the plasticiser is selected from the group consisting of adipates, eebacates, phosphates and phthalates.
6. Process according to any one of claims 1 to 5, wherein there is used a solvent membrane wherein the plasticiser is selected from the group consisting of butyl-phthalyl-butyl-glycolate, epoxidised soy bean oil, tri-tolyl- phosphate, dibutyl sebacate, dioctyl sebacate, tri-(diethyl-hexyl)-phosphate , 2-ethyl-hexyl-diphenyl phosphate, di-iso-butyl adipate fmethyl stearate, glycerol glyceryl monooleate, butylbenzyl phthalate, dioctyl phthalate, diphenyl-octyl phosphate, diethyl phthalate, di-(2-ethyl-hexyl)-phthalate and TBP.
7. Process according to any one of claims 1 to 6, wherein the plasticiser is used in an amount of at least 40$ by weight of the weight of the solvent membrane.
8. Process according to any one of claims 1 to 7, wherein the plasticiser is used in an amount of at least about 60$ by weight of the weight of the solvent membrane.
9. · Process according to any one of claims 1 to 8, wherein the plasticiser is used in an amount of a least about 80$ by weight of the weight of the solvent membrane.
10. Process accordin to any one of claims 1 to 9, wherein the therapeutic agent is selected from the group consisting of steroids, vitamins, antihistamines, stimulants, tranquilizers, antibiotics and arrhythmic agents.
11. Process according to any one of claims 1 to 10, wherein the therapeutic agent is selected from the group consisting of digitalis, antipyrine, procainamide hydrochlorid atropine sulfate, theophylline and dicumarol.
12. Process according to any one of claims 1 to 10, wherein the therapeutic agent is selected from the group consisting of benzodiazepines e.g. diazepam, triptylines e.g. amitriptyline , and dehydroemetine.
13. Process for the manufacture of a drug releasing preparation as hereinbefore particularly described, especially with reference to the foregoing examples.
14. A drug release preparation comprising a therapeutic agent encapsulated in or coated with a solvent membrane, whenever prepared by the process as claimed in any one of claims 1 to 13» or by an obvious equivalent thereof.
15. A drug releasing preparation which comprises a therapeutic agent being encapsulated in or coated by a solvent membranef as hereinbefore defined.
16. A drug releasing preparation according to claim 15, wherein the solvent membrane comprises at least one plasticiser and at least a polymer reinforcing said plasticiser.
17. A drug releasing preparation according to claim 15 or 16, wherein the solvent membrane comprises a plasticiser and a thermoplastic polymer reinforcing said plasticiser.
18. A drug releasing preparation according to claim 15, 16 or 17» wherein the polymer is polyvinylchloride or poly-vinylacetate.
19. A drug releasing preparation according to any one of claims 15 to 18, wherein the solvent membrane comprises a plasticiser selected from the group consisting of adipates, sebacates, phosphates and phthalates.
20. A drug releasing preparation according to any one of claims 15 to 19, wherein the solvent membrane comprises a plasticiser selected from the group consisting of butyl-phthalyl-butyl-glycolate, epoxidised soy bean oil, tri-tolyl-phosphate, dibutyl sebacate, dioctyl sebacate, tri-(diethyl-hexyl)-phosphate, 2-ethyl-hexyl-diphenyl phosphate, di-iso-butyl adipate,methyl stearate, glycerol glyceryl monooleate, butyl-benzyl phthalate , dioctyl phthalate, diphenyl-octyl phosphate, diethyl phthalate, di~(2-ethyl-hexyl)-phthalate and TBP.
21. A drug releasing preparation according to any one of claims 15 to 20, wherein the plasticiser is present in an amount of at least 40 by weight of the weight of the solvent membrane .
22. A drug releasing preparation according to an one of claims 15 to 21, wherein the plasticiser is present in an amount of at least about 60$ by weight of the weight of the solvent membrane.
23. A drug releasing preparation according to any one of claims 15 to 22, wherein the plasticiser is present in an amount of at least about 80$ by weight of the weight of the solvent membrane.
24. A drug releasing preparation according to any one of claims 15 to 23, wherein the therapeutic agent is selected from the group consisting of steroids, vitamins, antihistamines, stimulants, tranquilizers, antibiotics and arrjiytraic . agents. ■ ' '
25. A drug releasing preparation according to any one of claims 15 to 24, wherein the therapeutic agent is selected from the group consisting of digitalis, antipyrine, procainamid hydrochloride, atropine sulfate, theophylline and dicumarol.
26. A drug releasing preparation according to an one of claims 15 to 24, wherein the therapeutic agent is selected from the group consisting of benzodiazepines e.g. diazepam, triptylines e.g. amitriptyline , and dehydroemetine. For the Applicants Dr.Yitzhak Hess
0. ,\ m
IL42166A 1973-05-02 1973-05-02 Drug releasing preparation IL42166A (en)

Priority Applications (8)

Application Number Priority Date Filing Date Title
IL42166A IL42166A (en) 1973-05-02 1973-05-02 Drug releasing preparation
ZA00742682A ZA742682B (en) 1973-05-02 1974-04-29 Drug delivery preparation with controlled release time and rate
AU68402/74A AU6840274A (en) 1973-05-02 1974-04-30 Composition
FR7415014A FR2227875A1 (en) 1973-05-02 1974-04-30 Slow release agents for drugs - comprising drugs enrobed or encapsulated with a solubility
DE2421016A DE2421016A1 (en) 1973-05-02 1974-04-30 PREPARATION
JP49048382A JPS5029731A (en) 1973-05-02 1974-05-01
BE143873A BE814491A (en) 1973-05-02 1974-05-02 PHARMACEUTICAL COMPOSITION RELEASING THE ACTIVE SUBSTANCE AT A PRE-DETERMINED RATE.
NL7405903A NL7405903A (en) 1973-05-02 1974-05-02

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IL42166A IL42166A (en) 1973-05-02 1973-05-02 Drug releasing preparation

Publications (2)

Publication Number Publication Date
IL42166A0 IL42166A0 (en) 1973-07-30
IL42166A true IL42166A (en) 1976-01-30

Family

ID=11047093

Family Applications (1)

Application Number Title Priority Date Filing Date
IL42166A IL42166A (en) 1973-05-02 1973-05-02 Drug releasing preparation

Country Status (8)

Country Link
JP (1) JPS5029731A (en)
AU (1) AU6840274A (en)
BE (1) BE814491A (en)
DE (1) DE2421016A1 (en)
FR (1) FR2227875A1 (en)
IL (1) IL42166A (en)
NL (1) NL7405903A (en)
ZA (1) ZA742682B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE426548B (en) * 1978-12-05 1983-01-31 Haessle Ab SOLID PHARMACEUTICAL PREPARATION INCLUDING A THERAPEUTICALLY EFFECTIVE HEART GYCLOSIDE AND POLYMER
SE7813246L (en) * 1978-12-22 1980-06-23 Haessle Ab FIXED PHARMACEUTICAL PREPARATION INCLUDING BODIES WITH MULTIPLE LAYERS

Also Published As

Publication number Publication date
JPS5029731A (en) 1975-03-25
DE2421016A1 (en) 1974-11-21
NL7405903A (en) 1974-11-05
ZA742682B (en) 1975-08-27
BE814491A (en) 1974-09-02
IL42166A0 (en) 1973-07-30
AU6840274A (en) 1975-10-30
FR2227875A1 (en) 1974-11-29
FR2227875B1 (en) 1977-11-04

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