IL325580A - Treatment of chronic pain or gastrointestinal disorders using buprenorphine dimer - Google Patents

Treatment of chronic pain or gastrointestinal disorders using buprenorphine dimer

Info

Publication number
IL325580A
IL325580A IL325580A IL32558025A IL325580A IL 325580 A IL325580 A IL 325580A IL 325580 A IL325580 A IL 325580A IL 32558025 A IL32558025 A IL 32558025A IL 325580 A IL325580 A IL 325580A
Authority
IL
Israel
Prior art keywords
treatment
chronic pain
gastrointestinal disorders
buprenorphine dimer
buprenorphine
Prior art date
Application number
IL325580A
Other languages
Hebrew (he)
Inventor
Nikhilesh Singh
Original Assignee
Dimerx Inc
Nikhilesh Singh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dimerx Inc, Nikhilesh Singh filed Critical Dimerx Inc
Publication of IL325580A publication Critical patent/IL325580A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/468-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12Antidiarrhoeals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/08Bridged systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Emergency Medicine (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL325580A 2023-07-10 2025-12-23 Treatment of chronic pain or gastrointestinal disorders using buprenorphine dimer IL325580A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202363512783P 2023-07-10 2023-07-10
US202463568538P 2024-03-22 2024-03-22
PCT/US2024/037128 WO2025014912A1 (en) 2023-07-10 2024-07-09 Treatment of chronic pain or gastrointestinal disorders using buprenorphine dimer

Publications (1)

Publication Number Publication Date
IL325580A true IL325580A (en) 2026-02-01

Family

ID=94216216

Family Applications (1)

Application Number Title Priority Date Filing Date
IL325580A IL325580A (en) 2023-07-10 2025-12-23 Treatment of chronic pain or gastrointestinal disorders using buprenorphine dimer

Country Status (6)

Country Link
EP (1) EP4743466A1 (en)
KR (1) KR20260055394A (en)
CN (1) CN121773116A (en)
AU (1) AU2024288358A1 (en)
IL (1) IL325580A (en)
WO (1) WO2025014912A1 (en)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUE036084T2 (en) * 2014-04-28 2018-06-28 Orphomed Inc Buprenorphine dimer and its use in the treatment of gastrointestinal disorders
TW201725040A (en) * 2015-10-26 2017-07-16 奧佛麥德公司 Use of buprenorphine dimer in the treatment of peripheral neuropathic pain
WO2018222921A1 (en) * 2017-05-31 2018-12-06 Napo Pharmaceuticals, Inc. Methods and compositions for treating bile acid diarrhea, diarrhea associated with small intestine resection or gallbladder removal, and short bowel syndrome
WO2021262763A1 (en) * 2020-06-23 2021-12-30 Arriba Biopharma, Inc. Opioid receptor modulator and use thereof

Also Published As

Publication number Publication date
WO2025014912A1 (en) 2025-01-16
EP4743466A1 (en) 2026-05-20
CN121773116A (en) 2026-03-31
AU2024288358A1 (en) 2026-01-22
KR20260055394A (en) 2026-04-23

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