IL302948A - תכשירים למתן מעכבים של cgrp - Google Patents
תכשירים למתן מעכבים של cgrpInfo
- Publication number
- IL302948A IL302948A IL302948A IL30294823A IL302948A IL 302948 A IL302948 A IL 302948A IL 302948 A IL302948 A IL 302948A IL 30294823 A IL30294823 A IL 30294823A IL 302948 A IL302948 A IL 302948A
- Authority
- IL
- Israel
- Prior art keywords
- pharmaceutical composition
- composition according
- cgrp
- weight
- alkyl glycoside
- Prior art date
Links
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- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2063—Proteins, e.g. gelatin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Pain & Pain Management (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202063115789P | 2020-11-19 | 2020-11-19 | |
| US202063126550P | 2020-12-17 | 2020-12-17 | |
| PCT/US2021/059801 WO2022109077A1 (en) | 2020-11-19 | 2021-11-18 | Compositions for improved delivery of cgrp inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL302948A true IL302948A (he) | 2023-07-01 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL302948A IL302948A (he) | 2020-11-19 | 2021-11-18 | תכשירים למתן מעכבים של cgrp |
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| EP (1) | EP4247364A4 (he) |
| JP (1) | JP2023551146A (he) |
| KR (1) | KR20230088442A (he) |
| AU (1) | AU2021385052A1 (he) |
| CA (1) | CA3202137A1 (he) |
| IL (1) | IL302948A (he) |
| MX (1) | MX2023005846A (he) |
| WO (1) | WO2022109077A1 (he) |
| ZA (1) | ZA202304727B (he) |
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| CN115154469A (zh) * | 2022-07-22 | 2022-10-11 | 中国科学院广州生物医药与健康研究院 | 瑞美吉泮或其药学上可接受的盐在制备预防或治疗肥胖的药物中的应用 |
| CN117503704B (zh) * | 2023-11-09 | 2025-07-11 | 广州新济药业科技有限公司 | 一种作用于中枢神经系统的鼻喷雾剂及其制备方法及应用 |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| US8268791B2 (en) * | 2004-08-25 | 2012-09-18 | Aegis Therapeutics, Llc. | Alkylglycoside compositions for drug administration |
| US8715715B2 (en) * | 2008-11-03 | 2014-05-06 | Nal Pharmaceuticals Ltd. | Dosage form for insertion into the mouth |
| US8481546B2 (en) * | 2010-03-30 | 2013-07-09 | Bristol-Myers Squibb Company | CGRP receptor antagonist |
| JP6491669B2 (ja) * | 2014-02-05 | 2019-03-27 | メルク・シャープ・アンド・ドーム・コーポレーションMerck Sharp & Dohme Corp. | Cgrp活性化合物の錠剤製剤 |
| US20160346198A1 (en) * | 2014-02-05 | 2016-12-01 | Merck Sharp & Dohme Corp. | Novel disintegration systems for pharmaceutical dosage forms |
| EP3426288A4 (en) * | 2016-04-15 | 2019-10-30 | Alder Biopharmaceuticals, Inc. | ANTI-PACAP ANTIBODIES AND USES THEREOF |
| SI4088720T1 (sl) * | 2018-03-25 | 2026-01-30 | Pfizer Ireland Pharmaceuticals Unlimited Company | Rimegepant za motnje, povezane s cgrp |
| JP2022517433A (ja) * | 2019-01-20 | 2022-03-08 | バイオヘイブン・ファーマシューティカル・ホールディング・カンパニー・リミテッド | 突出性の片頭痛を処置するためのcgrpアンタゴニスト |
| BR112021018817A2 (pt) * | 2019-04-11 | 2021-11-23 | Scherer Technologies Llc R P | Formulação para suprimento oral de proteínas, peptídeos e moléculas pequenas com pouca permeabilidade |
| WO2020232379A1 (en) * | 2019-05-16 | 2020-11-19 | Aegis Therapeutics, Llc | Oil-soluble drug containing compositions and methods of use thereof |
| CA3156009A1 (en) * | 2019-09-25 | 2021-04-01 | Allergan Pharmaceuticals International Limited | POLYTHERAPY WITH CGRP ANTAGONISTS |
| CA3164445A1 (en) * | 2019-12-17 | 2021-06-24 | Biohaven Pharmaceutical Holding Company Ltd. | Intranasal pharmaceutical compositions of cgrp inhibitors |
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2021
- 2021-11-18 IL IL302948A patent/IL302948A/he unknown
- 2021-11-18 CA CA3202137A patent/CA3202137A1/en active Pending
- 2021-11-18 EP EP21895549.0A patent/EP4247364A4/en active Pending
- 2021-11-18 KR KR1020237016343A patent/KR20230088442A/ko not_active Ceased
- 2021-11-18 WO PCT/US2021/059801 patent/WO2022109077A1/en not_active Ceased
- 2021-11-18 JP JP2023529881A patent/JP2023551146A/ja active Pending
- 2021-11-18 AU AU2021385052A patent/AU2021385052A1/en not_active Abandoned
- 2021-11-18 MX MX2023005846A patent/MX2023005846A/es unknown
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2023
- 2023-04-24 ZA ZA2023/04727A patent/ZA202304727B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP4247364A4 (en) | 2024-10-23 |
| MX2023005846A (es) | 2023-06-02 |
| WO2022109077A1 (en) | 2022-05-27 |
| EP4247364A1 (en) | 2023-09-27 |
| AU2021385052A9 (en) | 2024-05-02 |
| CA3202137A1 (en) | 2022-05-27 |
| ZA202304727B (en) | 2023-12-20 |
| AU2021385052A1 (en) | 2023-06-01 |
| JP2023551146A (ja) | 2023-12-07 |
| KR20230088442A (ko) | 2023-06-19 |
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