IL211996A0 - Process for the preparation of substituted phenylalanines - Google Patents

Process for the preparation of substituted phenylalanines

Info

Publication number
IL211996A0
IL211996A0 IL211996A IL21199611A IL211996A0 IL 211996 A0 IL211996 A0 IL 211996A0 IL 211996 A IL211996 A IL 211996A IL 21199611 A IL21199611 A IL 21199611A IL 211996 A0 IL211996 A0 IL 211996A0
Authority
IL
Israel
Prior art keywords
preparation
substituted phenylalanines
phenylalanines
substituted
Prior art date
Application number
IL211996A
Original Assignee
Lexicon Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lexicon Pharmaceuticals Inc filed Critical Lexicon Pharmaceuticals Inc
Publication of IL211996A0 publication Critical patent/IL211996A0/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C43/00—Ethers; Compounds having groups, groups or groups
    • C07C43/02—Ethers
    • C07C43/20—Ethers having an ether-oxygen atom bound to a carbon atom of a six-membered aromatic ring
    • C07C43/23—Ethers having an ether-oxygen atom bound to a carbon atom of a six-membered aromatic ring containing hydroxy or O-metal groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
IL211996A 2008-10-24 2011-03-29 Process for the preparation of substituted phenylalanines IL211996A0 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US2008/081054 WO2010047712A1 (en) 2008-10-24 2008-10-24 Process for the preparation of substituted phenylalanines

Publications (1)

Publication Number Publication Date
IL211996A0 true IL211996A0 (en) 2011-06-30

Family

ID=40785295

Family Applications (1)

Application Number Title Priority Date Filing Date
IL211996A IL211996A0 (en) 2008-10-24 2011-03-29 Process for the preparation of substituted phenylalanines

Country Status (11)

Country Link
EP (1) EP2358685A1 (en)
JP (1) JP2012506427A (en)
KR (1) KR20110074875A (en)
CN (1) CN102203069A (en)
AU (1) AU2008363274A1 (en)
BR (1) BRPI0823136A2 (en)
CA (1) CA2741563A1 (en)
IL (1) IL211996A0 (en)
MX (1) MX2011004168A (en)
RU (1) RU2011120822A (en)
WO (1) WO2010047712A1 (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2015089137A1 (en) * 2013-12-11 2015-06-18 Karos Pharmaceuticals, Inc. Acylguanidines as tryptophan hydroxylase inhibitors
EP4056560A1 (en) 2018-03-08 2022-09-14 Incyte Corporation Aminopyrazine diol compounds as pi3k-y inhibitors
WO2020010003A1 (en) 2018-07-02 2020-01-09 Incyte Corporation AMINOPYRAZINE DERIVATIVES AS PI3K-γ INHIBITORS

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ568946A (en) * 2005-12-29 2010-07-30 Lexicon Pharmaceuticals Inc Multicyclic amino acid derivatives and methods of their use
UA99270C2 (en) * 2006-12-12 2012-08-10 Лексикон Фармасьютикалз, Инк. 4-phenyl-6-(2,2,2-trifluoro-1-phenylethoxy)pyrimidine-based compounds and methods of their use

Also Published As

Publication number Publication date
BRPI0823136A2 (en) 2015-06-16
AU2008363274A1 (en) 2010-04-29
KR20110074875A (en) 2011-07-04
JP2012506427A (en) 2012-03-15
CA2741563A1 (en) 2010-04-29
WO2010047712A1 (en) 2010-04-29
CN102203069A (en) 2011-09-28
EP2358685A1 (en) 2011-08-24
MX2011004168A (en) 2011-05-23
RU2011120822A (en) 2012-11-27

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