IL161157A - 3-azabicyclo (3.1.0) hexane derivatives as opioid receptor antagonists - Google Patents
3-azabicyclo (3.1.0) hexane derivatives as opioid receptor antagonistsInfo
- Publication number
- IL161157A IL161157A IL161157A IL16115704A IL161157A IL 161157 A IL161157 A IL 161157A IL 161157 A IL161157 A IL 161157A IL 16115704 A IL16115704 A IL 16115704A IL 161157 A IL161157 A IL 161157A
- Authority
- IL
- Israel
- Prior art keywords
- azabicyclo
- receptor antagonists
- opioid receptor
- hexane derivatives
- hexane
- Prior art date
Links
- 150000005228 3‐azabicyclo[3.1.0]hexanes Chemical class 0.000 title 1
- 229940123257 Opioid receptor antagonist Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/10—Laxatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/04—Antipruritics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/36—Opioid-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/04—Compounds containing oxirane rings containing only hydrogen and carbon atoms in addition to the ring oxygen atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Hospice & Palliative Care (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- Gynecology & Obstetrics (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Psychology (AREA)
- Child & Adolescent Psychology (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
- Diabetes (AREA)
- Immunology (AREA)
- Otolaryngology (AREA)
- Dermatology (AREA)
- Nutrition Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US33851101P | 2001-10-22 | 2001-10-22 | |
| PCT/IB2002/003668 WO2003035622A1 (en) | 2001-10-22 | 2002-09-09 | 3-azabicyclo (3.1.0) hexane derivatives as opioid receptor antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL161157A true IL161157A (en) | 2009-09-01 |
Family
ID=23325099
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL16115702A IL161157A0 (en) | 2001-10-22 | 2002-09-09 | 3-azabicyclo (3.1.0) hexane derivatives as opioid receptor antagonists |
| IL161157A IL161157A (en) | 2001-10-22 | 2004-03-29 | 3-azabicyclo (3.1.0) hexane derivatives as opioid receptor antagonists |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL16115702A IL161157A0 (en) | 2001-10-22 | 2002-09-09 | 3-azabicyclo (3.1.0) hexane derivatives as opioid receptor antagonists |
Country Status (41)
| Country | Link |
|---|---|
| US (3) | US7049335B2 (en) |
| EP (1) | EP1440059B1 (en) |
| JP (2) | JP4155522B2 (en) |
| KR (1) | KR100621292B1 (en) |
| CN (1) | CN100368398C (en) |
| AP (1) | AP1816A (en) |
| AR (1) | AR036905A1 (en) |
| AT (1) | ATE392415T1 (en) |
| AU (1) | AU2002329557B2 (en) |
| BR (1) | BR0213464A (en) |
| CA (1) | CA2463264C (en) |
| CR (1) | CR7317A (en) |
| DE (1) | DE60226161T2 (en) |
| DK (1) | DK1440059T3 (en) |
| EA (1) | EA006708B1 (en) |
| EC (1) | ECSP045077A (en) |
| ES (1) | ES2302839T3 (en) |
| GE (1) | GEP20084300B (en) |
| GT (1) | GT200200216A (en) |
| HN (1) | HN2002000299A (en) |
| HR (1) | HRP20040288A2 (en) |
| HU (1) | HUP0401884A2 (en) |
| IL (2) | IL161157A0 (en) |
| IS (1) | IS7187A (en) |
| MA (1) | MA27141A1 (en) |
| MX (1) | MXPA04003730A (en) |
| MY (1) | MY136580A (en) |
| NO (1) | NO329092B1 (en) |
| NZ (1) | NZ531807A (en) |
| OA (1) | OA12711A (en) |
| PA (1) | PA8556701A1 (en) |
| PE (1) | PE20030610A1 (en) |
| PL (1) | PL368919A1 (en) |
| PT (1) | PT1440059E (en) |
| RS (1) | RS25104A (en) |
| SI (1) | SI1440059T1 (en) |
| SV (1) | SV2004001363A (en) |
| TN (1) | TNSN04071A1 (en) |
| UA (1) | UA75714C2 (en) |
| WO (1) | WO2003035622A1 (en) |
| ZA (1) | ZA200402172B (en) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE424385T1 (en) | 2001-04-18 | 2009-03-15 | Euro Celtique Sa | 1-(4-PIPERIDINYL)-1,3-DIHYDRO-2H-BENZOXAZOLE-2-ONE DERIVATIVES AND RELATED COMPOUNDS AS NOCICEPTIN ANALOGUES AND ORL1 LIGANDS FOR THE TREATMENT OF PAIN |
| IL161157A0 (en) * | 2001-10-22 | 2004-08-31 | Pfizer Prod Inc | 3-azabicyclo (3.1.0) hexane derivatives as opioid receptor antagonists |
| CA2522323C (en) * | 2003-04-14 | 2009-09-15 | Pfizer Products Inc. | 3-azabicyclo[3.2.1]octane derivatives as opioid receptor ligands |
| US20050043327A1 (en) * | 2003-08-21 | 2005-02-24 | Pfizer Inc | Pharmaceutical composition for the prevention and treatment of addiction in a mammal |
| US7153976B2 (en) * | 2003-10-06 | 2006-12-26 | Pfizer Inc. | Purification process for an azabicyclo[3.1.0]hexane compound |
| AP2006003592A0 (en) * | 2003-10-14 | 2006-04-30 | Pfizer Prod Inc | Bicyclic [3.1.0] derivatives as glycine transporter inhibitors. |
| RU2006112576A (en) * | 2003-10-16 | 2006-08-27 | Пфайзер Продактс Инк. (Us) | PRODUCTION OF 3-AZABICYCLO [3.1.0] HEXANE DERIVATIVES |
| ATE451364T1 (en) * | 2004-02-23 | 2009-12-15 | Glaxo Group Ltd | AZABICYCLOÄ3.1.0ÜHEXANE DERIVATIVES SUITABLE AS MODULATORS OF THE DOPAMINE D3 RECEPTOR |
| US7855294B2 (en) * | 2004-03-05 | 2010-12-21 | Banyu Pharmaceutical Co., Ltd. | Cycloalkanopyridine derivative |
| US20080227803A1 (en) * | 2004-12-14 | 2008-09-18 | Shioonogi & Co., Ltd., A Legal Entity Of Japan | Indolomorphinan Derivative Having Carboxy in 6'-Position |
| GB0512099D0 (en) * | 2005-06-14 | 2005-07-20 | Glaxo Group Ltd | Compounds |
| GB0517191D0 (en) | 2005-08-22 | 2005-09-28 | Glaxo Group Ltd | Compounds |
| US7592461B2 (en) * | 2005-12-21 | 2009-09-22 | Bristol-Myers Squibb Company | Indane modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof |
| MY145633A (en) | 2006-03-01 | 2012-03-15 | Theravance Inc | 8-azabicyclo[3.2.1]octane compounds as mu opioid receptor antagonists |
| WO2008075162A2 (en) * | 2006-12-15 | 2008-06-26 | Pfizer Limited | Selective mu opioid receptor antagonists for the treatment of female sexual dysfunction |
| TWI409067B (en) | 2007-02-28 | 2013-09-21 | Theravance Inc | Crystalline forms of an 8-azabicyclo[3.2.1]octane compound |
| US7691878B2 (en) * | 2007-08-27 | 2010-04-06 | Theravance, Inc. | Heteroarylalkyl-8-azabicyclo[3.2.1]octane compounds as mu opioid receptor antagonists |
| TWI423801B (en) * | 2007-08-27 | 2014-01-21 | Theravance Inc | 8-azabicyclo[3.2.1]octyl-2-hydroxybenzamide compounds as mu opioid receptor antagonists |
| WO2009029257A1 (en) * | 2007-08-27 | 2009-03-05 | Theravance, Inc. | Disubstituted alkyl-8-azabicyclo [3.2.1.] octane compounds as mu opioid receptor antagonists |
| WO2009029252A1 (en) * | 2007-08-27 | 2009-03-05 | Theravance, Inc. | Amidoalkyl-8-azabicyclo[3.2.1]octane compounds as mu opioid receptor antagonists |
| JP2013542929A (en) | 2010-09-28 | 2013-11-28 | パナセア バイオテック リミテッド | New bicyclo ring compounds |
| WO2015076310A1 (en) | 2013-11-20 | 2015-05-28 | 株式会社 三和化学研究所 | Novel 3-azabicyclo[3.1.0]hexane derivative and use thereof for medical purposes |
| WO2016186184A1 (en) * | 2015-05-20 | 2016-11-24 | 株式会社 三和化学研究所 | Crystal of salt of novel 3-azabicyclo[3.1.0]hexane derivative and pharmaceutical use thereof |
| WO2018159716A1 (en) | 2017-03-02 | 2018-09-07 | 株式会社 三和化学研究所 | Therapeutic agent for alcohol use disorders |
Family Cites Families (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2099214A (en) * | 1937-11-16 | Process fob forming the sulphuric | ||
| US2099216A (en) * | 1934-05-04 | 1937-11-16 | Frederick H Nass | Metal testing machine |
| US3004340A (en) * | 1959-09-24 | 1961-10-17 | Bernice L Collins | Kitchen utensil |
| US3078282A (en) * | 1960-01-02 | 1963-02-19 | Bayer Ag | Anthraquinone dyestuffs |
| EP0287339B1 (en) | 1987-04-16 | 1994-08-17 | Eli Lilly And Company | Piperidine opioid antagonists |
| JPH04155522A (en) * | 1990-10-19 | 1992-05-28 | Nec Corp | First-in-random-out circuit |
| US5159081A (en) | 1991-03-29 | 1992-10-27 | Eli Lilly And Company | Intermediates of peripherally selective n-carbonyl-3,4,4-trisubstituted piperidine opioid antagonists |
| CZ284993B6 (en) | 1991-03-29 | 1999-04-14 | Eli Lilly And Company | Piperidine derivative, process of its preparation and pharmaceutical composition containing thereof |
| GB9725114D0 (en) * | 1997-11-28 | 1998-01-28 | Pfizer Ltd | Treatment of pruritus |
| GB9810671D0 (en) * | 1998-05-18 | 1998-07-15 | Pfizer Ltd | Anti-pruritic agents |
| TWI244481B (en) * | 1998-12-23 | 2005-12-01 | Pfizer | 3-azabicyclo[3.1.0]hexane derivatives useful in therapy |
| GB9912415D0 (en) * | 1999-05-28 | 1999-07-28 | Pfizer Ltd | Compounds useful in therapy |
| GB9912411D0 (en) * | 1999-05-28 | 1999-07-28 | Pfizer Ltd | Compounds useful in therapy |
| GB9912413D0 (en) * | 1999-05-28 | 1999-07-28 | Pfizer Ltd | Compounds useful in therapy |
| GB9912410D0 (en) * | 1999-05-28 | 1999-07-28 | Pfizer Ltd | Compounds useful in therapy |
| US20020064825A1 (en) * | 2000-05-19 | 2002-05-30 | Lewis Marilyn Evelyn | Novel polypeptide |
| US20030207876A1 (en) * | 2000-06-23 | 2003-11-06 | Banks Bernard Joseph | 3-Azabicyclo[3.1.0]hexane derivatives useful in therapy |
| GB0015562D0 (en) * | 2000-06-23 | 2000-08-16 | Pfizer Ltd | Heterocycles |
| US20020025948A1 (en) * | 2000-06-23 | 2002-02-28 | Banks Bernard Joseph | 3-azabicyclo[3.1.0]hexane derivatives useful in therapy |
| DE10042885A1 (en) * | 2000-08-31 | 2002-03-14 | Heidelberger Druckmasch Ag | Sheet transporting cylinder for printing press has throttled air jets set at minimum format |
| IL161157A0 (en) | 2001-10-22 | 2004-08-31 | Pfizer Prod Inc | 3-azabicyclo (3.1.0) hexane derivatives as opioid receptor antagonists |
| ATE308522T1 (en) | 2002-05-30 | 2005-11-15 | Lilly Co Eli | OPIOID RECEPTOR ANTAGONISTS |
| US20040204453A1 (en) * | 2003-04-14 | 2004-10-14 | Pfizer Inc | 4-Phenyl-piperidine compounds and their use as modulators of opioid receptors |
| US7056930B2 (en) * | 2003-04-14 | 2006-06-06 | Pfizer Inc. | 2-Azabicyclo[3.3.1]nonane derivatives |
| US20050043327A1 (en) * | 2003-08-21 | 2005-02-24 | Pfizer Inc | Pharmaceutical composition for the prevention and treatment of addiction in a mammal |
| US7153976B2 (en) * | 2003-10-06 | 2006-12-26 | Pfizer Inc. | Purification process for an azabicyclo[3.1.0]hexane compound |
-
2002
- 2002-09-09 IL IL16115702A patent/IL161157A0/en unknown
- 2002-09-09 MX MXPA04003730A patent/MXPA04003730A/en active IP Right Grant
- 2002-09-09 CA CA002463264A patent/CA2463264C/en not_active Expired - Fee Related
- 2002-09-09 PL PL02368919A patent/PL368919A1/en not_active Application Discontinuation
- 2002-09-09 JP JP2003538138A patent/JP4155522B2/en not_active Expired - Fee Related
- 2002-09-09 AT AT02765197T patent/ATE392415T1/en not_active IP Right Cessation
- 2002-09-09 GE GEAP20028173A patent/GEP20084300B/en unknown
- 2002-09-09 HR HRP20040288 patent/HRP20040288A2/en not_active Application Discontinuation
- 2002-09-09 SI SI200230688T patent/SI1440059T1/en unknown
- 2002-09-09 UA UA20040402979A patent/UA75714C2/en unknown
- 2002-09-09 BR BR0213464-0A patent/BR0213464A/en not_active IP Right Cessation
- 2002-09-09 PT PT02765197T patent/PT1440059E/en unknown
- 2002-09-09 ES ES02765197T patent/ES2302839T3/en not_active Expired - Lifetime
- 2002-09-09 KR KR1020047006011A patent/KR100621292B1/en not_active Expired - Fee Related
- 2002-09-09 HU HU0401884A patent/HUP0401884A2/en unknown
- 2002-09-09 WO PCT/IB2002/003668 patent/WO2003035622A1/en not_active Ceased
- 2002-09-09 DE DE60226161T patent/DE60226161T2/en not_active Expired - Lifetime
- 2002-09-09 CN CNB028208854A patent/CN100368398C/en not_active Expired - Fee Related
- 2002-09-09 AU AU2002329557A patent/AU2002329557B2/en not_active Ceased
- 2002-09-09 DK DK02765197T patent/DK1440059T3/en active
- 2002-09-09 OA OA1200400109A patent/OA12711A/en unknown
- 2002-09-09 RS YUP-251/04A patent/RS25104A/en unknown
- 2002-09-09 NZ NZ531807A patent/NZ531807A/en unknown
- 2002-09-09 EP EP02765197A patent/EP1440059B1/en not_active Expired - Lifetime
- 2002-09-09 AP APAP/P/2004/003007A patent/AP1816A/en active
- 2002-09-09 EA EA200400467A patent/EA006708B1/en not_active IP Right Cessation
- 2002-10-17 MY MYPI20023878A patent/MY136580A/en unknown
- 2002-10-17 PA PA20028556701A patent/PA8556701A1/en unknown
- 2002-10-18 PE PE2002001032A patent/PE20030610A1/en not_active Application Discontinuation
- 2002-10-18 HN HN2002000299A patent/HN2002000299A/en unknown
- 2002-10-21 AR ARP020103960A patent/AR036905A1/en unknown
- 2002-10-21 SV SV2002001363A patent/SV2004001363A/en not_active Application Discontinuation
- 2002-10-22 GT GT200200216A patent/GT200200216A/en unknown
- 2002-10-22 US US10/278,142 patent/US7049335B2/en not_active Expired - Fee Related
-
2004
- 2004-03-18 IS IS7187A patent/IS7187A/en unknown
- 2004-03-18 ZA ZA200402172A patent/ZA200402172B/en unknown
- 2004-03-29 IL IL161157A patent/IL161157A/en not_active IP Right Cessation
- 2004-04-15 MA MA27630A patent/MA27141A1/en unknown
- 2004-04-20 CR CR7317A patent/CR7317A/en unknown
- 2004-04-21 NO NO20041626A patent/NO329092B1/en not_active IP Right Cessation
- 2004-04-21 TN TNP2004000071A patent/TNSN04071A1/en unknown
- 2004-04-22 EC EC2004005077A patent/ECSP045077A/en unknown
-
2005
- 2005-02-24 US US11/066,095 patent/US20050171178A1/en not_active Abandoned
-
2006
- 2006-03-01 US US11/366,903 patent/US20070054950A1/en not_active Abandoned
-
2007
- 2007-10-19 JP JP2007272602A patent/JP2008069169A/en active Pending
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| IL161157A (en) | 3-azabicyclo (3.1.0) hexane derivatives as opioid receptor antagonists | |
| PL365377A1 (en) | Amide derivatives as nmda receptor antagonists | |
| IL162377A0 (en) | 5,6-Diaryl-pyrazine-2-amide derivatives as cb1 antagonists | |
| ZA200408670B (en) | Trizole derivatives as tachykinin receptor antagonists. | |
| AU2002367424A1 (en) | Androgen receptor antagonists | |
| AUPR833401A0 (en) | G protein-coupled receptor antagonists | |
| MXPA03006991A (en) | Piperidinee derivatives as neurokinin 1 antagonists. | |
| IL153427A0 (en) | 3-azabicyclo (3.1.0) hexane derivatives having opioid receptor affinity | |
| PL356990A1 (en) | Isoxazolecarboxamide derivatives as alpha1-adrenergic receptor antagonists | |
| AU2002366320A1 (en) | Lactams as tachykinin antagonists | |
| AU2002365655A1 (en) | 5-ht7 receptor antagonists | |
| PL370799A1 (en) | Aminotetralin derivatives as muscarinic receptor antagonists | |
| EP1359915A4 (en) | Urotensin-ii receptor antagonists | |
| IL144299A0 (en) | N-triazolymethyl-piperazine derivatives as neurokinin receptor antagonists | |
| AU2002216079A1 (en) | Bombesin receptor antagonists | |
| AU1100300A (en) | Piperidyloxadiazoles as dopamine receptor antagonists | |
| GB0203412D0 (en) | 5-HT 2B receptor antagonists | |
| AU2002217095A1 (en) | Bombesin receptor antagonists | |
| PL370821A1 (en) | N-ureido-piperidines as antagonists viii for ccr-3 receptor | |
| PL370367A1 (en) | Ccr-3 receptor antagonists v | |
| IL158063A0 (en) | Crf receptor antagonists | |
| HK1067366A (en) | Lactam derivatives as antagonists for human 11cby receptors | |
| AU2002351478A1 (en) | 3,4-di-substituted maleimide compounds as cxc-chemokine receptor antagonists | |
| HK1062301A (en) | 3,4-di-substituted maleimide compounds as cxc-chemokine receptor antagonists | |
| AU2002235453A1 (en) | Urotensin-ii receptor antagonists |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FF | Patent granted | ||
| KB | Patent renewed | ||
| MM9K | Patent not in force due to non-payment of renewal fees |