IL138228A0 - Glycine transport inhibitors - Google Patents
Glycine transport inhibitorsInfo
- Publication number
- IL138228A0 IL138228A0 IL13822899A IL13822899A IL138228A0 IL 138228 A0 IL138228 A0 IL 138228A0 IL 13822899 A IL13822899 A IL 13822899A IL 13822899 A IL13822899 A IL 13822899A IL 138228 A0 IL138228 A0 IL 138228A0
- Authority
- IL
- Israel
- Prior art keywords
- transport inhibitors
- glycine transport
- glycine
- inhibitors
- transport
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP98200701 | 1998-03-06 | ||
| PCT/EP1999/001309 WO1999044596A2 (en) | 1998-03-06 | 1999-02-26 | Glycine transport inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL138228A0 true IL138228A0 (en) | 2001-10-31 |
Family
ID=8233444
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL13822899A IL138228A0 (en) | 1998-03-06 | 1999-02-26 | Glycine transport inhibitors |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP1059922A2 (en) |
| JP (1) | JP2002505277A (en) |
| KR (1) | KR20010032968A (en) |
| CN (1) | CN1292698A (en) |
| AU (1) | AU3408999A (en) |
| BG (1) | BG104685A (en) |
| BR (1) | BR9907951A (en) |
| CA (1) | CA2322164A1 (en) |
| EE (1) | EE200000482A (en) |
| HR (1) | HRP20000523A2 (en) |
| HU (1) | HUP0101048A2 (en) |
| IL (1) | IL138228A0 (en) |
| NO (1) | NO20004431L (en) |
| PL (1) | PL343435A1 (en) |
| SK (1) | SK13082000A3 (en) |
| TR (1) | TR200002567T2 (en) |
| WO (1) | WO1999044596A2 (en) |
Families Citing this family (32)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU774829B2 (en) | 1999-06-28 | 2004-07-08 | Janssen Pharmaceutica N.V. | Respiratory syncytial virus replication inhibitors |
| UA73749C2 (en) * | 1999-11-01 | 2005-09-15 | Diarylenines | |
| US20030176461A1 (en) * | 2000-04-20 | 2003-09-18 | Egle Ian R. | Aminopiperidines |
| DE10040016A1 (en) * | 2000-08-16 | 2002-02-28 | Boehringer Ingelheim Pharma | Novel beta-amyloid inhibitors, process for their preparation and their use as pharmaceuticals |
| AU2001288896A1 (en) | 2000-09-08 | 2002-03-22 | Gliatech, Inc. | Substituted hydrazine derivatives |
| US20020082283A1 (en) | 2000-09-14 | 2002-06-27 | Gliatech, Inc. | Nitrogen-containing compounds and their use as glycine transport inhibitors |
| AR032653A1 (en) | 2001-02-09 | 2003-11-19 | Telik Inc | HYPERCYCLIC INHIBITORS OF THE GLICINE TRANSPORTER 2 PHARMACEUTICAL COMPOSITIONS, USE AND METHODS. |
| US7030150B2 (en) | 2001-05-11 | 2006-04-18 | Trimeris, Inc. | Benzimidazole compounds and antiviral uses thereof |
| JP4563387B2 (en) | 2003-09-09 | 2010-10-13 | エフ．ホフマン−ラ ロシュ アーゲー | 1-Benzoyl-piperazine derivatives as glycine uptake inhibitors for the treatment of psychosis |
| PT1663232E (en) * | 2003-09-09 | 2007-12-12 | Hoffmann La Roche | 1-(2-amino-benzoyl)-piperazine derivatives as glycine uptake inhibitors for the treatment of psychoses |
| WO2005058885A2 (en) * | 2003-12-18 | 2005-06-30 | Glaxo Group Limited | Piperidine derivatives and their use as glycine transporter inhibitors |
| TW200630337A (en) | 2004-10-14 | 2006-09-01 | Euro Celtique Sa | Piperidinyl compounds and the use thereof |
| NZ555290A (en) * | 2004-12-09 | 2009-09-25 | Hoffmann La Roche | Phenyl-piperazin methanone derivatives |
| DE602005019465D1 (en) * | 2004-12-15 | 2010-04-01 | Hoffmann La Roche | BI- AND TRICYCLIC SUBSTITUTED PHENYL-METHANONE AS INHIBITORS OF GLYCIN-I (GLYT-1) TRANSPORTERS FOR THE TREATMENT OF ALZHEIMER DISEASE |
| PE20061156A1 (en) | 2004-12-23 | 2006-12-16 | Glaxo Group Ltd | BENZAMIDE DERIVATIVES AS INHIBITING AGENTS OF THE GLYCINE TRANSPORTER |
| GB0428233D0 (en) * | 2004-12-23 | 2005-01-26 | Glaxo Group Ltd | Compounds |
| US7485637B2 (en) | 2005-01-04 | 2009-02-03 | Hoffmann-La Roche Inc. | Benzoyl-tetrahydropiperidine derivatives |
| BRPI0519744A2 (en) * | 2005-01-06 | 2009-03-10 | Hoffmann La Roche | sulfanyl-substituted phenyl methanones as glycine 1 (glyt-1) transporter inhibitors for the treatment of neurological and neuropsychiatric disorders |
| RU2396270C2 (en) * | 2005-01-07 | 2010-08-10 | Ф.Хоффманн-Ля Рош Аг | [4-(heteroaryl)piperazine-1-yl]-(2,5-substituted phenyl)methanone derivatives as glycine-1 (glyt-1) carrier inhibitors for treating neurologic and psychoneurological diseases |
| MX2007008616A (en) * | 2005-01-18 | 2007-09-11 | Hoffmann La Roche | 2, 5-disubstituted phenyl methanone derivatives as glycine transporter 1 (glyt-i) inhibitors for the treatment of neurological and neuropsychiatry disorders. |
| CN101146808B (en) | 2005-01-26 | 2011-10-12 | 弗·哈夫曼-拉罗切有限公司 | Phenyl methanone derivatives and their use as glycine transporter 1 inhibitors |
| SI1848694T1 (en) * | 2005-02-07 | 2010-01-29 | Hoffmann La Roche | Heterocyclic substituted phenyl methanones as inhibitors of the glycine transporter 1 |
| CN100341871C (en) * | 2005-06-03 | 2007-10-10 | 复旦大学 | Organic sulfur compound containing piperidine structure, its preparation and use |
| WO2007110449A1 (en) | 2006-03-29 | 2007-10-04 | Euro-Celtique S.A. | Benzenesulfonamide compounds and their use |
| WO2007118854A1 (en) | 2006-04-13 | 2007-10-25 | Euro-Celtique S.A. | Benzenesulfonamide compounds and the use thereof |
| TW200815353A (en) | 2006-04-13 | 2008-04-01 | Euro Celtique Sa | Benzenesulfonamide compounds and their use |
| EP2384768B1 (en) * | 2006-11-01 | 2013-08-21 | Purdue Pharma LP | Phenylpropionamide compounds and the use thereof |
| FR2910320B1 (en) * | 2006-12-21 | 2009-02-13 | Galderma Res & Dev S N C Snc | EMULSION COMPRISING AT LEAST ONE RETINOID AND BENZOLE PEROXIDE |
| FR2910321B1 (en) | 2006-12-21 | 2009-07-10 | Galderma Res & Dev S N C Snc | CREAM GEL COMPRISING AT LEAST ONE RETINOID AND BENZOLE PEROXIDE |
| US8399486B2 (en) | 2007-04-09 | 2013-03-19 | Purdue Pharma L.P. | Benzenesulfonyl compounds and the use thereof |
| US8765736B2 (en) | 2007-09-28 | 2014-07-01 | Purdue Pharma L.P. | Benzenesulfonamide compounds and the use thereof |
| US8258306B2 (en) * | 2007-12-12 | 2012-09-04 | Amgen Inc. | Glycine transporter-1 inhibitors |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4219559A (en) * | 1979-01-10 | 1980-08-26 | Janssen Pharmaceutica N.V. | N-Heterocyclyl-4-piperidinamines |
| CA1140119A (en) * | 1978-04-03 | 1983-01-25 | Joseph Torremans | N-heterocyclyl-4-piperidinamines |
| PH23995A (en) * | 1984-01-09 | 1990-02-09 | Janssen Pharmaceutica Nv | 4((bicycle heterocyclyl)-methyl and hetero)piperidines |
| US4695575A (en) * | 1984-11-13 | 1987-09-22 | Janssen Pharmaceutica, N.V. | 4-[(bicycle heterocyclyl)-methyl and -hetero]-piperidines |
| AU1041599A (en) * | 1997-11-13 | 1999-06-07 | Jose Luis Castro Pineiro | Therapeutic uses of triazolo-pyridazine derivatives |
-
1999
- 1999-02-26 PL PL99343435A patent/PL343435A1/en not_active Application Discontinuation
- 1999-02-26 IL IL13822899A patent/IL138228A0/en unknown
- 1999-02-26 JP JP2000534198A patent/JP2002505277A/en not_active Withdrawn
- 1999-02-26 HU HU0101048A patent/HUP0101048A2/en unknown
- 1999-02-26 EE EEP200000482A patent/EE200000482A/en unknown
- 1999-02-26 SK SK1308-2000A patent/SK13082000A3/en unknown
- 1999-02-26 BR BR9907951-8A patent/BR9907951A/en not_active Application Discontinuation
- 1999-02-26 WO PCT/EP1999/001309 patent/WO1999044596A2/en not_active Application Discontinuation
- 1999-02-26 CA CA002322164A patent/CA2322164A1/en not_active Abandoned
- 1999-02-26 CN CN998036471A patent/CN1292698A/en active Pending
- 1999-02-26 EP EP99915541A patent/EP1059922A2/en not_active Withdrawn
- 1999-02-26 KR KR1020007006315A patent/KR20010032968A/en not_active Application Discontinuation
- 1999-02-26 TR TR2000/02567T patent/TR200002567T2/en unknown
- 1999-02-26 AU AU34089/99A patent/AU3408999A/en not_active Abandoned
-
2000
- 2000-08-02 HR HR20000523A patent/HRP20000523A2/en not_active Application Discontinuation
- 2000-08-11 BG BG104685A patent/BG104685A/en unknown
- 2000-09-05 NO NO20004431A patent/NO20004431L/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| NO20004431L (en) | 2000-10-30 |
| WO1999044596A2 (en) | 1999-09-10 |
| EE200000482A (en) | 2002-02-15 |
| HUP0101048A2 (en) | 2001-10-28 |
| BG104685A (en) | 2001-04-30 |
| PL343435A1 (en) | 2001-08-13 |
| KR20010032968A (en) | 2001-04-25 |
| HRP20000523A2 (en) | 2001-02-28 |
| TR200002567T2 (en) | 2000-11-21 |
| EP1059922A2 (en) | 2000-12-20 |
| CN1292698A (en) | 2001-04-25 |
| WO1999044596A3 (en) | 2000-02-17 |
| NO20004431D0 (en) | 2000-09-05 |
| JP2002505277A (en) | 2002-02-19 |
| CA2322164A1 (en) | 1999-09-10 |
| AU3408999A (en) | 1999-09-20 |
| BR9907951A (en) | 2001-01-30 |
| SK13082000A3 (en) | 2001-03-12 |
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