IL105551A0 - Quinazolines and pharmaceutical compositions containing them - Google Patents

Quinazolines and pharmaceutical compositions containing them

Info

Publication number
IL105551A0
IL105551A0 IL105551A IL10555193A IL105551A0 IL 105551 A0 IL105551 A0 IL 105551A0 IL 105551 A IL105551 A IL 105551A IL 10555193 A IL10555193 A IL 10555193A IL 105551 A0 IL105551 A0 IL 105551A0
Authority
IL
Israel
Prior art keywords
quinazolines
pharmaceutical compositions
compositions containing
pharmaceutical
compositions
Prior art date
Application number
IL105551A
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of IL105551A0 publication Critical patent/IL105551A0/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • C07D239/80Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IL105551A 1992-05-07 1993-04-29 Quinazolines and pharmaceutical compositions containing them IL105551A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US88011992A 1992-05-07 1992-05-07
US99116492A 1992-12-16 1992-12-16

Publications (1)

Publication Number Publication Date
IL105551A0 true IL105551A0 (en) 1993-08-18

Family

ID=27128564

Family Applications (1)

Application Number Title Priority Date Filing Date
IL105551A IL105551A0 (en) 1992-05-07 1993-04-29 Quinazolines and pharmaceutical compositions containing them

Country Status (15)

Country Link
EP (2) EP0639184A1 (en)
JP (1) JPH0813805B2 (en)
KR (1) KR950701322A (en)
CN (1) CN1085550A (en)
AU (2) AU4220493A (en)
BG (1) BG99149A (en)
CA (1) CA2095194A1 (en)
CZ (1) CZ272494A3 (en)
FI (1) FI945199A0 (en)
HR (1) HRP930857A2 (en)
HU (1) HUT71401A (en)
IL (1) IL105551A0 (en)
MX (1) MX9302681A (en)
SI (1) SI9300244A (en)
WO (1) WO1993022292A1 (en)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2281297A (en) * 1993-08-27 1995-03-01 Merck & Co Inc Quinazoline compounds
US5434152A (en) * 1993-11-08 1995-07-18 Merck & Co., Inc. Asymmetric synthesis of (S)-(-)-6-chloro-4- cyclopropyl-3,4-dihydro-4-[(2-pyridyl)ethynyl]-2(1H)-quinazolinone
US6124302A (en) 1997-04-09 2000-09-26 Dupont Pharmaceuticals 4,4-disubstituted-3,4-dihydro-2(1H)-quinazolinones useful as HIV reverse transcriptase inhibitors
HRP980143A2 (en) * 1997-04-09 1999-02-28 Soo Sung Ko 4,4-disubstituted-3,4-dihydro-2 (1h)-quinazolinones useful as hiv reverse transcriptase inhibitors
EP1091939A1 (en) * 1998-06-30 2001-04-18 Du Pont Pharmaceuticals Company Substituted quinolin-2(1h)-ones useful as hiv reverse transcriptase inhibitors
CA2370141A1 (en) 1999-05-26 2000-12-07 James D. Rodgers 1,4-benzodiazepin-2-ones useful as hiv reverse transcriptase inhibitors
CA2377629A1 (en) * 2000-04-25 2001-11-08 Hae-Young Bae Biphenyl butyric acid derivative as a matrix metalloproteinase inhibitor
US7119111B2 (en) * 2002-05-29 2006-10-10 Amgen, Inc. 2-oxo-1,3,4-trihydroquinazolinyl derivatives and methods of use
ES2549084T3 (en) * 2007-10-05 2015-10-22 Msd K.K. Benzoxazinone derivatives
CN101544630B (en) * 2009-05-13 2013-03-13 中国科学院广州生物医药与健康研究院 Preparation method of hydroxylated indinavir
WO2017003724A1 (en) 2015-07-01 2017-01-05 Crinetics Pharmaceuticals, Inc. Somatostatin modulators and uses thereof
JOP20180009A1 (en) 2017-02-06 2019-01-30 Gilead Sciences Inc Hiv inhibitor compounds
WO2019023278A1 (en) 2017-07-25 2019-01-31 Crinetics Pharmaceuticals, Inc. Somatostatin modulators and uses thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL147140B (en) * 1968-11-26 1975-09-15 Farmaceutici Italia PROCEDURE FOR THE PREPARATION OF MEDICINAL PRODUCTS WITH AN INHIBITIVE ACTION ON THE CENTRAL NERVOUS SYSTEM.
IL102764A0 (en) * 1991-08-16 1993-01-31 Merck & Co Inc Quinazoline derivatives,and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
SI9300244A (en) 1993-12-31
HUT71401A (en) 1995-11-28
EP0639184A1 (en) 1995-02-22
CA2095194A1 (en) 1993-11-08
MX9302681A (en) 1994-05-31
CZ272494A3 (en) 1995-10-18
JPH069578A (en) 1994-01-18
JPH0813805B2 (en) 1996-02-14
FI945199A (en) 1994-11-04
FI945199A0 (en) 1994-11-04
AU3841393A (en) 1993-11-11
EP0569083A1 (en) 1993-11-10
WO1993022292A1 (en) 1993-11-11
HRP930857A2 (en) 1995-06-30
KR950701322A (en) 1995-03-23
CN1085550A (en) 1994-04-20
AU4220493A (en) 1993-11-29
BG99149A (en) 1995-06-30

Similar Documents

Publication Publication Date Title
IL105218A0 (en) Hexanones and pharmaceutical compositions containing them
IL105223A0 (en) Cyclohexane-ylidenes and pharmaceutical compositions containing them
IL105220A0 (en) Cyclohexanylidene compounds and pharmaceutical compositions containing them
IL105806A0 (en) Aminoquinoline derivatives and pharmaceutical compositions containing the same
IL106431A0 (en) Aminediol derivatives and pharmaceutical compositions containing the same
IL111221A0 (en) N-alkyl-n- arylpyrimidinamine derivatives and pharmaceutical compositions containing them
IL114622A0 (en) Heteroaryl-oxazolidinones and pharmaceutical compositions containing them
IL104824A0 (en) Heterobicyclic compounds and pharmaceutical compositions containing them
NZ314376A (en) Substituted sulphonamides and pharmaceutical compositions
NZ244766A (en) Bi-aromatic compounds and pharmaceutical compositions
GB9209078D0 (en) Pharmaceutical compositions
IL111518A (en) Isoquinolines their preparation and pharmaceutical compositions containing them
IL110988A0 (en) 4-arylamino-benzopyran derivatives and pharmaceutical compositions containing the same
IL106553A0 (en) Substituted imidazoles and pharmaceutical compositions containing them
IL106098A0 (en) Heteroarylnaphthalenes and pharmaceutical compositions containing them
IL97122A0 (en) Aromatase-inhibiting androstendiones and pharmaceutical compositions containing them
IL108073A0 (en) Substituted 6-azaandrostenones their preparation and pharmaceutical compositions containing them
IL105551A0 (en) Quinazolines and pharmaceutical compositions containing them
HUT65713A (en) Thienyl-pyrrolidinyl-carbapenem-derivatives providing antibiotic effect and pharmaceutical compositions containing it
IL104623A0 (en) Biphenyl-substituted quinoline derivatives and pharmaceutical compositions containing the same
IL107611A0 (en) Steroid compounds and pharmaceutical compositions containing them
GB9209874D0 (en) Pharmaceutical compositions
IL104944A0 (en) Anti-tumor agents and pharmaceutical compositions containing the same
IL111692A0 (en) Quinoxalines and pharmaceutical compositions containing them
GB9220143D0 (en) Compounds and compositions