IE780918L - 3, 5-disubstituted-1h-1, 2, 4-triazoles. - Google Patents
3, 5-disubstituted-1h-1, 2, 4-triazoles.Info
- Publication number
- IE780918L IE780918L IE780918A IE91878A IE780918L IE 780918 L IE780918 L IE 780918L IE 780918 A IE780918 A IE 780918A IE 91878 A IE91878 A IE 91878A IE 780918 L IE780918 L IE 780918L
- Authority
- IE
- Ireland
- Prior art keywords
- hydrogen
- alkyl
- fluoro
- chloro
- chosen
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
The 3,5-disubstitited-1H-1,2,4-triazoles <IMAGE> in which: R is chosen from: hydrogen, (C1-4)alkyl, (C1-4)alkoxy, allyloxy, propargyloxy, trifluoromethyl, phenyl, fluoro, chloro and dimethylamino; R1 represents a (C1-4)alkyl group; R2 is chosen from: hydrogen, fluoro, chloro, (C1-4)alkyl, methoxy and ethoxy; R3 is chosen from: hydrogen, fluoro, chloro, (C1-4)alkyl and (C1-4)alkoxy; R and R3, taken together, represent a methylenedioxy group; on condition that, when R, R2 and R3 simultaneously represent hydrogen, R1 is not the methyl group; and also on condition that, when R2 and one of the groups R and R3 represent hydrogen, R1 and the other of the groups R and R3 are not simultaneously the methyl group; and their salts obtained with pharmaceutically acceptable acids are described. These compounds have antireproductive properties and act on the central nervous system.
[GB1579352A]
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB19012/77A GB1579352A (en) | 1977-05-06 | 1977-05-06 | 3,5-disubstituted-1h-1,2,4-triazoles |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IE780918L true IE780918L (en) | 1978-11-06 |
| IE46821B1 IE46821B1 (en) | 1983-10-05 |
Family
ID=10122292
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IE918/78A IE46821B1 (en) | 1977-05-06 | 1978-05-05 | 3,5-disubstituted-1h-1,2,4-triazoles |
Country Status (26)
| Country | Link |
|---|---|
| JP (1) | JPS53137965A (en) |
| AT (1) | AT360530B (en) |
| AU (1) | AU520348B2 (en) |
| BE (1) | BE866728A (en) |
| CA (1) | CA1100511A (en) |
| CH (1) | CH630909A5 (en) |
| DE (1) | DE2819372A1 (en) |
| DK (1) | DK149469C (en) |
| ES (1) | ES469482A1 (en) |
| FI (1) | FI64150C (en) |
| FR (1) | FR2389615B1 (en) |
| GB (1) | GB1579352A (en) |
| GR (1) | GR66126B (en) |
| HK (1) | HK26281A (en) |
| IE (1) | IE46821B1 (en) |
| IL (1) | IL54517A (en) |
| IT (1) | IT1158700B (en) |
| LU (1) | LU79601A1 (en) |
| NL (1) | NL7804211A (en) |
| NO (2) | NO148525C (en) |
| NZ (1) | NZ187181A (en) |
| PH (1) | PH15364A (en) |
| PT (1) | PT68005B (en) |
| SE (1) | SE444316B (en) |
| YU (1) | YU41311B (en) |
| ZA (1) | ZA782118B (en) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0011129B1 (en) * | 1978-10-30 | 1981-11-11 | Gruppo Lepetit S.P.A. | New 1,2,4-triazole derivatives, a process for their manufacture and pharmaceutical compositions containing them |
| DE3173083D1 (en) * | 1980-03-22 | 1986-01-16 | Fbc Ltd | Pesticidal heterocyclic compounds, processes for preparing them, compositions containing them, and their use |
| AU557034B2 (en) * | 1981-10-20 | 1986-12-04 | Gruppo Lepetit S.P.A. | 3,5-diphenyl-1h-1,2,4-trazoles with contragestational |
| US5017386A (en) * | 1989-10-05 | 1991-05-21 | University Of Kentucky Research Foundation | Method of reducing odor associated with hexanal production in plant products |
| WO1995033732A1 (en) * | 1994-06-09 | 1995-12-14 | Nippon Soda Co., Ltd. | Triazole compound, production process, and pest control agent |
| IT1292092B1 (en) * | 1997-06-05 | 1999-01-25 | Geange Ltd | USE OF NITROGEN AROMATIC HETEROCYCLIC DERIVATIVES IN THE TOPICAL TREATMENT OF EPITHELIAL TISSUES |
| PT1070708E (en) * | 1999-07-21 | 2004-05-31 | Hoffmann La Roche | TRIAZOL DERIVATIVES |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SU508198A3 (en) * | 1971-07-22 | 1976-03-25 | Группо Лепетит С.П.А. (Фирма) | Method for preparing 1,2,4-triazole derivatives |
| JPS5241264B2 (en) * | 1973-05-21 | 1977-10-17 | ||
| JPS5082066A (en) * | 1973-10-30 | 1975-07-03 | ||
| AU497898B2 (en) * | 1975-01-10 | 1979-01-18 | Commonwealth Scientific And Industrial Research Organisation | Plant growth regulating method and composition for use therein |
-
1977
- 1977-05-06 GB GB19012/77A patent/GB1579352A/en not_active Expired
-
1978
- 1978-04-07 GR GR55921A patent/GR66126B/el unknown
- 1978-04-12 ZA ZA00782118A patent/ZA782118B/en unknown
- 1978-04-17 IL IL54517A patent/IL54517A/en unknown
- 1978-04-17 AU AU35140/78A patent/AU520348B2/en not_active Expired
- 1978-04-20 NL NL7804211A patent/NL7804211A/en not_active Application Discontinuation
- 1978-04-25 DK DK178978A patent/DK149469C/en not_active IP Right Cessation
- 1978-04-26 YU YU1036/78A patent/YU41311B/en unknown
- 1978-04-28 FI FI781339A patent/FI64150C/en not_active IP Right Cessation
- 1978-05-02 JP JP5324478A patent/JPS53137965A/en active Granted
- 1978-05-02 AT AT315678A patent/AT360530B/en not_active IP Right Cessation
- 1978-05-03 IT IT22928/78A patent/IT1158700B/en active
- 1978-05-03 NO NO781560A patent/NO148525C/en unknown
- 1978-05-03 CH CH483478A patent/CH630909A5/en not_active IP Right Cessation
- 1978-05-03 DE DE19782819372 patent/DE2819372A1/en active Granted
- 1978-05-03 FR FR7813205A patent/FR2389615B1/fr not_active Expired
- 1978-05-05 IE IE918/78A patent/IE46821B1/en unknown
- 1978-05-05 LU LU79601A patent/LU79601A1/en unknown
- 1978-05-05 PT PT68005A patent/PT68005B/en unknown
- 1978-05-05 SE SE7805184A patent/SE444316B/en not_active IP Right Cessation
- 1978-05-05 ES ES469482A patent/ES469482A1/en not_active Expired
- 1978-05-05 CA CA302,712A patent/CA1100511A/en not_active Expired
- 1978-05-05 NZ NZ187181A patent/NZ187181A/en unknown
- 1978-05-05 BE BE187412A patent/BE866728A/en not_active IP Right Cessation
-
1979
- 1979-06-01 PH PH22600A patent/PH15364A/en unknown
-
1981
- 1981-06-18 HK HK262/81A patent/HK26281A/en unknown
-
1982
- 1982-11-03 NO NO823654A patent/NO823654L/en unknown
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