IE41223L - 1, 3-disubstituted indoles - Google Patents
1, 3-disubstituted indolesInfo
- Publication number
- IE41223L IE41223L IE750695A IE69575A IE41223L IE 41223 L IE41223 L IE 41223L IE 750695 A IE750695 A IE 750695A IE 69575 A IE69575 A IE 69575A IE 41223 L IE41223 L IE 41223L
- Authority
- IE
- Ireland
- Prior art keywords
- alkyl
- acyl
- march
- compound
- tertiary
- Prior art date
Links
- -1 1, 3-disubstituted indoles Chemical class 0.000 title 1
- 125000004103 aminoalkyl group Chemical group 0.000 abstract 3
- 125000002252 acyl group Chemical group 0.000 abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- HTSGKJQDMSTCGS-UHFFFAOYSA-N 1,4-bis(4-chlorophenyl)-2-(4-methylphenyl)sulfonylbutane-1,4-dione Chemical compound C1=CC(C)=CC=C1S(=O)(=O)C(C(=O)C=1C=CC(Cl)=CC=1)CC(=O)C1=CC=C(Cl)C=C1 HTSGKJQDMSTCGS-UHFFFAOYSA-N 0.000 abstract 1
- 230000002152 alkylating effect Effects 0.000 abstract 1
- 230000001430 anti-depressive effect Effects 0.000 abstract 1
- 230000000845 anti-microbial effect Effects 0.000 abstract 1
- 239000000935 antidepressant agent Substances 0.000 abstract 1
- 229940005513 antidepressants Drugs 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 150000002475 indoles Chemical class 0.000 abstract 1
- 238000007911 parenteral administration Methods 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/16—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms condensed with carbocyclic rings or ring systems
- C07D249/18—Benzotriazoles
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Psychiatry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pain & Pain Management (AREA)
- Indole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
1502821 Indoles SIEGFRIED AG 26 March 1975 [29 March 1974] 12785/75 Heading C2C Novel compounds I in which R 1 is H, alkyl or tertiary aminoalkyl, R 2 is tertiary amino-alkyl or acyl and each of R 3 and R 4 is H or a substituent, are prepared by reacting a compound II in which R is H, acyl, alkyl or tertiary aminoalkyl, with an appropriate alkylating or acylating agent. Pharmaceutical compositions having antimicrobial and antidepressant activity, for oral or parenteral administration, comprise a compound I and a carrier.
[GB1502821A]
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH439974A CH603581A5 (en) | 1974-03-29 | 1974-03-29 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IE41223L true IE41223L (en) | 1975-09-29 |
| IE41223B1 IE41223B1 (en) | 1979-11-21 |
Family
ID=4275407
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IE695/75A IE41223B1 (en) | 1974-03-29 | 1975-03-27 | Hydrazine derivatives having pharmacological activity |
Country Status (15)
| Country | Link |
|---|---|
| JP (1) | JPS6036423B2 (en) |
| AT (1) | AT346840B (en) |
| BE (1) | BE827399A (en) |
| CA (1) | CA1054601A (en) |
| CH (1) | CH603581A5 (en) |
| DE (1) | DE2512702C2 (en) |
| DK (1) | DK133175A (en) |
| ES (1) | ES435944A1 (en) |
| FR (1) | FR2265365B1 (en) |
| GB (1) | GB1502821A (en) |
| IE (1) | IE41223B1 (en) |
| LU (1) | LU72170A1 (en) |
| NL (1) | NL7502722A (en) |
| SE (1) | SE409113B (en) |
| ZA (1) | ZA752001B (en) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1113879B (en) * | 1979-03-15 | 1986-01-27 | Farmatis Spa | ISOINDOLINE DERIVATIVE, PROCESS FOR ITS PREPARATION AND THERAPEUTIC COMPOSITIONS THAT INCLUDE IT AS AN ACTIVE PRINCIPLE |
| DE3022097A1 (en) * | 1980-06-12 | 1981-12-24 | Siegfried AG, Zofingen | 1-AMINO-3-PHENYL INDOLES AND THEIR USE |
| DE3852335T2 (en) * | 1987-04-24 | 1995-05-11 | Hoechst Roussel Pharma | N- (Pyridinyl) -1H-indol-1-amines, process for their preparation and their use as medicaments. |
-
1974
- 1974-03-29 CH CH439974A patent/CH603581A5/xx not_active IP Right Cessation
-
1975
- 1975-03-07 NL NL7502722A patent/NL7502722A/en not_active Application Discontinuation
- 1975-03-19 FR FR7508545A patent/FR2265365B1/fr not_active Expired
- 1975-03-21 CA CA223211A patent/CA1054601A/en not_active Expired
- 1975-03-22 DE DE2512702A patent/DE2512702C2/en not_active Expired
- 1975-03-24 ES ES435944A patent/ES435944A1/en not_active Expired
- 1975-03-25 AT AT226975A patent/AT346840B/en not_active IP Right Cessation
- 1975-03-26 DK DK133175A patent/DK133175A/da not_active Application Discontinuation
- 1975-03-26 GB GB12785/75A patent/GB1502821A/en not_active Expired
- 1975-03-26 SE SE7503533-7A patent/SE409113B/en not_active IP Right Cessation
- 1975-03-27 IE IE695/75A patent/IE41223B1/en unknown
- 1975-03-28 BE BE154965A patent/BE827399A/en not_active IP Right Cessation
- 1975-03-28 JP JP50037014A patent/JPS6036423B2/en not_active Expired
- 1975-03-28 LU LU72170A patent/LU72170A1/xx unknown
- 1975-04-01 ZA ZA00752001A patent/ZA752001B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JPS6036423B2 (en) | 1985-08-20 |
| SE7503533L (en) | 1975-09-30 |
| ZA752001B (en) | 1976-02-25 |
| DE2512702C2 (en) | 1982-09-23 |
| CH603581A5 (en) | 1978-08-31 |
| GB1502821A (en) | 1978-03-01 |
| DK133175A (en) | 1975-09-30 |
| IE41223B1 (en) | 1979-11-21 |
| AT346840B (en) | 1978-11-27 |
| NL7502722A (en) | 1975-10-01 |
| FR2265365B1 (en) | 1978-07-28 |
| JPS50130758A (en) | 1975-10-16 |
| SE409113B (en) | 1979-07-30 |
| FR2265365A1 (en) | 1975-10-24 |
| ATA226975A (en) | 1978-04-15 |
| CA1054601A (en) | 1979-05-15 |
| DE2512702A1 (en) | 1975-10-09 |
| BE827399A (en) | 1975-09-29 |
| LU72170A1 (en) | 1976-02-04 |
| ES435944A1 (en) | 1976-12-16 |
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