HUT57730A - Process for producing isomer-free4-hydroxy-7-chloroquinoline
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Process for producing isomer-free4-hydroxy-7-chloroquinoline
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Publication number
HUT57730A
HUT57730AHU903314AHU331490AHUT57730AHU T57730 AHUT57730 AHU T57730AHU 903314 AHU903314 AHU 903314AHU 331490 AHU331490 AHU 331490AHU T57730 AHUT57730 AHU T57730A
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Application filed by Alkaloida Vegyeszeti GyarfiledCriticalAlkaloida Vegyeszeti Gyar
Priority to HU903314ApriorityCriticalpatent/HU205907B/en
Publication of HU903314D0publicationCriticalpatent/HU903314D0/en
Publication of HUT57730ApublicationCriticalpatent/HUT57730A/en
Publication of HU205907BpublicationCriticalpatent/HU205907B/en
Organic Low-Molecular-Weight Compounds And Preparation Thereof
(AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts
(AREA)
Abstract
4-hydroxy-7-chloro-quinoline of general formula (I) is prepd. free of isomers at 60-130 deg. C temp. and 0.1-0.6 MPa pressure from di: or tri:-ethyl-malonate, tri:ethyl-or tri:methyl-o-formate and 3-chloro-aniline, in the presence of metallic magnesium or of magnesium-oxide hydroxide or carbonate and/or unsubstd. chloro-aniline-, or 1-4C alkyl gp. (identical or dissimilar) substd. ammonium-chloride as catalyst. 2-carbomethoxy-3-(3-chloro-anilino)- methyl-acrylate (VI) is obtd. and is converted to cyclic quinoline-3-carboxylic-ester (II) at 180-280 deg. C in an inert solvent R:methyl gp. in (II). The prod. is hydrolysed and is decarboxylated thermally to cpd.(I). (1pp Dwg.No.0/0)
HU903314A1990-05-041990-05-04Process for producing 4-hidroxy-7-chloro-quinoline
HU205907B
(en)