HUP0203412A2 - Kinazolinszármazékok és azok alkalmazása az AKT protein kináz rendszer aktiválására és/vagy az NFKB transzkripciós faktor gátlására alkalmas gyógyászati készítmény előállítására - Google Patents

Kinazolinszármazékok és azok alkalmazása az AKT protein kináz rendszer aktiválására és/vagy az NFKB transzkripciós faktor gátlására alkalmas gyógyászati készítmény előállítására

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Publication number
HUP0203412A2
HUP0203412A2 HU0203412A HUP0203412A HUP0203412A2 HU P0203412 A2 HUP0203412 A2 HU P0203412A2 HU 0203412 A HU0203412 A HU 0203412A HU P0203412 A HUP0203412 A HU P0203412A HU P0203412 A2 HUP0203412 A2 HU P0203412A2
Authority
HU
Hungary
Prior art keywords
protein kinase
transcription factor
inhibition
activation
production
Prior art date
Application number
HU0203412A
Other languages
English (en)
Inventor
Balázs Sümegi
Ferenc Gallyas
Tamás Lóránd
Balázs Veres
Original Assignee
Balázs Sümegi
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Balázs Sümegi filed Critical Balázs Sümegi
Priority to HU0203412A priority Critical patent/HUP0203412A3/hu
Publication of HU0203412D0 publication Critical patent/HU0203412D0/hu
Publication of HUP0203412A2 publication Critical patent/HUP0203412A2/hu
Publication of HUP0203412A3 publication Critical patent/HUP0203412A3/hu

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Abstract

57) A találmány tárgyát az (I) általános képletű kinazolinszármazékokalkalmazása képezi - a képletben R jelentése hidrogénatom vagy -SR1általános képletű csoport, ahol R1 jelentése hidrogénatom, C1-8 alkil-vagy C6-18 arilcsoport - az Akt protein kináz rendszer aktiválásáraés/vagy az NFkB transzkripciós faktor gátlására alkalmas gyógyászatikészítmény előállítására. A találmány tárgyát képezik továbbá a fentivegyületek közül az (la) általános képlettel jellemezhető újkinazolinszármazékok, ahol a képletben R2 jelentése C1-8 alkil- vagyC6-18 arilcsoport, és az új vegyületeket tartalmazó gyógyászatikészítmények. Ó
HU0203412A 2002-10-09 2002-10-09 Quinazoline derivatives and their use for the production of pharmaceutical composition for activation of akt protein kinase and/or inhibition of nfkb transcription factor HUP0203412A3 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
HU0203412A HUP0203412A3 (en) 2002-10-09 2002-10-09 Quinazoline derivatives and their use for the production of pharmaceutical composition for activation of akt protein kinase and/or inhibition of nfkb transcription factor

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU0203412A HUP0203412A3 (en) 2002-10-09 2002-10-09 Quinazoline derivatives and their use for the production of pharmaceutical composition for activation of akt protein kinase and/or inhibition of nfkb transcription factor

Publications (3)

Publication Number Publication Date
HU0203412D0 HU0203412D0 (en) 2002-12-28
HUP0203412A2 true HUP0203412A2 (hu) 2004-06-28
HUP0203412A3 HUP0203412A3 (en) 2005-01-28

Family

ID=89980848

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0203412A HUP0203412A3 (en) 2002-10-09 2002-10-09 Quinazoline derivatives and their use for the production of pharmaceutical composition for activation of akt protein kinase and/or inhibition of nfkb transcription factor

Country Status (1)

Country Link
HU (1) HUP0203412A3 (hu)

Also Published As

Publication number Publication date
HUP0203412A3 (en) 2005-01-28
HU0203412D0 (en) 2002-12-28

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FD9A Lapse of provisional protection due to non-payment of fees