HU197929B - Process for producing vasopressin-antagonist compounds of cyclic desproline-vasopressin and pharmaceutical compositions comprising these compounds - Google Patents

Process for producing vasopressin-antagonist compounds of cyclic desproline-vasopressin and pharmaceutical compositions comprising these compounds Download PDF

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Publication number
HU197929B
HU197929B HU85849A HU84985A HU197929B HU 197929 B HU197929 B HU 197929B HU 85849 A HU85849 A HU 85849A HU 84985 A HU84985 A HU 84985A HU 197929 B HU197929 B HU 197929B
Authority
HU
Hungary
Prior art keywords
formula
tyr
arg
compound
preparation
Prior art date
Application number
HU85849A
Other languages
English (en)
Hungarian (hu)
Other versions
HUT37807A (en
Inventor
Fadia E Ali
William F Huffman
Original Assignee
Smithkline Beckman Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/586,934 external-priority patent/US4481194A/en
Priority claimed from US06/586,933 external-priority patent/US4481193A/en
Application filed by Smithkline Beckman Corp filed Critical Smithkline Beckman Corp
Publication of HUT37807A publication Critical patent/HUT37807A/hu
Publication of HU197929B publication Critical patent/HU197929B/hu

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/16—Oxytocins; Vasopressins; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Noodles (AREA)
HU85849A 1984-03-07 1985-03-06 Process for producing vasopressin-antagonist compounds of cyclic desproline-vasopressin and pharmaceutical compositions comprising these compounds HU197929B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/586,934 US4481194A (en) 1984-03-07 1984-03-07 Des-proline-des-glycine vasopressin antagonists
US06/586,933 US4481193A (en) 1984-03-07 1984-03-07 Des-proline vasopressin antagonists

Publications (2)

Publication Number Publication Date
HUT37807A HUT37807A (en) 1986-02-28
HU197929B true HU197929B (en) 1989-06-28

Family

ID=27079864

Family Applications (1)

Application Number Title Priority Date Filing Date
HU85849A HU197929B (en) 1984-03-07 1985-03-06 Process for producing vasopressin-antagonist compounds of cyclic desproline-vasopressin and pharmaceutical compositions comprising these compounds

Country Status (15)

Country Link
EP (1) EP0154544A3 (cg-RX-API-DMAC7.html)
AU (1) AU573788B2 (cg-RX-API-DMAC7.html)
CA (1) CA1249397A (cg-RX-API-DMAC7.html)
DK (1) DK98585A (cg-RX-API-DMAC7.html)
ES (1) ES8608539A1 (cg-RX-API-DMAC7.html)
FI (1) FI850894L (cg-RX-API-DMAC7.html)
GR (1) GR850543B (cg-RX-API-DMAC7.html)
HU (1) HU197929B (cg-RX-API-DMAC7.html)
IL (1) IL74483A (cg-RX-API-DMAC7.html)
JO (1) JO1362B1 (cg-RX-API-DMAC7.html)
NO (1) NO850895L (cg-RX-API-DMAC7.html)
NZ (1) NZ211274A (cg-RX-API-DMAC7.html)
PH (1) PH21037A (cg-RX-API-DMAC7.html)
PT (1) PT80054B (cg-RX-API-DMAC7.html)
ZW (1) ZW3585A1 (cg-RX-API-DMAC7.html)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT83455B (en) * 1985-10-02 1988-10-20 Smithkline Beckman Corp Vasopressin compounds
US4687758A (en) * 1985-11-19 1987-08-18 Smithkline Beckman Corporation Des-proline-N-methylarginine vasopressins
PT84342B (pt) * 1986-02-25 1989-09-14 Smithkline Beecham Corp Processo de preparacao de compostos de vasopressina

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE399252B (sv) * 1976-05-24 1978-02-06 Ferring Ab Forfarande for framstellnign av antidiuretiskt verkande desamino-asparagin Ÿ4-d-argininŸ8-vasopressin
SE407682B (sv) * 1976-11-12 1979-04-09 Ferring Ab Forfarande for framstellning av antidiuretiskt verkande desamino-d-argininÿ8-vasopressinderivat
DK81082A (da) * 1981-03-06 1982-09-07 Sandoz Ag Fremgangsmaade til fremstilling af polypeptider
US4367225A (en) * 1981-03-24 1983-01-04 The Medical College Of Ohio Novel antagonists of the antidiuretic and/or vasopressor action of arginine vasopressin
US4399125A (en) * 1981-03-24 1983-08-16 Maurice Manning Novel antagonists of the antidiuretic action of arginine vasopressin
DK153883A (da) * 1982-04-20 1983-10-21 Ceskoslovenska Akademie Ved Vasopressin-analoge

Also Published As

Publication number Publication date
JO1362B1 (en) 1986-11-30
PT80054B (en) 1987-04-07
PT80054A (en) 1985-04-01
IL74483A (en) 1991-07-18
PH21037A (en) 1987-06-30
NO850895L (no) 1985-09-09
HUT37807A (en) 1986-02-28
IL74483A0 (en) 1985-06-30
EP0154544A2 (en) 1985-09-11
FI850894A7 (fi) 1985-09-08
EP0154544A3 (en) 1988-10-05
AU3951485A (en) 1985-10-10
FI850894L (fi) 1985-09-08
DK98585D0 (da) 1985-03-04
AU573788B2 (en) 1988-06-23
ES540922A0 (es) 1986-06-16
GR850543B (cg-RX-API-DMAC7.html) 1985-07-05
DK98585A (da) 1985-09-08
ES8608539A1 (es) 1986-06-16
NZ211274A (en) 1988-06-30
ZW3585A1 (en) 1985-05-29
FI850894A0 (fi) 1985-03-06
CA1249397A (en) 1989-01-24

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Legal Events

Date Code Title Description
HU90 Patent valid on 900628
HMM4 Cancellation of final prot. due to non-payment of fee